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CES2

receptor: PXRTier 1

Drug substrates

irinotecan (activation to SN-38); prodrug esters

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of CES2 expression, impairing the hydrolytic bioactivation of key prodrugs such as irinotecan.

Affected substrate drugs (PharmGKB): irinotecan

Scored variants near CES2

chr16:66,834,470..67,045,091, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr16_66934353_G_Cchr16:669343530.5070.1110.135—   
chr16_66934236_T_Achr16:669342360.2850.1710.697—   
chr16_66934277_C_Achr16:669342770.2210.3480.663—   
chr16_66934263_G_Cchr16:669342630.1480.2420.573—   
chr16_66934353_G_Tchr16:669343530.3300.1690.213—   
chr16_66912684_T_Achr16:669126840.296-0.0670.087—   
chr16_66934345_A_Cchr16:66934345-0.210-0.179-0.483—   
chr16_66934311_G_Achr16:669343110.2720.0450.056—   
chr16_66934351_C_Gchr16:669343510.2590.0710.270—   
chr16_66934257_C_Gchr16:669342570.0520.0600.438—   
chr16_66934289_G_Cchr16:669342890.2390.1690.213—   
chr16_66934214_G_Tchr16:66934214-0.093-0.083-0.404—   
chr16_66934289_G_Achr16:669342890.2300.1340.2130.0020%
chr16_66934221_A_Gchr16:669342210.0160.0810.382—   
chr16_66934238_C_Achr16:669342380.1840.0880.371—   
chr16_66934225_A_Cchr16:669342250.0360.0630.360—   
chr16_66934343_C_Tchr16:669343430.2100.0730.169—   
chr16_66934220_T_Achr16:669342200.0850.1180.337—   
chr16_66934233_G_Tchr16:66934233-0.057-0.048-0.326—   
chr16_66934230_C_Gchr16:66934230-0.105-0.091-0.315—   
chr16_66934230_C_Tchr16:66934230-0.105-0.045-0.315<0.001%
chr16_66934319_T_Cchr16:66934319-0.180-0.060-0.067—   
chr16_66934227_G_Tchr16:66934227-0.079-0.063-0.3030.054%
chr16_66934232_C_Tchr16:66934232-0.110-0.040-0.303—   
chr16_66934355_C_Gchr16:669343550.0950.0580.303—   
chr16_66934347_C_Gchr16:66934347-0.1740.048-0.067—   
chr16_66934349_C_Gchr16:669343490.1740.0280.146—   
chr16_66934235_G_Tchr16:66934235-0.074-0.033-0.292—   
chr16_66934316_G_Cchr16:669343160.1700.0150.202—   
chr16_66934348_C_Achr16:669343480.167-0.0230.191—   
chr16_66934348_C_Gchr16:669343480.1640.0580.135—   
chr16_66934226_A_Tchr16:669342260.0490.0580.270—   
chr16_66934233_G_Cchr16:66934233-0.039-0.050-0.270—   
chr16_66934214_G_Cchr16:66934214-0.026-0.083-0.258—   
chr16_66934234_C_Tchr16:66934234-0.062-0.058-0.258<0.001%
chr16_66934235_G_Cchr16:66934235-0.077-0.040-0.258—   
chr16_66934240_T_Achr16:66934240-0.052-0.086-0.258—   
chr16_66934291_T_Cchr16:66934291-0.087-0.028-0.258—   
chr16_66934334_G_Tchr16:66934334-0.075-0.008-0.258—   
chr16_66934348_C_Tchr16:669343480.1510.0600.045—   
chr16_66934351_C_Achr16:669343510.1510.0710.124—   
chr16_66936462_C_Achr16:66936462-0.079-0.131-0.258—   
chr16_66934357_C_Gchr16:669343570.146-0.0100.135—   
chr16_66934234_C_Achr16:66934234-0.062-0.050-0.247—   
chr16_66934244_T_Gchr16:669342440.0590.0630.247—   
chr16_66934231_T_Gchr16:66934231-0.1410.0880.135—   
chr16_66934345_A_Gchr16:669343450.1410.0130.157—   
chr16_66934225_A_Tchr16:66934225-0.0030.0330.236—   
chr16_66934326_C_Gchr16:669343260.1380.0050.146—   
chr16_66934352_C_Gchr16:669343520.1050.0150.236—   
chr16_66934232_C_Achr16:66934232-0.064-0.073-0.225—   
chr16_66934234_C_Gchr16:66934234-0.075-0.060-0.225—   
chr16_66934338_G_Cchr16:66934338-0.075-0.071-0.225—   
chr16_66934339_C_Gchr16:669343390.131-0.0030.169—   
chr16_66934354_C_Tchr16:669343540.1310.0430.067—   
chr16_66934291_T_Gchr16:669342910.1300.0430.135—   
chr16_66934224_G_Achr16:66934224-0.002-0.010-0.213—   
chr16_66934235_G_Achr16:66934235-0.061-0.025-0.213—   
chr16_66934340_C_Gchr16:669343400.1250.0200.112—   
chr16_66934219_A_Tchr16:669342190.1210.0380.067—   
chr16_66934354_C_Gchr16:669343540.1210.0280.169—   
chr16_66934359_T_Cchr16:66934359-0.121-0.096-0.045—   
chr16_66934214_G_Achr16:66934214-0.013-0.048-0.2020.0039%
chr16_66934227_G_Achr16:66934227-0.036-0.010-0.202—   
chr16_66934232_C_Gchr16:66934232-0.090-0.050-0.202—   
chr16_66934261_T_Gchr16:669342610.0280.0680.202—   
chr16_66934321_G_Achr16:669343210.016-0.018-0.202—   
chr16_66934358_C_Achr16:669343580.1180.0810.101—   
chr16_66934349_C_Achr16:669343490.1150.0430.079—   
chr16_66934215_G_Cchr16:669342150.0390.0880.191—   
chr16_66934220_T_Gchr16:669342200.0560.0180.191—   
chr16_66934230_C_Achr16:66934230-0.049-0.013-0.191—   
chr16_66934309_A_Gchr16:669343090.0110.0080.191—   
chr16_66934341_G_Cchr16:66934341-0.030-0.073-0.191—   
chr16_66934228_A_Cchr16:66934228-0.110-0.093-0.135—   
chr16_66934344_G_Tchr16:669343440.1080.020-0.0340.0020%
chr16_66934356_G_Cchr16:66934356-0.108-0.065-0.090—   
chr16_66934216_C_Achr16:669342160.007-0.028-0.180—   
chr16_66934219_A_Cchr16:669342190.0430.0300.180—   
chr16_66934226_A_Cchr16:66934226-0.030-0.0100.180—   
chr16_66934240_T_Gchr16:66934240-0.062-0.091-0.180<0.001%
chr16_66934251_G_Cchr16:669342510.0330.0100.180—   
chr16_66934264_T_Gchr16:669342640.0130.0710.180—   
chr16_66934273_C_Gchr16:669342730.0360.0650.180—   
chr16_66934322_C_Gchr16:669343220.1050.0080.056—   
chr16_66934342_C_Tchr16:669343420.1050.033-0.011—   
chr16_66934346_C_Gchr16:669343460.1050.0130.045—   
chr16_66934248_G_Achr16:669342480.102-0.025-0.101—   
chr16_66934333_A_Tchr16:669343330.1020.008-0.011—   
chr16_66934337_C_Gchr16:669343370.1020.0330.079—   
chr16_66934339_C_Tchr16:669343390.1020.0130.045—   
chr16_66934351_C_Tchr16:669343510.1020.0630.146—   
chr16_66934238_C_Gchr16:66934238-0.100-0.063-0.146—   
chr16_66934211_A_Gchr16:66934211-0.0130.0350.169—   
chr16_66934212_G_Tchr16:669342120.003-0.035-0.169—   
chr16_66934220_T_Cchr16:669342200.010-0.0430.169—   
chr16_66934228_A_Gchr16:66934228-0.098-0.096-0.124—   
chr16_66934237_G_Achr16:66934237-0.0020.025-0.169—   
chr16_66934237_G_Cchr16:66934237-0.026-0.030-0.169—   
chr16_66934241_C_Gchr16:66934241-0.079-0.050-0.169—   
chr16_66934248_G_Tchr16:66934248-0.043-0.028-0.169<0.001%
chr16_66934257_C_Tchr16:66934257-0.0230.0450.169—   
chr16_66934268_C_Achr16:669342680.0720.1130.169—   
chr16_66934274_C_Gchr16:669342740.0430.0330.169—   
chr16_66934350_G_Cchr16:669343500.0660.035-0.169—   
chr16_66934311_G_Tchr16:669343110.0950.0430.034—   
chr16_66934316_G_Tchr16:669343160.0950.0080.056—   
chr16_66934341_G_Tchr16:669343410.0930.033-0.011—   
chr16_66934215_G_Achr16:66934215-0.003-0.030-0.157<0.001%
chr16_66934231_T_Cchr16:66934231-0.025-0.058-0.157—   
chr16_66934239_G_Achr16:669342390.036-0.040-0.157—   
chr16_66934252_G_Cchr16:669342520.0720.0300.157—   
chr16_66934263_G_Achr16:669342630.033-0.020-0.157—   
chr16_66934269_C_Achr16:669342690.007-0.015-0.157—   
chr16_66934270_T_Gchr16:669342700.0130.0400.157—   
chr16_66934277_C_Gchr16:669342770.0110.0600.157—   
chr16_66934278_C_Achr16:66934278-0.007-0.040-0.157—   
chr16_66934310_T_Gchr16:66934310-0.0030.0280.157—   
chr16_66936480_C_Gchr16:669364800.0920.0830.090—   
chr16_66934319_T_Achr16:66934319-0.089-0.0400.000—   
chr16_66934320_G_Cchr16:66934320-0.089-0.035-0.022—   
chr16_66934226_A_Gchr16:66934226-0.087-0.065-0.112—   
chr16_66934353_G_Achr16:669343530.0870.0230.000—   
chr16_66936479_C_Achr16:669364790.0870.0910.045—   
chr16_66912608_G_Cchr16:669126080.034-0.0040.146—   
chr16_66934213_C_Achr16:66934213-0.066-0.030-0.146—   
chr16_66934213_C_Tchr16:66934213-0.034-0.040-0.146—   
chr16_66934217_G_Tchr16:669342170.030-0.045-0.146—   
chr16_66934222_T_Gchr16:669342220.020-0.0050.146—   
chr16_66934227_G_Cchr16:66934227-0.008-0.030-0.146—   
chr16_66934242_G_Tchr16:66934242-0.013-0.015-0.146—   
chr16_66934243_A_Gchr16:669342430.0070.0130.146—   
chr16_66934279_G_Achr16:669342790.000-0.023-0.146—   
chr16_66934281_C_Tchr16:669342810.034-0.038-0.146—   
chr16_66934285_G_Tchr16:66934285-0.0410.010-0.146<0.001%
chr16_66934299_G_Tchr16:66934299-0.033-0.048-0.146—   
chr16_66934309_A_Cchr16:669343090.0230.0350.146—   
chr16_66934310_T_Cchr16:669343100.0230.0180.1460.0020%
chr16_66934319_T_Gchr16:66934319-0.085-0.0450.079—   
chr16_66934340_C_Achr16:669343400.0850.0000.034—   
chr16_66934344_G_Cchr16:669343440.003-0.088-0.146—   
chr16_66934352_C_Tchr16:669343520.0850.0080.1240.0033%
chr16_66934358_C_Gchr16:669343580.0850.0530.146—   
chr16_66936478_T_Gchr16:669364780.0840.0930.146—   
chr16_66936489_C_Gchr16:669364890.0850.0730.011—   
chr16_66936492_T_Gchr16:669364920.0850.0350.112—   
chr16_66934231_T_Achr16:66934231-0.082-0.005-0.022—   
chr16_66934337_C_Achr16:669343370.0820.0150.045—   
chr16_66934352_C_Achr16:669343520.082-0.0050.045—   
chr16_66936464_G_Achr16:669364640.0820.0550.056—   
chr16_66936491_C_Gchr16:669364910.0820.0580.045—   
chr16_66936479_C_Gchr16:669364790.0800.0760.090—   
chr16_66934217_G_Achr16:669342170.023-0.033-0.1350.0013%
chr16_66934236_T_Cchr16:66934236-0.079-0.0180.011—   
chr16_66934245_G_Achr16:669342450.002-0.023-0.135—   
chr16_66934306_T_Cchr16:669343060.0390.0580.135—   
chr16_66934313_G_Tchr16:66934313-0.028-0.038-0.135—   
chr16_66934327_T_Gchr16:669343270.0750.0300.135—   
chr16_66934329_C_Achr16:66934329-0.079-0.018-0.135—   
chr16_66934331_G_Achr16:66934331-0.023-0.003-0.1350.0020%
chr16_66934336_C_Tchr16:66934336-0.0790.0080.022—   
chr16_66934228_A_Tchr16:66934228-0.0750.005-0.022—   
chr16_66934292_C_Tchr16:66934292-0.075-0.038-0.112—   
chr16_66934327_T_Cchr16:669343270.0750.0280.045—   
chr16_66936476_C_Achr16:669364760.0750.1060.112—   
chr16_66936476_C_Gchr16:669364760.0750.1460.112—   
chr16_66934217_G_Cchr16:669342170.026-0.063-0.124—   
chr16_66934218_G_Tchr16:669342180.023-0.020-0.124—   
chr16_66934233_G_Achr16:669342330.028-0.020-0.124—   
chr16_66934242_G_Achr16:66934242-0.0490.013-0.124—   
chr16_66934264_T_Cchr16:669342640.0490.0710.124—   
chr16_66934265_C_Gchr16:669342650.0590.0400.124—   
chr16_66934266_C_Achr16:66934266-0.0590.0880.124—   
chr16_66934276_G_Achr16:669342760.003-0.018-0.124—   
chr16_66934284_A_Tchr16:669342840.0460.0230.124—   
chr16_66934308_G_Tchr16:669343080.0720.0330.079—   
chr16_66934316_G_Achr16:669343160.0720.0280.101—   
chr16_66934334_G_Achr16:669343340.0160.091-0.124<0.001%
chr16_66934349_C_Tchr16:669343490.0660.0530.124—   
chr16_66936458_G_Cchr16:669364580.0720.0830.011—   
chr16_66934317_G_Cchr16:66934317-0.070-0.0180.045<0.001%
chr16_66934321_G_Cchr16:66934321-0.070-0.028-0.056—   
chr16_66936478_T_Achr16:669364780.0700.0760.101—   
chr16_66934252_G_Achr16:669342520.0690.0180.0220.0013%
chr16_66934306_T_Achr16:66934306-0.069-0.033-0.079—   
chr16_66934334_G_Cchr16:66934334-0.0690.018-0.079—   
chr16_66934343_C_Gchr16:669343430.069-0.0330.090—   
chr16_66934354_C_Achr16:669343540.0690.0430.034—   
chr16_66936474_T_Cchr16:669364740.0690.0530.056—   
chr16_66934215_G_Tchr16:669342150.049-0.038-0.112—   
chr16_66934216_C_Tchr16:66934216-0.052-0.055-0.112—   
chr16_66934223_C_Gchr16:669342230.0070.0230.112—   
chr16_66934224_G_Cchr16:66934224-0.066-0.043-0.112—   
chr16_66934224_G_Tchr16:669342240.0030.013-0.112—   
chr16_66934237_G_Tchr16:669342370.0360.005-0.112—   
chr16_66934243_A_Cchr16:669342430.0000.0150.112—   
chr16_66934244_T_Cchr16:669342440.0660.0730.101—   
chr16_66934246_C_Tchr16:66934246-0.007-0.015-0.1120.0013%
chr16_66934251_G_Achr16:66934251-0.013-0.010-0.112—   
chr16_66934253_G_Achr16:669342530.0660.0350.045—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.