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CYP2A6

receptor: PXRTier 1

Drug substrates

nicotine; letrozole; tegafur; coumarin

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of CYP2A6 decreases the hepatic oxidative metabolism and clearance of its substrates such as nicotine and coumarin.

Affected substrate drugs (PharmGKB): nicotine; coumarin; tegafur; efavirenz; letrozole; metronidazole

Scored variants near CYP2A6

chr19:40,743,540..40,950,447, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr19_40751082_C_Tchr19:407510820.044-0.164-0.775—   
chr19_40751083_G_Cchr19:407510830.067-0.295-0.584—   
chr19_40751082_C_Achr19:407510820.061-0.081-0.573—   
chr19_40751082_C_Gchr19:407510820.033-0.073-0.562—   
chr19_40751083_G_Achr19:407510830.030-0.242-0.562—   
chr19_40751081_C_Tchr19:407510810.000-0.134-0.528—   
chr19_40751080_T_Cchr19:407510800.156-0.065-0.506—   
chr19_40751080_T_Achr19:407510800.074-0.048-0.494—   
chr19_40751081_C_Achr19:407510810.049-0.113-0.494—   
chr19_40750940_A_Cchr19:407509400.1640.3430.483—   
chr19_40751083_G_Tchr19:40751083-0.052-0.196-0.483—   
chr19_40751079_A_Tchr19:40751079-0.1380.1260.472—   
chr19_40751081_C_Gchr19:407510810.046-0.156-0.472—   
chr19_40751084_G_Achr19:407510840.025-0.141-0.472—   
chr19_40751120_C_Achr19:40751120-0.059-0.451-0.461—   
chr19_40798060_C_Achr19:40798060-0.0490.1490.461—   
chr19_40751144_G_Cchr19:40751144-0.267-0.149-0.416—   
chr19_40751145_C_Gchr19:40751145-0.257-0.184-0.348—   
chr19_40751077_A_Cchr19:40751077-0.043-0.144-0.404—   
chr19_40751080_T_Gchr19:407510800.131-0.068-0.404—   
chr19_40751078_C_Achr19:407510780.038-0.254-0.393—   
chr19_40751079_A_Cchr19:407510790.144-0.073-0.382—   
chr19_40750981_C_Achr19:40750981-0.046-0.065-0.371—   
chr19_40751146_T_Gchr19:40751146-0.211-0.103-0.270—   
chr19_40750917_G_Tchr19:407509170.197-0.0100.337—   
chr19_40751017_A_Cchr19:407510170.0360.0650.337—   
chr19_40750916_A_Tchr19:407509160.0720.0910.315—   
chr19_40798087_G_Tchr19:407980870.1800.1740.101—   
chr19_40750976_C_Achr19:40750976-0.089-0.058-0.292—   
chr19_40751015_G_Cchr19:40751015-0.0160.0500.292—   
chr19_40751061_T_Achr19:407510610.1690.0600.067—   
chr19_40750988_C_Gchr19:40750988-0.075-0.018-0.281—   
chr19_40751024_C_Achr19:40751024-0.049-0.086-0.281—   
chr19_40751063_C_Achr19:407510630.1640.0710.011—   
chr19_40751144_G_Tchr19:40751144-0.126-0.063-0.281—   
chr19_40750939_T_Achr19:40750939-0.161-0.171-0.169—   
chr19_40751146_T_Achr19:40751146-0.154-0.020-0.157—   
chr19_40750921_T_Achr19:407509210.111-0.071-0.258—   
chr19_40751089_T_Gchr19:40751089-0.0430.0730.258—   
chr19_40751144_G_Achr19:40751144-0.079-0.033-0.258—   
chr19_40751145_C_Achr19:40751145-0.149-0.068-0.202—   
chr19_40750916_A_Cchr19:407509160.0720.0100.247—   
chr19_40750924_G_Achr19:407509240.059-0.065-0.236—   
chr19_40750938_G_Achr19:40750938-0.046-0.116-0.236—   
chr19_40750957_A_Cchr19:407509570.0230.0200.236—   
chr19_40751020_C_Achr19:40751020-0.039-0.098-0.236—   
chr19_40751039_C_Achr19:40751039-0.030-0.065-0.236—   
chr19_40751084_G_Tchr19:40751084-0.056-0.063-0.236—   
chr19_40750962_C_Achr19:407509620.1340.0730.056—   
chr19_40750919_A_Cchr19:407509190.0030.0860.225—   
chr19_40750927_C_Tchr19:407509270.023-0.060-0.225—   
chr19_40750940_A_Tchr19:407509400.1310.0550.000—   
chr19_40750972_C_Achr19:40750972-0.052-0.010-0.225—   
chr19_40751055_C_Tchr19:40751055-0.059-0.043-0.225—   
chr19_40751077_A_Tchr19:407510770.011-0.098-0.225—   
chr19_40798072_A_Cchr19:40798072-0.0180.1130.225—   
chr19_40751100_C_Achr19:40751100-0.130-0.101-0.079—   
chr19_40798066_C_Gchr19:407980660.1300.0780.034—   
chr19_40798076_T_Achr19:407980760.1300.1310.079—   
chr19_40750949_T_Achr19:40750949-0.128-0.025-0.135—   
chr19_40798014_G_Cchr19:40798014-0.125-0.111-0.219—   
chr19_40750935_A_Tchr19:407509350.098-0.065-0.213—   
chr19_40750971_G_Achr19:407509710.0000.013-0.213—   
chr19_40751069_T_Achr19:40751069-0.013-0.050-0.213—   
chr19_40751085_G_Achr19:407510850.010-0.068-0.213—   
chr19_40751101_G_Cchr19:407511010.1230.0030.101—   
chr19_40750927_C_Gchr19:40750927-0.010-0.081-0.202—   
chr19_40750928_C_Achr19:40750928-0.118-0.101-0.146—   
chr19_40750960_A_Tchr19:407509600.0790.1810.202—   
chr19_40750972_C_Tchr19:40750972-0.023-0.003-0.202—   
chr19_40750981_C_Gchr19:40750981-0.056-0.048-0.202—   
chr19_40750987_G_Tchr19:40750987-0.026-0.028-0.202—   
chr19_40750999_T_Achr19:407509990.118-0.015-0.056—   
chr19_40751015_G_Tchr19:407510150.0100.0180.202—   
chr19_40751023_G_Cchr19:40751023-0.0300.0380.202—   
chr19_40751029_C_Gchr19:407510290.011-0.013-0.202—   
chr19_40751064_T_Cchr19:40751064-0.038-0.0730.202—   
chr19_40751110_G_Cchr19:407511100.0100.0530.202—   
chr19_40798051_A_Tchr19:407980510.1100.1610.202—   
chr19_40750949_T_Cchr19:40750949-0.115-0.0550.090—   
chr19_40751090_T_Achr19:407510900.1150.0760.169—   
chr19_40798049_C_Gchr19:40798049-0.115-0.068-0.090—   
chr19_40750942_C_Achr19:40750942-0.111-0.081-0.169—   
chr19_40750954_A_Tchr19:407509540.1110.0250.056—   
chr19_40750974_A_Cchr19:407509740.0490.0150.191—   
chr19_40750981_C_Tchr19:40750981-0.016-0.048-0.191—   
chr19_40750997_C_Tchr19:407509970.003-0.030-0.191—   
chr19_40751031_A_Gchr19:40751031-0.039-0.010-0.191—   
chr19_40751089_T_Cchr19:40751089-0.0110.0860.191—   
chr19_40751145_C_Tchr19:40751145-0.111-0.013-0.146—   
chr19_40798058_T_Gchr19:407980580.1100.1060.101—   
chr19_40750934_G_Cchr19:407509340.1080.0860.146—   
chr19_40750950_G_Achr19:40750950-0.108-0.020-0.011—   
chr19_40750951_C_Achr19:40750951-0.1080.000-0.011—   
chr19_40750951_C_Gchr19:40750951-0.108-0.0200.045—   
chr19_40751079_A_Gchr19:407510790.108-0.053-0.180—   
chr19_40798085_G_Tchr19:40798085-0.108-0.098-0.146—   
chr19_40751123_A_Tchr19:40751123-0.107-0.275-0.101—   
chr19_40750916_A_Gchr19:40750916-0.0160.0050.180—   
chr19_40750939_T_Gchr19:40750939-0.105-0.176-0.112—   
chr19_40750952_A_Gchr19:40750952-0.105-0.0350.090—   
chr19_40750961_T_Cchr19:40750961-0.105-0.0500.022—   
chr19_40750966_G_Tchr19:407509660.1050.000-0.022—   
chr19_40750983_C_Tchr19:40750983-0.016-0.030-0.180—   
chr19_40750996_C_Tchr19:40750996-0.003-0.008-0.180—   
chr19_40751032_G_Tchr19:40751032-0.0030.005-0.180—   
chr19_40751036_A_Cchr19:40751036-0.0030.010-0.180—   
chr19_40751049_C_Tchr19:40751049-0.049-0.101-0.180—   
chr19_40751052_G_Tchr19:40751052-0.072-0.088-0.180—   
chr19_40751077_A_Gchr19:407510770.010-0.123-0.180—   
chr19_40751078_C_Gchr19:407510780.102-0.181-0.180—   
chr19_40751088_T_Cchr19:40751088-0.0410.0600.180—   
chr19_40751091_T_Gchr19:407510910.0150.0580.180—   
chr19_40750950_G_Tchr19:40750950-0.1020.0200.101—   
chr19_40750976_C_Gchr19:40750976-0.102-0.033-0.124—   
chr19_40751142_G_Tchr19:407511420.102-0.0030.101—   
chr19_40798082_A_Cchr19:40798082-0.102-0.058-0.022—   
chr19_40751053_T_Cchr19:407510530.100-0.055-0.011—   
chr19_40751121_C_Achr19:40751121-0.100-0.217-0.135—   
chr19_40750918_A_Cchr19:407509180.089-0.0050.169—   
chr19_40750923_C_Tchr19:407509230.0980.0500.045—   
chr19_40750924_G_Tchr19:407509240.098-0.005-0.056—   
chr19_40750932_C_Achr19:407509320.023-0.065-0.169—   
chr19_40750933_G_Cchr19:407509330.0260.0200.169—   
chr19_40750942_C_Gchr19:40750942-0.072-0.171-0.169—   
chr19_40750950_G_Cchr19:40750950-0.0890.0050.169—   
chr19_40750975_G_Achr19:40750975-0.026-0.015-0.169—   
chr19_40750987_G_Achr19:40750987-0.039-0.020-0.169—   
chr19_40750988_C_Achr19:40750988-0.016-0.008-0.169—   
chr19_40750999_T_Gchr19:407509990.056-0.0080.169—   
chr19_40751035_C_Achr19:407510350.0110.008-0.169—   
chr19_40751035_C_Gchr19:40751035-0.015-0.003-0.169—   
chr19_40751064_T_Gchr19:40751064-0.0250.0430.169—   
chr19_40751085_G_Cchr19:407510850.025-0.073-0.169—   
chr19_40751092_C_Gchr19:407510920.0020.0350.169—   
chr19_40751118_G_Cchr19:407511180.0440.0450.169—   
chr19_40751139_A_Tchr19:407511390.028-0.0300.169—   
chr19_40798057_A_Tchr19:407980570.0980.0880.067—   
chr19_40798078_G_Tchr19:40798078-0.064-0.078-0.169—   
chr19_40751121_C_Tchr19:40751121-0.097-0.222-0.101—   
chr19_40798050_T_Gchr19:40798050-0.097-0.0710.011—   
chr19_40750963_G_Tchr19:407509630.0950.0100.090—   
chr19_40798081_A_Cchr19:407980810.0950.0910.056—   
chr19_40751065_A_Tchr19:40751065-0.093-0.033-0.022—   
chr19_40798057_A_Cchr19:407980570.0930.0910.135—   
chr19_40750917_G_Cchr19:407509170.0030.0150.157—   
chr19_40750918_A_Gchr19:40750918-0.016-0.0150.157—   
chr19_40750938_G_Cchr19:40750938-0.026-0.151-0.157—   
chr19_40750941_A_Cchr19:40750941-0.092-0.121-0.022—   
chr19_40750953_A_Cchr19:407509530.0330.0350.157—   
chr19_40750960_A_Cchr19:40750960-0.0920.0050.112—   
chr19_40750975_G_Tchr19:407509750.010-0.023-0.157—   
chr19_40750983_C_Achr19:40750983-0.049-0.043-0.157—   
chr19_40750986_G_Achr19:407509860.0200.000-0.157—   
chr19_40750986_G_Tchr19:40750986-0.0130.008-0.157—   
chr19_40751015_G_Achr19:40751015-0.043-0.008-0.157—   
chr19_40751020_C_Tchr19:40751020-0.031-0.050-0.157—   
chr19_40751051_T_Gchr19:40751051-0.048-0.118-0.157—   
chr19_40751084_G_Cchr19:407510840.000-0.038-0.157—   
chr19_40751088_T_Gchr19:40751088-0.0030.0580.157—   
chr19_40751089_T_Achr19:40751089-0.0020.0780.157—   
chr19_40751104_C_Gchr19:40751104-0.043-0.078-0.157—   
chr19_40751104_C_Tchr19:40751104-0.069-0.076-0.157—   
chr19_40751110_G_Tchr19:40751110-0.0080.0550.157—   
chr19_40751119_G_Tchr19:40751119-0.048-0.131-0.157—   
chr19_40751121_C_Gchr19:40751121-0.092-0.214-0.157—   
chr19_40797999_A_Cchr19:407979990.0360.0430.157—   
chr19_40798033_T_Gchr19:40798033-0.092-0.018-0.022—   
chr19_40750949_T_Gchr19:40750949-0.0890.0760.079—   
chr19_40750970_G_Cchr19:407509700.0890.0000.146—   
chr19_40751088_T_Achr19:407510880.0890.0860.146—   
chr19_40751055_C_Achr19:40751055-0.0870.020-0.045—   
chr19_40751146_T_Cchr19:407511460.0870.013-0.056—   
chr19_40798056_C_Gchr19:40798056-0.087-0.050-0.124—   
chr19_40750958_C_Achr19:407509580.0100.015-0.146—   
chr19_40750964_G_Achr19:407509640.0030.0200.146—   
chr19_40750994_G_Cchr19:407509940.0690.0400.146—   
chr19_40751018_A_Cchr19:407510180.0130.0380.146—   
chr19_40751030_G_Achr19:407510300.0620.0780.146—   
chr19_40751050_C_Tchr19:40751050-0.034-0.015-0.146—   
chr19_40751086_T_Achr19:40751086-0.008-0.076-0.146—   
chr19_40751091_T_Cchr19:40751091-0.008-0.0300.146—   
chr19_40751097_G_Tchr19:40751097-0.0280.1030.146—   
chr19_40751100_C_Gchr19:40751100-0.082-0.050-0.146—   
chr19_40751122_A_Tchr19:40751122-0.085-0.0880.000—   
chr19_40751132_G_Tchr19:40751132-0.002-0.035-0.146—   
chr19_40798031_G_Tchr19:40798031-0.044-0.053-0.146—   
chr19_40751123_A_Cchr19:40751123-0.084-0.229-0.011—   
chr19_40750954_A_Cchr19:407509540.0820.020-0.045—   
chr19_40750995_G_Achr19:407509950.0820.030-0.124—   
chr19_40751047_G_Tchr19:407510470.0820.0710.112—   
chr19_40751048_A_Cchr19:40751048-0.082-0.0080.045—   
chr19_40751136_T_Gchr19:407511360.0820.008-0.011—   
chr19_40798039_C_Gchr19:40798039-0.082-0.043-0.011—   
chr19_40798080_C_Gchr19:40798080-0.082-0.081-0.090—   
chr19_40798082_A_Tchr19:40798082-0.082-0.063-0.101—   
chr19_40751060_T_Achr19:407510600.0800.005-0.090—   
chr19_40798017_C_Tchr19:407980170.0800.0600.000—   
chr19_40798075_C_Gchr19:40798075-0.080-0.068-0.034—   
chr19_40798078_G_Cchr19:40798078-0.080-0.086-0.011—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.