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ABCC3

receptor: PXRTier 1

Drug substrates

methotrexate; morphine-glucuronide; bile acids

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of ABCC3 expression, weakening basolateral transport capacity for organic anions and drug conjugates such as methotrexate and morphine-glucuronide.

Affected substrate drugs (PharmGKB): cisplatin; morphine; cyclophosphamide; doxorubicin; methotrexate; vincristine

Scored variants near ABCC3

chr17:50,534,880..50,792,253, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr17_50543044_C_Gchr17:505430441.0001.0001.000—   
chr17_50542998_A_Tchr17:505429981.0000.8891.000—   
chr17_50543214_A_Gchr17:505432140.2850.3651.000—   
chr17_50543035_A_Tchr17:505430351.0000.9371.000—   
chr17_50543051_T_Gchr17:505430510.9410.8991.000—   
chr17_50543205_C_Gchr17:505432050.8340.7711.000—   
chr17_50543044_C_Tchr17:505430440.7930.5140.9660.0039%
chr17_50543067_T_Achr17:50543067-0.744-0.637-1.000—   
chr17_50543067_T_Gchr17:50543067-0.743-0.615-1.000—   
chr17_50543051_T_Cchr17:505430510.6100.6420.798—   
chr17_50543067_T_Cchr17:50543067-0.607-0.544-0.972—   
chr17_50543060_C_Tchr17:505430600.5900.5390.742—   
chr17_50543195_T_Cchr17:50543195-0.575-0.443-0.978—   
chr17_50543060_C_Achr17:50543060-0.508-0.363-0.966—   
chr17_50543064_T_Gchr17:50543064-0.559-0.348-0.826—   
chr17_50543068_G_Cchr17:50543068-0.559-0.388-0.933—   
chr17_50543035_A_Cchr17:505430350.5490.4940.551—   
chr17_50543064_T_Achr17:50543064-0.546-0.338-0.860—   
chr17_50543196_C_Gchr17:505431960.5410.4380.742—   
chr17_50542998_A_Cchr17:505429980.3900.2670.921—   
chr17_50543031_T_Cchr17:50543031-0.525-0.398-0.843—   
chr17_50543054_A_Gchr17:505430540.5020.4810.775—   
chr17_50543060_C_Gchr17:50543060-0.475-0.325-0.843—   
chr17_50543063_A_Cchr17:50543063-0.489-0.341-0.764—   
chr17_50543052_T_Gchr17:505430520.4770.4310.6970.0059%
chr17_50543065_A_Tchr17:50543065-0.425-0.300-0.809—   
chr17_50543022_G_Cchr17:505430220.4570.2750.573—   
chr17_50543063_A_Gchr17:50543063-0.454-0.320-0.713—   
chr17_50543064_T_Cchr17:50543064-0.449-0.305-0.685—   
chr17_50543070_C_Gchr17:50543070-0.402-0.272-0.758—   
chr17_50543047_A_Gchr17:505430470.4390.3600.697—   
chr17_50543069_A_Cchr17:50543069-0.372-0.282-0.753—   
chr17_50543065_A_Cchr17:50543065-0.398-0.282-0.736—   
chr17_50543055_T_Gchr17:505430550.4230.4690.652—   
chr17_50543000_A_Gchr17:505430000.4050.5790.629—   
chr17_50543057_C_Achr17:505430570.4050.3550.640—   
chr17_50543069_A_Tchr17:50543069-0.339-0.272-0.691—   
chr17_50543053_A_Cchr17:505430530.4020.4160.674—   
chr17_50543070_C_Achr17:50543070-0.351-0.254-0.680—   
chr17_50543052_T_Achr17:505430520.3920.3380.483—   
chr17_50543041_G_Tchr17:505430410.3890.3000.545—   
chr17_50542934_G_Achr17:505429340.2410.2540.663—   
chr17_50543061_A_Gchr17:50543061-0.316-0.259-0.624—   
chr17_50543065_A_Gchr17:50543065-0.356-0.272-0.624—   
chr17_50543035_A_Gchr17:505430350.3610.2470.382<0.001%
chr17_50543038_C_Gchr17:50543038-0.325-0.244-0.612—   
chr17_50543047_A_Cchr17:50543047-0.352-0.307-0.444—   
chr17_50543220_T_Achr17:50543220-0.144-0.164-0.601—   
chr17_50543238_T_Cchr17:50543238-0.031-0.1060.601—   
chr17_50543062_A_Tchr17:50543062-0.348-0.227-0.579—   
chr17_50543066_T_Achr17:50543066-0.305-0.196-0.596—   
chr17_50543232_T_Gchr17:505432320.3460.3450.534—   
chr17_50543066_T_Cchr17:50543066-0.308-0.217-0.590—   
chr17_50543220_T_Gchr17:50543220-0.152-0.174-0.590—   
chr17_50543222_A_Cchr17:50543222-0.143-0.169-0.590—   
chr17_50543044_C_Achr17:505430440.3390.2570.461—   
chr17_50543028_A_Cchr17:505430280.3000.2290.573—   
chr17_50543066_T_Gchr17:50543066-0.307-0.209-0.573—   
chr17_50543063_A_Tchr17:50543063-0.321-0.196-0.556—   
chr17_50542995_T_Gchr17:505429950.2700.2190.551—   
chr17_50543045_C_Gchr17:505430450.2920.2040.551—   
chr17_50543055_T_Achr17:505430550.3210.3450.483—   
chr17_50543062_A_Cchr17:50543062-0.321-0.204-0.511—   
chr17_50543062_A_Gchr17:50543062-0.320-0.207-0.517—   
chr17_50543222_A_Tchr17:50543222-0.123-0.176-0.545—   
chr17_50543045_C_Achr17:505430450.3150.2170.506—   
chr17_50543053_A_Gchr17:505430530.2740.2750.539—   
chr17_50542999_G_Tchr17:505429990.3130.2820.393—   
chr17_50543050_T_Gchr17:505430500.3030.3550.494—   
chr17_50543040_G_Tchr17:505430400.3020.2220.449—   
chr17_50543215_C_Achr17:505432150.2950.2220.517—   
chr17_50543011_C_Achr17:50543011-0.289-0.234-0.393<0.001%
chr17_50543013_G_Tchr17:50543013-0.264-0.259-0.494—   
chr17_50543219_G_Tchr17:50543219-0.098-0.098-0.494—   
chr17_50542996_C_Gchr17:505429960.2850.2370.472—   
chr17_50543219_G_Achr17:50543219-0.105-0.113-0.483—   
chr17_50543015_C_Gchr17:505430150.2750.3800.337—   
chr17_50543055_T_Cchr17:505430550.2750.3050.449—   
chr17_50542966_A_Cchr17:505429660.2740.2920.404—   
chr17_50543188_C_Achr17:50543188-0.244-0.212-0.466—   
chr17_50543202_C_Achr17:505432020.1690.1560.466—   
chr17_50543206_T_Gchr17:505432060.2720.2420.455—   
chr17_50543205_C_Achr17:505432050.2570.2700.461—   
chr17_50543192_A_Gchr17:50543192-0.234-0.181-0.455—   
chr17_50543071_T_Gchr17:50543071-0.262-0.244-0.393—   
chr17_50543030_A_Tchr17:505430300.2590.2540.371—   
chr17_50543222_A_Gchr17:50543222-0.052-0.149-0.444—   
chr17_50542972_C_Achr17:50542972-0.248-0.191-0.438—   
chr17_50543053_A_Tchr17:505430530.2230.2090.438—   
chr17_50543061_A_Tchr17:50543061-0.203-0.191-0.438—   
chr17_50543223_C_Gchr17:505432230.2560.2040.000—   
chr17_50543223_C_Tchr17:505432230.2020.0980.4330.0020%
chr17_50543237_C_Tchr17:505432370.2520.3700.337—   
chr17_50542984_G_Cchr17:505429840.2160.1890.427—   
chr17_50543243_T_Cchr17:50543243-0.249-0.234-0.3600.0013%
chr17_50542997_A_Cchr17:505429970.1930.1740.416—   
chr17_50542999_G_Achr17:505429990.2430.2920.4160.0020%
chr17_50543014_G_Cchr17:50543014-0.239-0.184-0.315<0.001%
chr17_50543040_G_Achr17:50543040-0.239-0.139-0.360—   
chr17_50543204_C_Gchr17:505432040.2110.1990.410—   
chr17_50543220_T_Cchr17:50543220-0.031-0.081-0.410—   
chr17_50542983_C_Gchr17:50542983-0.223-0.035-0.404—   
chr17_50542997_A_Tchr17:505429970.2300.2390.404—   
chr17_50543025_T_Gchr17:505430250.1930.1080.404—   
chr17_50543194_C_Gchr17:50543194-0.179-0.121-0.404—   
chr17_50543243_T_Achr17:50543243-0.236-0.217-0.191—   
chr17_50543001_G_Cchr17:50543001-0.233-0.209-0.388—   
chr17_50542962_A_Gchr17:505429620.1950.3000.393—   
chr17_50543014_G_Tchr17:50543014-0.221-0.184-0.393—   
chr17_50543054_A_Tchr17:505430540.2260.1740.348—   
chr17_50543223_C_Achr17:50543223-0.054-0.081-0.388—   
chr17_50543211_T_Cchr17:50543211-0.223-0.234-0.365—   
chr17_50542940_A_Cchr17:505429400.2160.1460.242—   
chr17_50543034_C_Achr17:50543034-0.166-0.128-0.371—   
chr17_50543043_C_Gchr17:505430430.2160.1760.292—   
chr17_50543059_G_Cchr17:50543059-0.195-0.171-0.371—   
chr17_50543068_G_Achr17:50543068-0.1300.038-0.371—   
chr17_50543003_C_Achr17:50543003-0.215-0.186-0.281—   
chr17_50543203_T_Achr17:505432030.2150.3320.242—   
chr17_50543042_G_Achr17:50543042-0.192-0.126-0.365—   
chr17_50543221_C_Tchr17:50543221-0.044-0.078-0.365—   
chr17_50543057_C_Gchr17:505430570.1790.1710.360—   
chr17_50543069_A_Gchr17:50543069-0.159-0.149-0.360—   
chr17_50542995_T_Achr17:505429950.2080.1810.292—   
chr17_50542956_G_Cchr17:50542956-0.205-0.156-0.348—   
chr17_50543203_T_Cchr17:50543203-0.187-0.096-0.348—   
chr17_50543215_C_Gchr17:505432150.2020.1030.348—   
chr17_50543042_G_Tchr17:50543042-0.154-0.113-0.343—   
chr17_50543195_T_Achr17:50543195-0.198-0.136-0.270—   
chr17_50543030_A_Gchr17:50543030-0.197-0.151-0.264—   
chr17_50542969_A_Cchr17:505429690.0740.0100.331—   
chr17_50543068_G_Tchr17:505430680.1930.2040.292—   
chr17_50543217_G_Cchr17:50543217-0.034-0.053-0.331—   
chr17_50542998_A_Gchr17:505429980.1130.0960.326—   
chr17_50542987_G_Tchr17:50542987-0.187-0.078-0.180—   
chr17_50543027_G_Achr17:50543027-0.169-0.154-0.320—   
chr17_50543028_A_Gchr17:50543028-0.187-0.161-0.287—   
chr17_50543029_G_Achr17:505430290.1870.1960.281—   
chr17_50543052_T_Cchr17:505430520.1870.1660.315—   
chr17_50543192_A_Tchr17:50543192-0.164-0.076-0.320—   
chr17_50543217_G_Achr17:50543217-0.013-0.033-0.320<0.001%
chr17_50542987_G_Achr17:50542987-0.185-0.063-0.067—   
chr17_50542953_C_Gchr17:50542953-0.143-0.128-0.315—   
chr17_50542983_C_Tchr17:50542983-0.175-0.128-0.3150.0020%
chr17_50542992_A_Tchr17:50542992-0.167-0.103-0.315—   
chr17_50543004_A_Tchr17:50543004-0.184-0.159-0.292—   
chr17_50543033_C_Achr17:505430330.1840.2020.253—   
chr17_50543058_A_Cchr17:505430580.1460.1440.315—   
chr17_50543204_C_Achr17:505432040.1840.2620.264—   
chr17_50543021_G_Tchr17:505430210.1820.0960.202—   
chr17_50543025_T_Achr17:505430250.1640.1160.309<0.001%
chr17_50543036_G_Achr17:50543036-0.180-0.154-0.309—   
chr17_50543231_G_Achr17:50543231-0.128-0.086-0.309—   
chr17_50543285_C_Tchr17:505432850.0930.0500.309—   
chr17_50543210_T_Cchr17:505432100.1790.1460.303—   
chr17_50542980_G_Cchr17:505429800.0840.0680.303—   
chr17_50542997_A_Gchr17:505429970.1380.0880.303—   
chr17_50543026_G_Tchr17:50543026-0.092-0.077-0.303—   
chr17_50543051_T_Achr17:505430510.1770.2440.225—   
chr17_50543061_A_Cchr17:50543061-0.169-0.169-0.303—   
chr17_50543208_T_Achr17:50543208-0.162-0.103-0.303—   
chr17_50543211_T_Gchr17:505432110.1770.1030.146—   
chr17_50543215_C_Tchr17:50543215-0.052-0.083-0.303—   
chr17_50543011_C_Tchr17:505430110.1740.1590.281—   
chr17_50543194_C_Achr17:50543194-0.139-0.078-0.298—   
chr17_50543216_T_Gchr17:50543216-0.030-0.058-0.298—   
chr17_50543235_C_Achr17:50543235-0.149-0.113-0.298<0.001%
chr17_50543243_T_Gchr17:50543243-0.172-0.214-0.219—   
chr17_50542939_G_Cchr17:505429390.1700.1310.022—   
chr17_50543001_G_Tchr17:50543001-0.170-0.161-0.292—   
chr17_50543016_T_Gchr17:505430160.1620.1160.292—   
chr17_50543020_A_Tchr17:505430200.1700.1460.258—   
chr17_50543196_C_Achr17:50543196-0.169-0.101-0.292—   
chr17_50543225_T_Gchr17:505432250.0700.0130.292—   
chr17_50543189_A_Tchr17:505431890.1640.1030.287—   
chr17_50543202_C_Gchr17:50543202-0.095-0.050-0.287—   
chr17_50543209_G_Achr17:50543209-0.128-0.101-0.287—   
chr17_50542988_C_Achr17:50542988-0.166-0.096-0.213—   
chr17_50542999_G_Cchr17:505429990.1660.1690.281—   
chr17_50543022_G_Tchr17:505430220.1660.0860.146—   
chr17_50542986_G_Achr17:505429860.1110.1230.281—   
chr17_50542996_C_Achr17:505429960.1640.1710.258—   
chr17_50543207_T_Gchr17:505432070.1640.1560.185—   
chr17_50542983_C_Achr17:50542983-0.162-0.048-0.236—   
chr17_50543014_G_Achr17:50543014-0.162-0.116-0.247—   
chr17_50543071_T_Achr17:505430710.1620.1910.191—   
chr17_50543039_T_Achr17:505430390.1610.0980.225—   
chr17_50543189_A_Gchr17:505431890.0920.0450.275—   
chr17_50543239_G_Cchr17:50543239-0.152-0.161-0.275—   
chr17_50549487_G_Cchr17:505494870.0000.0980.275—   
chr17_50549489_T_Gchr17:505494890.0160.1300.275—   
chr17_50542981_G_Tchr17:505429810.1130.1340.270—   
chr17_50542989_T_Cchr17:505429890.0820.0760.270—   
chr17_50543000_A_Cchr17:505430000.1340.0930.270—   
chr17_50543013_G_Achr17:50543013-0.152-0.136-0.270—   
chr17_50543203_T_Gchr17:505432030.1570.1210.230<0.001%
chr17_50543023_C_Tchr17:505430230.1560.1080.112<0.001%
chr17_50543034_C_Tchr17:50543034-0.111-0.073-0.264<0.001%
chr17_50543189_A_Cchr17:505431890.1300.0880.264—   
chr17_50543193_G_Achr17:505431930.0770.0530.264—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.