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CYP2C19

receptor: PXRTier 1

Drug substrates

clopidogrel (activation); voriconazole; omeprazole; escitalopram

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated induction of CYP2C19 lowers antiplatelet effect of the prodrug clopidogrel, and raises exposure of voriconazole.

Affected substrate drugs (PharmGKB): clopidogrel; voriconazole; omeprazole; lansoprazole; citalopram; escitalopram

Scored variants near CYP2C19

chr10:94,662,680..94,955,547, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr10_94673779_C_Achr10:946737790.2910.3300.246—   
chr10_94673775_A_Gchr10:946737750.0430.1260.506—   
chr10_94673794_C_Gchr10:946737940.2200.2910.497—   
chr10_94673789_G_Tchr10:946737890.1420.2970.491—   
chr10_94673789_G_Achr10:946737890.2680.3320.102—   
chr10_94673793_T_Achr10:946737930.2550.3890.357—   
chr10_94673773_T_Achr10:94673773-0.227-0.168-0.433—   
chr10_94673778_T_Achr10:946737780.2240.2410.222—   
chr10_94673794_C_Tchr10:946737940.2100.3060.386—   
chr10_94673773_T_Gchr10:94673773-0.206-0.137-0.383—   
chr10_94673773_T_Cchr10:94673773-0.198-0.144-0.368—   
chr10_94673780_A_Cchr10:94673780-0.123-0.067-0.368—   
chr10_94673793_T_Gchr10:946737930.1950.3140.269—   
chr10_94673743_C_Gchr10:946737430.1890.3650.228—   
chr10_94673731_C_Tchr10:946737310.1830.1730.292—   
chr10_94673780_A_Tchr10:94673780-0.086-0.064-0.316<0.001%
chr10_94673774_T_Cchr10:94673774-0.115-0.093-0.313—   
chr10_94673775_A_Cchr10:94673775-0.138-0.099-0.313—   
chr10_94673794_C_Achr10:946737940.1560.2300.228—   
chr10_94673779_C_Gchr10:94673779-0.0840.001-0.275—   
chr10_94673782_C_Gchr10:94673782-0.096-0.084-0.275—   
chr10_94673774_T_Achr10:94673774-0.022-0.065-0.266—   
chr10_94673780_A_Gchr10:94673780-0.075-0.057-0.246—   
chr10_94673788_T_Achr10:94673788-0.0560.029-0.243—   
chr10_94673792_A_Cchr10:946737920.1330.1890.216—   
chr10_94673776_C_Tchr10:94673776-0.065-0.043-0.234—   
chr10_94673790_A_Gchr10:946737900.1320.2050.076—   
chr10_94673741_A_Cchr10:946737410.1300.2040.219—   
chr10_94673686_C_Tchr10:946736860.1290.1420.219—   
chr10_94673737_T_Achr10:94673737-0.108-0.067-0.2250.011%
chr10_94673778_T_Gchr10:94673778-0.047-0.005-0.222—   
chr10_94673731_C_Achr10:946737310.1130.1170.216—   
chr10_94673742_T_Achr10:94673742-0.092-0.037-0.216—   
chr10_94673776_C_Achr10:94673776-0.074-0.033-0.213—   
chr10_94673779_C_Tchr10:94673779-0.104-0.015-0.213—   
chr10_94673774_T_Gchr10:94673774-0.100-0.136-0.211—   
chr10_94673742_T_Cchr10:94673742-0.095-0.063-0.208—   
chr10_94673776_C_Gchr10:94673776-0.064-0.060-0.208—   
chr10_94673757_A_Tchr10:94673757-0.116-0.073-0.126—   
chr10_94673744_A_Cchr10:94673744-0.075-0.048-0.202—   
chr10_94673744_A_Tchr10:94673744-0.064-0.038-0.202—   
chr10_94673793_T_Cchr10:946737930.1140.2000.076—   
chr10_94673717_C_Gchr10:946737170.0620.0820.199—   
chr10_94673731_C_Gchr10:946737310.0960.1100.199—   
chr10_94673757_A_Gchr10:94673757-0.111-0.110-0.135—   
chr10_94673730_T_Gchr10:946737300.0500.0640.196—   
chr10_94673817_T_Achr10:946738170.1100.1450.073—   
chr10_94673795_A_Cchr10:94673795-0.0260.028-0.193—   
chr10_94673699_A_Tchr10:946736990.1090.1550.149—   
chr10_94673818_T_Achr10:946738180.0130.0180.190—   
chr10_94673709_A_Cchr10:946737090.1070.1060.187—   
chr10_94673766_C_Achr10:94673766-0.051-0.058-0.187—   
chr10_94673785_A_Cchr10:94673785-0.105-0.123-0.135—   
chr10_94673791_C_Achr10:946737910.1050.1790.096—   
chr10_94673790_A_Tchr10:946737900.1040.1710.184—   
chr10_94673808_A_Gchr10:946738080.0790.0810.184—   
chr10_94673742_T_Gchr10:94673742-0.079-0.040-0.181—   
chr10_94673826_A_Cchr10:94673826-0.044-0.034-0.181—   
chr10_94673777_A_Gchr10:94673777-0.102-0.128-0.123—   
chr10_94673738_G_Cchr10:94673738-0.071-0.025-0.178—   
chr10_94673743_C_Achr10:946737430.1000.1510.102—   
chr10_94673739_A_Gchr10:94673739-0.084-0.044-0.173—   
chr10_94673763_C_Tchr10:94673763-0.096-0.0180.161—   
chr10_94673772_A_Tchr10:94673772-0.046-0.020-0.170—   
chr10_94673782_C_Achr10:94673782-0.019-0.031-0.170—   
chr10_94673824_T_Gchr10:946738240.0950.1590.094—   
chr10_94673775_A_Tchr10:946737750.0890.1340.167—   
chr10_94673802_T_Gchr10:946738020.0740.0840.167—   
chr10_94673826_A_Tchr10:94673826-0.035-0.011-0.167—   
chr10_94673787_A_Cchr10:946737870.0920.1500.020—   
chr10_94673788_T_Gchr10:946737880.0020.098-0.161—   
chr10_94673825_G_Tchr10:946738250.0900.1160.079—   
chr10_94673754_A_Gchr10:946737540.0390.0380.158—   
chr10_94673777_A_Cchr10:94673777-0.084-0.053-0.158—   
chr10_94673788_T_Cchr10:94673788-0.0340.039-0.158<0.001%
chr10_94673813_A_Gchr10:946738130.0180.0190.158—   
chr10_94673818_T_Gchr10:94673818-0.0090.0090.158—   
chr10_94673716_A_Cchr10:94673716-0.078-0.076-0.155—   
chr10_94673746_C_Achr10:94673746-0.071-0.065-0.155—   
chr10_94673791_C_Gchr10:946737910.0880.1080.129—   
chr10_94673828_T_Gchr10:946738280.035-0.0600.155—   
chr10_94673791_C_Tchr10:946737910.0850.1150.050—   
chr10_94673717_C_Achr10:946737170.0620.0650.146—   
chr10_94673739_A_Cchr10:94673739-0.065-0.028-0.146—   
chr10_94673740_C_Achr10:94673740-0.065-0.009-0.146—   
chr10_94673781_C_Achr10:94673781-0.034-0.010-0.146—   
chr10_94673814_T_Achr10:94673814-0.0100.0140.1460.0053%
chr10_94673831_A_Tchr10:94673831-0.043-0.039-0.146—   
chr10_94673722_A_Tchr10:946737220.0680.0940.140—   
chr10_94673787_A_Tchr10:946737870.0020.063-0.140—   
chr10_94673725_C_Gchr10:94673725-0.078-0.093-0.111—   
chr10_94673737_T_Gchr10:94673737-0.0540.003-0.135—   
chr10_94673795_A_Tchr10:946737950.0230.076-0.135—   
chr10_94673738_G_Tchr10:946737380.0590.1070.132—   
chr10_94673741_A_Gchr10:946737410.063-0.0240.132—   
chr10_94673797_T_Cchr10:946737970.0190.0140.132—   
chr10_94673809_C_Tchr10:946738090.0750.0420.099—   
chr10_94673755_G_Tchr10:94673755-0.074-0.084-0.123—   
chr10_94673681_A_Cchr10:94673681-0.058-0.059-0.129—   
chr10_94673765_G_Cchr10:94673765-0.061-0.037-0.129—   
chr10_94673745_C_Tchr10:946737450.0650.0290.126<0.001%
chr10_94673753_C_Achr10:94673753-0.071-0.077-0.114—   
chr10_94673831_A_Cchr10:94673831-0.057-0.074-0.126—   
chr10_94673762_A_Gchr10:94673762-0.070-0.084-0.079—   
chr10_94673767_T_Gchr10:94673767-0.070-0.058-0.099—   
chr10_94673797_T_Gchr10:94673797-0.070-0.059-0.114—   
chr10_94673748_T_Cchr10:946737480.003-0.0090.123—   
chr10_94673783_T_Cchr10:946737830.0380.0250.123—   
chr10_94673789_G_Cchr10:946737890.0310.106-0.123—   
chr10_94673714_A_Gchr10:94673714-0.068-0.082-0.091—   
chr10_94673673_G_Tchr10:946736730.0540.0710.120—   
chr10_94673737_T_Cchr10:94673737-0.058-0.031-0.120<0.001%
chr10_94673743_C_Tchr10:94673743-0.0380.020-0.120—   
chr10_94673765_G_Tchr10:94673765-0.048-0.031-0.120—   
chr10_94673836_T_Cchr10:946738360.0670.0340.070—   
chr10_94673716_A_Gchr10:94673716-0.067-0.081-0.064—   
chr10_94673701_G_Cchr10:94673701-0.046-0.055-0.117—   
chr10_94673746_C_Gchr10:94673746-0.058-0.055-0.117—   
chr10_94673747_T_Cchr10:946737470.011-0.0200.117—   
chr10_94673772_A_Cchr10:94673772-0.048-0.038-0.117—   
chr10_94673778_T_Cchr10:946737780.0660.078-0.018—   
chr10_94673824_T_Achr10:94673824-0.0210.006-0.117—   
chr10_94673707_A_Gchr10:946737070.0480.0620.114—   
chr10_94673797_T_Achr10:94673797-0.058-0.039-0.114—   
chr10_94673827_C_Achr10:94673827-0.0240.019-0.114—   
chr10_94673810_C_Gchr10:94673810-0.064-0.055-0.070—   
chr10_94673790_A_Cchr10:946737900.0630.122-0.023—   
chr10_94673817_T_Gchr10:946738170.0410.0590.111—   
chr10_94673832_C_Achr10:94673832-0.0150.006-0.111—   
chr10_94673804_C_Gchr10:94673804-0.062-0.034-0.056—   
chr10_94673808_A_Tchr10:946738080.0620.0690.099—   
chr10_94673714_A_Cchr10:94673714-0.062-0.081-0.091—   
chr10_94673723_T_Cchr10:946737230.0610.0820.096—   
chr10_94673785_A_Tchr10:94673785-0.061-0.067-0.038—   
chr10_94673826_A_Gchr10:94673826-0.0230.003-0.108—   
chr10_94673675_A_Tchr10:946736750.0600.0710.053—   
chr10_94673624_C_Tchr10:946736240.0560.0820.105—   
chr10_94673749_G_Tchr10:946737490.0420.0720.105—   
chr10_94673762_A_Tchr10:94673762-0.055-0.064-0.105—   
chr10_94673792_A_Tchr10:946737920.0330.0930.105—   
chr10_94673813_A_Tchr10:946738130.0370.0530.105—   
chr10_94673729_A_Cchr10:94673729-0.059-0.057-0.041—   
chr10_94673693_A_Cchr10:946736930.0590.0590.102—   
chr10_94673806_A_Gchr10:946738060.0590.0650.073—   
chr10_94673782_C_Tchr10:94673782-0.013-0.021-0.102<0.001%
chr10_94673801_G_Achr10:94673801-0.033-0.045-0.102—   
chr10_94673795_A_Gchr10:946737950.0570.086-0.015—   
chr10_94673836_T_Gchr10:946738360.0570.0400.067—   
chr10_94673657_C_Achr10:946736570.0570.0740.099—   
chr10_94673719_A_Gchr10:946737190.0230.0300.099—   
chr10_94673728_C_Gchr10:946737280.0490.0550.099—   
chr10_94673745_C_Gchr10:946737450.0310.0400.099—   
chr10_94673812_A_Cchr10:94673812-0.055-0.042-0.073—   
chr10_94673679_C_Achr10:946736790.0350.0390.096—   
chr10_94673710_A_Tchr10:94673710-0.022-0.030-0.096—   
chr10_94673730_T_Cchr10:946737300.0110.0210.096—   
chr10_94673740_C_Tchr10:94673740-0.0120.015-0.096—   
chr10_94673768_G_Tchr10:94673768-0.031-0.026-0.096—   
chr10_94673796_C_Tchr10:946737960.0250.0160.096<0.001%
chr10_94673811_T_Cchr10:94673811-0.054-0.052-0.096—   
chr10_94673815_C_Tchr10:946738150.0360.0570.096—   
chr10_94673752_C_Achr10:946737520.0540.0500.035—   
chr10_94673724_C_Gchr10:94673724-0.038-0.057-0.094—   
chr10_94673754_A_Cchr10:946737540.0320.0260.094—   
chr10_94673765_G_Achr10:94673765-0.026-0.031-0.094—   
chr10_94673824_T_Cchr10:94673824-0.026-0.015-0.094<0.001%
chr10_94673827_C_Tchr10:94673827-0.0310.000-0.094—   
chr10_94673834_C_Achr10:94673834-0.026-0.024-0.094—   
chr10_94673729_A_Gchr10:946737290.0170.0340.091—   
chr10_94673750_G_Cchr10:94673750-0.030-0.0100.091—   
chr10_94673762_A_Cchr10:94673762-0.051-0.060-0.050—   
chr10_94673766_C_Tchr10:94673766-0.012-0.018-0.091—   
chr10_94673817_T_Cchr10:946738170.0270.0400.0910.0013%
chr10_94673827_C_Gchr10:94673827-0.026-0.003-0.091—   
chr10_94707948_A_Cchr10:947079480.0350.0500.091<0.001%
chr10_94673686_C_Gchr10:946736860.0500.0470.064—   
chr10_94673697_G_Achr10:94673697-0.033-0.052-0.088—   
chr10_94673727_A_Cchr10:94673727-0.050-0.053-0.088—   
chr10_94673733_C_Gchr10:946737330.0090.0180.088—   
chr10_94673747_T_Gchr10:94673747-0.007-0.0430.088—   
chr10_94673771_G_Tchr10:94673771-0.050-0.024-0.067—   
chr10_94673783_T_Gchr10:94673783-0.032-0.053-0.088—   
chr10_94673786_G_Achr10:94673786-0.046-0.020-0.088—   
chr10_94673786_G_Tchr10:94673786-0.027-0.018-0.088—   
chr10_94673833_C_Gchr10:94673833-0.047-0.034-0.088—   
chr10_94673755_G_Cchr10:94673755-0.049-0.0490.044—   
chr10_94673663_T_Gchr10:946736630.0480.0490.082—   
chr10_94673681_A_Tchr10:94673681-0.046-0.043-0.085—   
chr10_94673714_A_Tchr10:94673714-0.038-0.045-0.085—   
chr10_94673802_T_Achr10:94673802-0.048-0.037-0.056—   
chr10_94673825_G_Achr10:946738250.0470.097-0.056—   
chr10_94673623_G_Tchr10:94673623-0.007-0.013-0.082—   
chr10_94673679_C_Tchr10:946736790.0360.0350.082—   
chr10_94673825_G_Cchr10:946738250.0090.050-0.082—   
chr10_94673705_T_Cchr10:94673705-0.046-0.055-0.079—   
chr10_94673771_G_Achr10:94673771-0.0460.015-0.003—   
chr10_94673747_T_Achr10:94673747-0.045-0.076-0.018—   
chr10_94673643_G_Achr10:94673643-0.022-0.026-0.0790.0026%
chr10_94673669_A_Gchr10:946736690.0050.0180.079—   
chr10_94673674_A_Cchr10:946736740.0110.0240.079—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.