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CYP1B1

receptor: AhRTier 1

Drug substrates

estradiol 4-hydroxylation; pro-carcinogen activation

refs: 37707797

CAMIP causal chains

AhR

Impaired receptor-mediated signaling that abolishes both the basal constitutive expression and chemical inducibility of CYP1B1 in extrahepatic tissues, perturbing the localized pathway of estradiol 4-hydroxylation and procarcinogen activation that drives tissue-specific susceptibility to malignancies.

Affected substrate drugs (PharmGKB): cyclophosphamide; doxorubicin; fluorouracil; risperidone; epirubicin; paclitaxel

Scored variants near CYP1B1

chr2:37,967,509..38,176,151, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr2_38015061_T_Gchr2:380150610.4540.3730.878—   
chr2_38076076_G_Achr2:380760760.3210.0910.247—   
chr2_38075966_G_Cchr2:380759660.3150.2040.348—   
chr2_38076022_G_Cchr2:380760220.1900.0960.270—   
chr2_38075974_C_Tchr2:38075974-0.092-0.096-0.303<0.001%
chr2_38076020_T_Gchr2:380760200.1700.0960.135—   
chr2_38015049_A_Cchr2:380150490.1230.1450.288—   
chr2_38075971_G_Tchr2:380759710.1570.0550.079—   
chr2_38075968_T_Cchr2:380759680.1180.1060.258—   
chr2_38076015_G_Tchr2:380760150.1440.0680.090—   
chr2_38076038_C_Gchr2:380760380.1440.0400.101—   
chr2_38076122_A_Tchr2:38076122-0.125-0.131-0.247—   
chr2_38075942_C_Gchr2:38075942-0.138-0.043-0.101—   
chr2_38076037_C_Achr2:380760370.1340.078-0.135—   
chr2_38075967_A_Cchr2:380759670.1310.1360.157—   
chr2_38075969_G_Cchr2:380759690.1280.0810.225—   
chr2_38075982_G_Cchr2:380759820.0980.0480.225—   
chr2_38075983_G_Cchr2:380759830.1050.0680.225—   
chr2_38076030_G_Cchr2:380760300.1310.0880.101—   
chr2_38076118_C_Achr2:38076118-0.072-0.035-0.225—   
chr2_38076127_T_Gchr2:38076127-0.131-0.003-0.079—   
chr2_38076062_G_Tchr2:380760620.1280.0760.169—   
chr2_38075966_G_Achr2:380759660.1110.1160.213—   
chr2_38075968_T_Gchr2:38075968-0.0260.0930.213—   
chr2_38076015_G_Cchr2:380760150.1250.0500.090—   
chr2_38076024_A_Cchr2:380760240.1250.0430.213—   
chr2_38076087_C_Gchr2:380760870.020-0.025-0.213—   
chr2_38076093_C_Gchr2:380760930.1250.035-0.056—   
chr2_38075935_G_Achr2:380759350.1210.038-0.011—   
chr2_38076062_G_Cchr2:380760620.1210.0710.135—   
chr2_38075966_G_Tchr2:380759660.1180.1110.135—   
chr2_38076102_C_Gchr2:380761020.1180.0230.090—   
chr2_38076008_C_Achr2:380760080.1150.0780.090—   
chr2_38076013_G_Tchr2:380760130.1150.0500.045—   
chr2_38076113_A_Cchr2:38076113-0.115-0.065-0.169—   
chr2_38075940_G_Achr2:380759400.1110.0630.0670.0039%
chr2_38075942_C_Achr2:38075942-0.111-0.0050.022—   
chr2_38075952_A_Gchr2:38075952-0.111-0.040-0.079—   
chr2_38075970_G_Tchr2:380759700.1110.0730.135—   
chr2_38075986_C_Achr2:380759860.0980.0830.191—   
chr2_38076057_G_Achr2:380760570.0690.0680.1910.0026%
chr2_38076067_C_Gchr2:380760670.0460.0630.191—   
chr2_38076080_C_Tchr2:38076080-0.111-0.025-0.079—   
chr2_38076087_C_Achr2:380760870.039-0.015-0.191—   
chr2_38076063_G_Cchr2:380760630.1080.0810.169—   
chr2_38076064_G_Tchr2:380760640.1080.0480.101—   
chr2_38075949_A_Cchr2:38075949-0.105-0.015-0.022—   
chr2_38075950_G_Tchr2:38075950-0.105-0.068-0.112—   
chr2_38075963_T_Cchr2:380759630.1050.0710.180—   
chr2_38075965_G_Cchr2:380759650.1050.0930.169—   
chr2_38075995_C_Tchr2:38075995-0.010-0.023-0.180—   
chr2_38076004_G_Cchr2:38076004-0.105-0.045-0.124—   
chr2_38076014_G_Tchr2:380760140.1050.0380.067—   
chr2_38076030_G_Achr2:38076030-0.105-0.0100.011—   
chr2_38076078_G_Achr2:38076078-0.066-0.043-0.180—   
chr2_38076078_G_Cchr2:38076078-0.105-0.005-0.034—   
chr2_38076125_G_Cchr2:38076125-0.105-0.0380.034—   
chr2_38075949_A_Gchr2:38075949-0.098-0.055-0.045—   
chr2_38075995_C_Achr2:38075995-0.023-0.028-0.169—   
chr2_38076016_G_Achr2:380760160.0980.0280.090—   
chr2_38076016_G_Tchr2:380760160.098-0.005-0.056—   
chr2_38076028_T_Cchr2:380760280.0460.0480.169—   
chr2_38076063_G_Achr2:380760630.0890.0530.169—   
chr2_38076097_C_Gchr2:38076097-0.098-0.003-0.045—   
chr2_38075961_A_Gchr2:38075961-0.095-0.028-0.112<0.001%
chr2_38076127_T_Cchr2:38076127-0.095-0.015-0.022—   
chr2_38075950_G_Cchr2:38075950-0.092-0.048-0.056—   
chr2_38075952_A_Cchr2:38075952-0.092-0.013-0.034—   
chr2_38075970_G_Achr2:380759700.0920.0600.090—   
chr2_38075971_G_Cchr2:380759710.0920.0530.090—   
chr2_38076015_G_Achr2:380760150.0920.0380.000—   
chr2_38076031_A_Cchr2:38076031-0.0200.0150.157<0.001%
chr2_38076038_C_Achr2:380760380.0920.0400.022—   
chr2_38076066_T_Gchr2:380760660.0260.0400.157—   
chr2_38076075_G_Tchr2:380760750.0920.0430.067—   
chr2_38076077_C_Gchr2:38076077-0.0920.0350.056—   
chr2_38076086_C_Tchr2:38076086-0.059-0.033-0.157—   
chr2_38076108_A_Gchr2:380761080.0390.0280.1570.0013%
chr2_38076111_G_Tchr2:38076111-0.089-0.030-0.022—   
chr2_38075935_G_Tchr2:380759350.0850.010-0.045—   
chr2_38075943_A_Gchr2:38075943-0.075-0.023-0.146<0.001%
chr2_38075946_G_Achr2:38075946-0.052-0.050-0.146—   
chr2_38075968_T_Achr2:380759680.0070.0350.146<0.001%
chr2_38075979_A_Cchr2:380759790.0460.0200.146—   
chr2_38075983_G_Achr2:38075983-0.030-0.060-0.146—   
chr2_38075987_C_Achr2:38075987-0.039-0.048-0.146—   
chr2_38076003_C_Achr2:380760030.0850.0350.056—   
chr2_38076004_G_Tchr2:38076004-0.062-0.050-0.146—   
chr2_38076057_G_Cchr2:380760570.0360.0180.146—   
chr2_38076061_G_Achr2:380760610.0260.0230.146—   
chr2_38076068_G_Tchr2:38076068-0.020-0.050-0.146<0.001%
chr2_38076079_T_Cchr2:38076079-0.0850.0000.000—   
chr2_38076097_C_Achr2:38076097-0.085-0.035-0.1010.0033%
chr2_38076107_A_Cchr2:380761070.0850.0180.135—   
chr2_38075969_G_Tchr2:380759690.0820.0300.034—   
chr2_38076061_G_Cchr2:380760610.0820.0430.0900.0013%
chr2_38075938_T_Cchr2:38075938-0.079-0.0130.045—   
chr2_38075948_C_Achr2:38075948-0.079-0.038-0.101—   
chr2_38075951_G_Cchr2:380759510.0790.0500.124—   
chr2_38075980_A_Tchr2:38075980-0.013-0.048-0.135—   
chr2_38075983_G_Tchr2:380759830.0790.0500.079—   
chr2_38075984_T_Gchr2:38075984-0.079-0.043-0.045—   
chr2_38075985_G_Achr2:38075985-0.033-0.028-0.135—   
chr2_38076014_G_Cchr2:380760140.0790.0380.135—   
chr2_38076019_C_Gchr2:380760190.0490.0180.135—   
chr2_38076026_A_Gchr2:380760260.0070.0030.135—   
chr2_38076032_G_Tchr2:380760320.0790.0300.045—   
chr2_38076042_C_Achr2:38076042-0.079-0.018-0.135—   
chr2_38076053_T_Gchr2:380760530.0300.0350.135—   
chr2_38076054_T_Cchr2:380760540.0750.0480.135—   
chr2_38076062_G_Achr2:380760620.0690.0380.135—   
chr2_38076069_G_Achr2:380760690.039-0.033-0.135—   
chr2_38076073_G_Tchr2:380760730.020-0.048-0.135—   
chr2_38076086_C_Achr2:38076086-0.007-0.015-0.135—   
chr2_38076102_C_Tchr2:380761020.0720.0630.135—   
chr2_38076104_C_Gchr2:380761040.0790.0250.101—   
chr2_38076120_G_Tchr2:380761200.0160.0350.135—   
chr2_38075936_C_Tchr2:380759360.0750.0250.000<0.001%
chr2_38075961_A_Cchr2:380759610.0750.0430.056—   
chr2_38076121_A_Cchr2:380761210.0750.0200.079—   
chr2_38076121_A_Tchr2:380761210.0750.0250.079—   
chr2_38075936_C_Gchr2:38075936-0.072-0.0350.022—   
chr2_38075946_G_Cchr2:38075946-0.072-0.040-0.034—   
chr2_38075955_G_Tchr2:380759550.0720.010-0.079—   
chr2_38075958_T_Achr2:38075958-0.072-0.0150.011—   
chr2_38075964_G_Cchr2:380759640.0720.0530.124—   
chr2_38075975_G_Tchr2:380759750.0720.023-0.022—   
chr2_38075979_A_Gchr2:380759790.0660.0350.124—   
chr2_38075981_G_Cchr2:380759810.0590.0280.1240.070%
chr2_38075990_G_Tchr2:38075990-0.003-0.003-0.124—   
chr2_38075992_T_Cchr2:38075992-0.072-0.018-0.034—   
chr2_38075992_T_Gchr2:38075992-0.072-0.018-0.011—   
chr2_38075999_G_Achr2:38075999-0.007-0.010-0.1240.0013%
chr2_38076026_A_Cchr2:38076026-0.046-0.055-0.124—   
chr2_38076029_C_Achr2:38076029-0.0720.000-0.045—   
chr2_38076039_T_Achr2:380760390.0720.0130.022—   
chr2_38076064_G_Achr2:380760640.0490.0530.1240.042%
chr2_38076065_G_Achr2:380760650.0490.0380.124—   
chr2_38076081_A_Tchr2:38076081-0.072-0.003-0.022—   
chr2_38076093_C_Achr2:380760930.072-0.008-0.0900.0020%
chr2_38076096_G_Cchr2:380760960.0720.0710.034—   
chr2_38076108_A_Tchr2:38076108-0.072-0.043-0.067—   
chr2_38076112_G_Cchr2:380761120.0330.0250.124—   
chr2_38075934_G_Achr2:38075934-0.069-0.0130.056—   
chr2_38075949_A_Tchr2:38075949-0.069-0.055-0.045—   
chr2_38075973_A_Tchr2:380759730.0690.003-0.034—   
chr2_38075985_G_Cchr2:38075985-0.069-0.043-0.090—   
chr2_38076001_C_Tchr2:380760010.0690.0280.000—   
chr2_38076040_C_Achr2:38076040-0.0690.023-0.011—   
chr2_38076071_G_Tchr2:380760710.069-0.018-0.045—   
chr2_38075942_C_Tchr2:38075942-0.066-0.023-0.0340.0026%
chr2_38075945_T_Gchr2:38075945-0.066-0.0380.0220.0013%
chr2_38075947_C_Tchr2:38075947-0.046-0.038-0.112—   
chr2_38075953_G_Tchr2:380759530.0660.0130.022—   
chr2_38075959_G_Cchr2:380759590.0660.0330.067—   
chr2_38075961_A_Tchr2:38075961-0.066-0.020-0.112—   
chr2_38075964_G_Tchr2:380759640.0660.0450.056—   
chr2_38075970_G_Cchr2:380759700.0460.0430.112<0.001%
chr2_38075972_G_Tchr2:380759720.0660.020-0.011—   
chr2_38075973_A_Gchr2:380759730.0360.0710.112—   
chr2_38075977_A_Tchr2:380759770.0660.0080.000—   
chr2_38075978_G_Tchr2:380759780.046-0.018-0.112—   
chr2_38076002_C_Tchr2:380760020.0660.0280.034—   
chr2_38076003_C_Tchr2:380760030.0660.0250.022—   
chr2_38076007_G_Achr2:38076007-0.030-0.025-0.112—   
chr2_38076009_C_Tchr2:380760090.013-0.003-0.112—   
chr2_38076016_G_Cchr2:380760160.0660.0150.067—   
chr2_38076023_C_Gchr2:38076023-0.066-0.023-0.011—   
chr2_38076042_C_Gchr2:38076042-0.039-0.013-0.112—   
chr2_38076044_G_Achr2:38076044-0.066-0.003-0.067—   
chr2_38076048_T_Cchr2:38076048-0.066-0.008-0.079—   
chr2_38076056_A_Cchr2:380760560.0330.0250.112—   
chr2_38076057_G_Tchr2:380760570.0660.015-0.011—   
chr2_38076059_C_Tchr2:38076059-0.039-0.025-0.112—   
chr2_38076060_T_Achr2:380760600.0660.0450.090—   
chr2_38076066_T_Achr2:38076066-0.066-0.0130.079—   
chr2_38076089_T_Cchr2:38076089-0.0200.0050.112—   
chr2_38076091_C_Achr2:38076091-0.066-0.030-0.034—   
chr2_38076110_T_Gchr2:380761100.0130.0380.112—   
chr2_38076111_G_Achr2:38076111-0.066-0.0050.011—   
chr2_38076113_A_Gchr2:38076113-0.066-0.0180.090—   
chr2_38076123_G_Cchr2:38076123-0.066-0.045-0.090—   
chr2_38076127_T_Achr2:38076127-0.066-0.023-0.022—   
chr2_38075934_G_Tchr2:38075934-0.062-0.0180.022—   
chr2_38075969_G_Achr2:380759690.0620.0450.0900.0046%
chr2_38076013_G_Cchr2:380760130.0620.0300.101—   
chr2_38076054_T_Achr2:380760540.0620.0100.000—   
chr2_38076065_G_Cchr2:380760650.0620.0530.090—   
chr2_38015052_G_Cchr2:380150520.0600.0720.105—   
chr2_38075937_G_Cchr2:38075937-0.043-0.0030.101—   
chr2_38075939_C_Achr2:380759390.0300.0330.101—   
chr2_38075939_C_Gchr2:38075939-0.0330.0150.101—   
chr2_38075941_T_Gchr2:38075941-0.0590.0100.011—   
chr2_38075945_T_Cchr2:38075945-0.007-0.0050.101—   
chr2_38075954_C_Gchr2:38075954-0.059-0.035-0.011—   
chr2_38075967_A_Tchr2:380759670.0590.0910.011—   
chr2_38075976_G_Cchr2:380759760.0390.0200.1010.0039%
chr2_38075991_C_Gchr2:38075991-0.013-0.020-0.101—   
chr2_38075994_G_Cchr2:38075994-0.046-0.048-0.101—   
chr2_38075994_G_Tchr2:380759940.007-0.018-0.101—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.