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ABCC2

receptor: PXRTier 1

Drug substrates

methotrexate; pravastatin; cisplatin; conjugated bilirubin

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of ABCC2 expression, diminishing canalicular efflux capacity and reducing the clearance of clearance-dependent substrates.

Affected substrate drugs (PharmGKB): tenofovir; methotrexate; mycophenolic acid; talinolol; lopinavir; tacrolimus

Scored variants near ABCC2

chr10:99,682,639..99,952,594, gene body plus 100 kb. Showing the strongest 200 by effect size.

VariantPosition PXR FXR AhR AF
chr10_99732714_A_Gchr10:9973271460,73610,78425,216—   
chr10_99732715_T_Cchr10:9973271544,5447,58420,352—   
chr10_99696002_A_Tchr10:9969600244,28818,72046,656—   
chr10_99695953_T_Cchr10:9969595326,3369,63222,848—   
chr10_99732718_C_Tchr10:9973271818,6242,4323,328—   
chr10_99732709_C_Achr10:9973270917,9842,9125,120—   
chr10_99732687_T_Gchr10:9973268715,0402,6889,984—   
chr10_99695943_T_Cchr10:9969594314,4006,24016,064—   
chr10_99696004_G_Tchr10:9969600412,4166,24014,272—   
chr10_99696019_C_Gchr10:99696019-11,936-5,504-12,800—   
chr10_99695951_T_Achr10:9969595111,5204,57611,840—   
chr10_99696019_C_Achr10:99696019-10,432-4,576-11,008—   
chr10_99732699_C_Tchr10:9973269910,3041,7284,864—   
chr10_99732708_A_Cchr10:99732708-9,920-1,024-6,528—   
chr10_99695989_A_Cchr10:996959899,8563,87212,032—   
chr10_99732727_C_Gchr10:997327279,8561,3444,864—   
chr10_99732704_C_Achr10:99732704-9,344-1,440-6,912—   
chr10_99732706_A_Cchr10:99732706-9,216-1,408-4,480—   
chr10_99696019_C_Tchr10:99696019-8,864-4,096-9,728—   
chr10_99732725_G_Cchr10:99732725-8,768-1,536-9,472—   
chr10_99732704_C_Tchr10:99732704-8,704-864-5,376—   
chr10_99732703_G_Cchr10:99732703-8,256-1,632-4,224—   
chr10_99732704_C_Gchr10:99732704-8,064-928-3,456—   
chr10_99732692_T_Cchr10:99732692-7,872-1,568-6,144—   
chr10_99696022_G_Cchr10:99696022-7,584-3,456-9,472—   
chr10_99695969_A_Tchr10:99695969-7,456-3,488-10,048—   
chr10_99732692_T_Gchr10:99732692-7,168-1,760-6,528—   
chr10_99732566_G_Achr10:99732566-7,040-1,088-6,656—   
chr10_99695969_A_Cchr10:99695969-6,976-3,264-7,872—   
chr10_99732555_T_Achr10:997325556,9122561,792—   
chr10_99732627_G_Achr10:997326276,9121,1202561.3e-5
chr10_99695946_T_Cchr10:996959466,8163,1366,9127.2e-5
chr10_99732625_T_Cchr10:997326256,784-544-2,816—   
chr10_99696024_G_Cchr10:99696024-6,720-3,136-7,872—   
chr10_99732567_A_Cchr10:997325676,6561,1848,192—   
chr10_99732710_G_Achr10:99732710-6,528-1,024-7,296—   
chr10_99732708_A_Tchr10:99732708-6,528-576-4,992—   
chr10_99695951_T_Cchr10:996959516,4962,6248,128—   
chr10_99696022_G_Achr10:99696022-6,496-3,104-7,232—   
chr10_99696024_G_Achr10:99696024-6,464-3,008-7,936—   
chr10_99695965_G_Cchr10:99695965-6,400-3,104-8,384—   
chr10_99696021_C_Gchr10:99696021-6,400-2,816-8,192—   
chr10_99695982_T_Achr10:996959826,4002,9125,952—   
chr10_99732711_A_Gchr10:997327116,4001,1204,352—   
chr10_99732718_C_Gchr10:99732718-6,400-1,056-2,944—   
chr10_99696021_C_Tchr10:99696021-6,208-2,944-6,7202.6e-5
chr10_99732712_G_Achr10:99732712-6,208-672-5,888—   
chr10_99732674_G_Cchr10:997326746,1441,8565,120—   
chr10_99732706_A_Tchr10:99732706-6,144-704-3,072—   
chr10_99696022_G_Tchr10:99696022-6,112-2,944-7,616—   
chr10_99696021_C_Achr10:99696021-6,016-2,656-7,168—   
chr10_99732708_A_Gchr10:99732708-6,016-320-2,688—   
chr10_99696020_A_Gchr10:99696020-5,984-3,104-6,336—   
chr10_99695967_C_Gchr10:99695967-5,856-2,560-7,424—   
chr10_99696025_T_Gchr10:996960255,8242,5606,592—   
chr10_99696023_T_Cchr10:99696023-5,824-2,784-4,2246.6e-6
chr10_99695965_G_Achr10:99695965-5,760-2,784-8,320—   
chr10_99696027_C_Tchr10:99696027-5,760-2,528-6,720—   
chr10_99695965_G_Tchr10:99695965-5,728-2,624-7,744—   
chr10_99696032_T_Gchr10:996960325,7282,7846,592—   
chr10_99696009_A_Tchr10:99696009-5,728-2,624-6,464—   
chr10_99695981_C_Gchr10:99695981-5,728-1,632-3,776—   
chr10_99695948_T_Cchr10:996959485,6962,9448,384—   
chr10_99732705_C_Achr10:99732705-5,696-832-4,224—   
chr10_99695973_C_Gchr10:99695973-5,664-2,656-6,208—   
chr10_99732689_A_Tchr10:99732689-5,632-1,792-4,864—   
chr10_99732701_T_Achr10:99732701-5,568-992-4,736—   
chr10_99732683_A_Cchr10:997326835,5043,04012,416—   
chr10_99732692_T_Achr10:99732692-5,504-1,408-7,936—   
chr10_99695963_C_Achr10:99695963-5,504-2,400-6,464—   
chr10_99732727_C_Achr10:997327275,5048641,920—   
chr10_99695905_A_Gchr10:996959055,4721,8886,784—   
chr10_99732684_G_Tchr10:99732684-5,440-1,376-6,144—   
chr10_99732710_G_Cchr10:99732710-5,440-320-4,608—   
chr10_99695967_C_Achr10:99695967-5,376-2,432-7,168—   
chr10_99696011_A_Cchr10:99696011-5,376-2,400-5,248—   
chr10_99732629_G_Achr10:997326295,3761,3442,560—   
chr10_99732707_C_Achr10:99732707-5,312-896-7,296—   
chr10_99732717_C_Gchr10:99732717-5,3120-128—   
chr10_99695981_C_Achr10:99695981-5,280-1,888-5,184—   
chr10_99696023_T_Gchr10:99696023-5,248-2,336-5,4406.6e-6
chr10_99732640_C_Achr10:997326405,2483,3924,864—   
chr10_99732699_C_Achr10:997326995,2487361,920—   
chr10_99732705_C_Gchr10:99732705-5,248-928-4,224—   
chr10_99695967_C_Tchr10:99695967-5,216-2,592-6,976—   
chr10_99696032_T_Achr10:996960325,2162,4644,928—   
chr10_99696024_G_Tchr10:99696024-5,184-2,336-4,992—   
chr10_99696027_C_Gchr10:99696027-5,184-2,240-4,928—   
chr10_99732703_G_Tchr10:99732703-5,184-1,248-4,7366.6e-6
chr10_99695994_G_Tchr10:996959945,1201,8245,248—   
chr10_99732558_A_Tchr10:997325585,1208324,864—   
chr10_99732709_C_Gchr10:99732709-5,120-768-4,352—   
chr10_99696034_T_Achr10:99696034-5,088-2,368-6,400—   
chr10_99732688_C_Achr10:99732688-5,056-992-3,584—   
chr10_99695968_A_Gchr10:99695968-4,992-2,464-6,528—   
chr10_99732724_C_Tchr10:99732724-4,992-736-2,8166.6e-6
chr10_99732710_G_Tchr10:99732710-4,928-224-4,480—   
chr10_99695964_T_Cchr10:99695964-4,864-2,048-5,248—   
chr10_99732567_A_Tchr10:997325674,8641,1523,584—   
chr10_99732712_G_Cchr10:99732712-4,8640-2,048—   
chr10_99695972_T_Cchr10:99695972-4,800-2,144-5,632—   
chr10_99695957_A_Tchr10:996959574,7681,7923,264—   
chr10_99695981_C_Tchr10:99695981-4,736-1,920-5,760—   
chr10_99696020_A_Cchr10:99696020-4,704-2,560-5,952—   
chr10_99696010_C_Gchr10:99696010-4,672-2,080-5,184—   
chr10_99732619_C_Achr10:997326194,608672256—   
chr10_99695968_A_Tchr10:99695968-4,576-2,432-6,912—   
chr10_99695966_C_Tchr10:99695966-4,544-2,240-6,272—   
chr10_99696009_A_Cchr10:99696009-4,480-2,176-5,312—   
chr10_99696009_A_Gchr10:99696009-4,480-2,176-5,120—   
chr10_99732583_G_Tchr10:997325834,4807044,608—   
chr10_99732719_A_Gchr10:99732719-4,480-1,216-2,1766.6e-6
chr10_99695966_C_Achr10:99695966-4,448-2,144-5,888—   
chr10_99695979_G_Tchr10:99695979-4,416-1,760-4,928—   
chr10_99695977_C_Achr10:99695977-4,384-1,888-6,528—   
chr10_99732707_C_Tchr10:99732707-4,352-448-4,4802.6e-4
chr10_99732536_A_Gchr10:997325364,352-642,3046.6e-6
chr10_99732593_T_Gchr10:99732593-4,352-544256—   
chr10_99732624_T_Gchr10:997326244,352-320-4,096—   
chr10_99696003_T_Cchr10:996960034,2881,9845,376—   
chr10_99695971_A_Cchr10:99695971-4,288-1,824-3,520—   
chr10_99696020_A_Tchr10:99696020-4,256-2,272-5,440—   
chr10_99696018_A_Tchr10:996960184,2562,0165,312—   
chr10_99695932_T_Gchr10:996959324,2561,5684,480—   
chr10_99732573_A_Gchr10:99732573-4,224-1,248-3,840—   
chr10_99732717_C_Tchr10:99732717-4,224-384-3,0722.6e-5
chr10_99696033_T_Achr10:99696033-4,192-1,792-4,928—   
chr10_99695968_A_Cchr10:99695968-4,160-2,144-5,248—   
chr10_99732690_C_Tchr10:99732690-4,160-896-2,304—   
chr10_99696017_A_Cchr10:99696017-4,096-2,144-3,904—   
chr10_99696027_C_Achr10:99696027-4,096-1,568-3,328—   
chr10_99696016_G_Tchr10:99696016-4,064-1,920-4,480—   
chr10_99732707_C_Gchr10:99732707-3,968-928-5,120—   
chr10_99695998_T_Achr10:996959983,9361,9844,544—   
chr10_99695989_A_Tchr10:99695989-3,872-1,536-4,992—   
chr10_99732537_C_Tchr10:99732537-3,840-608-6,912—   
chr10_99696025_T_Achr10:996960253,8401,9525,312—   
chr10_99695977_C_Gchr10:99695977-3,808-1,536-4,864—   
chr10_99695964_T_Gchr10:99695964-3,776-1,600-4,160—   
chr10_99732577_C_Gchr10:99732577-3,712-128-6,400—   
chr10_99695976_G_Tchr10:99695976-3,712-1,760-4,928—   
chr10_99695980_G_Cchr10:99695980-3,584-1,664-5,376—   
chr10_99695945_T_Achr10:996959453,5841,2804,288—   
chr10_99696006_G_Achr10:99696006-3,520-1,696-5,696—   
chr10_99732604_G_Achr10:997326043,4561,6645,376—   
chr10_99695962_G_Achr10:99695962-3,456-1,536-4,864—   
chr10_99695985_G_Achr10:99695985-3,456-1,024-4,288—   
chr10_99695966_C_Gchr10:99695966-3,456-1,696-4,160—   
chr10_99695998_T_Gchr10:996959983,3921,8566,272—   
chr10_99696005_T_Gchr10:99696005-3,392-1,824-4,608—   
chr10_99695980_G_Tchr10:99695980-3,264-1,504-5,568—   
chr10_99696034_T_Cchr10:99696034-3,232-1,664-4,352—   
chr10_99695954_A_Gchr10:996959543,1041,4084,288—   
chr10_99732714_A_Cchr10:997327143,0721,4409,472—   
chr10_99696018_A_Cchr10:996960183,0401,5364,544—   
chr10_99732665_T_Cchr10:997326653,0081,8885,376—   
chr10_99695916_A_Gchr10:996959162,9122,7846,528—   
chr10_99695962_G_Tchr10:99695962-2,912-1,408-4,544—   
chr10_99732693_T_Cchr10:99732693-2,880-768-4,736—   
chr10_99732691_G_Cchr10:99732691-2,816-576-4,352—   
chr10_99732558_A_Gchr10:997325582,8164164,096—   
chr10_99695973_C_Achr10:99695973-2,784-1,344-4,160—   
chr10_99696006_G_Tchr10:99696006-2,752-1,088-4,224—   
chr10_99695976_G_Achr10:99695976-2,656-1,344-4,4801.3e-5
chr10_99696002_A_Cchr10:996960022,5927364,672—   
chr10_99732725_G_Achr10:99732725-2,496-448-4,992—   
chr10_99695953_T_Gchr10:996959532,4649924,736—   
chr10_99732562_T_Gchr10:997325622,4323846,912—   
chr10_99732661_C_Tchr10:99732661-2,432-1,024-5,120—   
chr10_99732723_C_Achr10:99732723-2,304-352-4,480—   
chr10_99732680_T_Gchr10:997326802,0481,2167,168—   
chr10_99695971_A_Tchr10:996959712,0481,0884,160—   
chr10_99696008_A_Tchr10:99696008-1,984-1,120-4,480—   
chr10_99732713_G_Cchr10:997327131,9209606,7846.6e-6
chr10_99732686_T_Gchr10:997326861,7921,5367,680—   
chr10_99732623_G_Achr10:997326231,664-896-4,864—   
chr10_99732633_C_Gchr10:99732633-1,664-704-4,608—   
chr10_99732544_T_Cchr10:997325441,6645764,096—   
chr10_99732562_T_Cchr10:99732562-1,536-4804,352—   
chr10_99732664_G_Cchr10:99732664-1,472-736-5,632—   
chr10_99732563_G_Achr10:997325631,408256-4,608—   
chr10_99732625_T_Gchr10:99732625-1,408-1,536-4,352—   
chr10_99732711_A_Tchr10:99732711-1,3446724,992—   
chr10_99695911_C_Achr10:996959111,2802,3364,928—   
chr10_99732625_T_Achr10:997326251,280-672-4,352—   
chr10_99732635_G_Cchr10:99732635-1,280-2244,352—   
chr10_99732626_C_Tchr10:99732626-1,152-1,312-8,448—   
chr10_99732628_A_Gchr10:99732628-1,152-1,280-4,608—   
chr10_99732622_G_Tchr10:99732622-1,024-672-4,864—   
chr10_99732596_C_Gchr10:99732596-1,024-256-4,352—   
chr10_99732639_C_Gchr10:997326398969924,608—   
chr10_99732660_C_Achr10:99732660-832-800-5,632—   
chr10_99732693_T_Gchr10:997326936409287,168—   
chr10_99732680_T_Cchr10:99732680-6401284,864—   
chr10_99732626_C_Gchr10:99732626-512-1,280-7,424—   
chr10_99732714_A_Tchr10:99732714-5128004,864—   
chr10_99732715_T_Gchr10:99732715-4482564,224—   
chr10_99732626_C_Achr10:99732626-384-928-7,936—   
chr10_99732627_G_Tchr10:99732627-256-992-5,120—   
chr10_99732564_T_Cchr10:9973256408964,352—   

Showing 200 of 200 in this window. Scores are the raw center bin Δ, ALT minus REF; click a column to sort.