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CYP8B1

receptor: FXRTier 1

Drug substrates

bile-acid pool composition

refs: 25198545

CAMIP causal chains

FXR

Altered receptor-mediated feedback repression of CYP8B1, shifting the cholic acid to chenodeoxycholic acid synthesis ratio in endogenous bile acid pathways.

Affected substrate drugs (PharmGKB): none in routine clinical use, endogenous or bile acid pathway

Scored variants near CYP8B1

chr3:42,772,191..42,975,879, gene body plus 100 kb. Showing the strongest 200 by effect size.

VariantPosition PXR FXR AhR AF
chr3_42804558_A_Tchr3:4280455823,4247,58415,1046.6e-6
chr3_42804607_T_Cchr3:4280460722,720-4,35211,008—   
chr3_42804709_G_Cchr3:4280470922,3364,5448,960—   
chr3_42804710_G_Achr3:4280471020,1604,6087,680—   
chr3_42804609_G_Achr3:4280460919,712-2,46412,544—   
chr3_42804708_G_Cchr3:4280470819,5843,8086,656—   
chr3_42804609_G_Cchr3:4280460918,688-3,32811,776—   
chr3_42804709_G_Achr3:4280470918,6242,5602,5601.1e-4
chr3_42804709_G_Tchr3:4280470918,3043,8087,168—   
chr3_42804532_A_Gchr3:4280453217,984-2,4008,448—   
chr3_42804703_T_Gchr3:4280470317,9205,63225,600—   
chr3_42804708_G_Achr3:4280470817,9203,6803,8406.6e-6
chr3_42804707_G_Achr3:4280470717,4724,4488,1922.0e-5
chr3_42804625_C_Achr3:42804625-17,024352-7,168—   
chr3_42804609_G_Tchr3:4280460916,704-4,1927,936—   
chr3_42804707_G_Cchr3:4280470716,7044,99211,008—   
chr3_42804710_G_Cchr3:4280471016,3203,96810,496—   
chr3_42804605_A_Cchr3:4280460516,256-4,06412,288—   
chr3_42804607_T_Gchr3:4280460715,936-3,80811,520—   
chr3_42804576_C_Gchr3:4280457615,488576512—   
chr3_42804708_G_Tchr3:4280470815,4883,8085,888—   
chr3_42804606_T_Cchr3:4280460615,360-3,26412,288—   
chr3_42804707_G_Tchr3:4280470714,9763,0726,400—   
chr3_42804611_T_Achr3:4280461113,568-7367,936—   
chr3_42804530_C_Achr3:4280453012,992-5,2161,792—   
chr3_42804635_A_Gchr3:4280463512,2242,8483,328—   
chr3_42804612_G_Tchr3:4280461211,776-5128,192—   
chr3_42804531_C_Tchr3:4280453111,648-3,3604,864—   
chr3_42804711_C_Achr3:4280471111,6482,6885,376—   
chr3_42804593_A_Gchr3:4280459310,880-1,9844,608—   
chr3_42804608_G_Achr3:4280460810,880-3,32810,752—   
chr3_42804687_G_Cchr3:4280468710,8162,0801,536—   
chr3_42804534_T_Gchr3:4280453410,752-4,7045,888—   
chr3_42804756_T_Gchr3:4280475610,6883,4247,680—   
chr3_42804605_A_Tchr3:4280460510,624-4,1288,448—   
chr3_42804532_A_Cchr3:4280453210,432-4,2245,120—   
chr3_42804606_T_Gchr3:4280460610,304-3,8408,960—   
chr3_42804711_C_Tchr3:4280471110,3042,8803,840—   
chr3_42804606_T_Achr3:4280460610,240-4,57610,240—   
chr3_42804757_C_Gchr3:4280475710,1764,0965,888—   
chr3_42804566_G_Achr3:4280456610,112-1,1209,9841.3e-5
chr3_42804517_A_Cchr3:428045179,920-32-256—   
chr3_42804559_C_Achr3:42804559-9,728-416-5,632—   
chr3_42804692_C_Achr3:428046929,6001,98411,008—   
chr3_42804528_A_Tchr3:42804528-9,472-7042,304—   
chr3_42804604_G_Cchr3:428046049,408-2,1767,936—   
chr3_42804630_C_Achr3:428046309,4082,368768—   
chr3_42804706_A_Tchr3:428047069,4082,2405,376—   
chr3_42804616_C_Achr3:428046169,3443,61610,240—   
chr3_42804608_G_Cchr3:428046089,280-3,9364,864—   
chr3_42804711_C_Gchr3:428047119,2162,8163,328—   
chr3_42804628_G_Achr3:428046288,8963,1368,960—   
chr3_42804534_T_Achr3:428045348,896-2,8484,352—   
chr3_42804726_C_Achr3:428047268,8962,5925,376—   
chr3_42804529_G_Cchr3:42804529-8,832-3,904-5,888—   
chr3_42804530_C_Gchr3:428045308,768-2,5604,352—   
chr3_42804560_G_Tchr3:428045608,7688965,376—   
chr3_42804706_A_Cchr3:428047068,7041,3443,840—   
chr3_42804603_G_Achr3:428046038,640-1,6643,328—   
chr3_42804621_A_Gchr3:42804621-8,6404163,328—   
chr3_42804605_A_Gchr3:428046058,384-2,9128,448—   
chr3_42804516_C_Gchr3:42804516-8,384512256—   
chr3_42804625_C_Gchr3:42804625-8,256672-1,0241.0e-3
chr3_42804634_T_Gchr3:428046348,1922,1767,168—   
chr3_42804846_T_Gchr3:428048468,1287368,704—   
chr3_42804652_C_Tchr3:42804652-8,1282,816-3,840—   
chr3_42804627_G_Cchr3:42804627-7,936-224-6,144—   
chr3_42804562_G_Achr3:42804562-7,8081,024-12,288—   
chr3_42804633_C_Gchr3:428046337,6805441,792—   
chr3_42804551_C_Gchr3:42804551-7,616-963,328—   
chr3_42804660_G_Achr3:42804660-7,6162,2403,0721.3e-5
chr3_42804604_G_Achr3:428046047,552-3,0406,912—   
chr3_42804611_T_Cchr3:428046117,424-1,2802,8166.6e-6
chr3_42804649_G_Cchr3:42804649-7,3601,312-2,816—   
chr3_42804633_C_Achr3:428046337,2961,2804,096—   
chr3_42804631_C_Tchr3:428046317,2325124,608—   
chr3_42804577_G_Achr3:428045777,1683,61614,3366.6e-6
chr3_42804520_G_Tchr3:42804520-7,168-384-4,352—   
chr3_42804594_G_Cchr3:428045947,1681923,584—   
chr3_42804612_G_Cchr3:428046127,168-9924,096—   
chr3_42804623_T_Gchr3:42804623-7,040288-7,680—   
chr3_42804594_G_Tchr3:428045947,0404162,560—   
chr3_42804705_G_Achr3:428047057,0401,4721,024—   
chr3_42804568_G_Cchr3:42804568-6,912-256-7,936—   
chr3_42804565_C_Achr3:428045656,9127363,072—   
chr3_42804604_G_Tchr3:428046046,912-2,2725,888—   
chr3_42804556_G_Tchr3:42804556-6,7202,0800—   
chr3_42804666_C_Gchr3:428046666,720-5121,536—   
chr3_42804687_G_Achr3:428046876,5281,024-7685.9e-4
chr3_42804732_C_Tchr3:428047326,4641,3762,560—   
chr3_42804611_T_Gchr3:428046116,400-2,0801,024—   
chr3_42804541_C_Tchr3:428045416,3363,1362,816—   
chr3_42804575_G_Tchr3:42804575-6,3361,056512—   
chr3_42804550_G_Achr3:428045506,2083526,656—   
chr3_42804712_T_Gchr3:428047126,2088966,400—   
chr3_42804584_G_Cchr3:42804584-6,208-928-256—   
chr3_42804758_C_Achr3:428047586,2083,0083,072—   
chr3_42804529_G_Tchr3:42804529-6,144-928-2,560—   
chr3_42804567_T_Gchr3:428045676,144-1,4402,560—   
chr3_42804613_G_Tchr3:428046136,1441600—   
chr3_42804698_G_Cchr3:428046986,1443,0405,120—   
chr3_42804559_C_Tchr3:42804559-5,952-1,152-6,144—   
chr3_42804550_G_Tchr3:428045505,9521,7925,376—   
chr3_42804607_T_Achr3:428046075,952-1,2163,072—   
chr3_42804618_G_Tchr3:42804618-5,9521,344-4,608—   
chr3_42804722_G_Tchr3:428047225,9521,9845,120—   
chr3_42804620_G_Cchr3:428046205,888328,192—   
chr3_42804712_T_Achr3:428047125,8881,7286,400—   
chr3_42804553_A_Tchr3:428045535,8881,1203,584—   
chr3_42804757_C_Achr3:428047575,8242,4323,8406.6e-6
chr3_42804559_C_Gchr3:42804559-5,760-2,272-11,776—   
chr3_42804696_C_Achr3:428046965,7602,1762,304—   
chr3_42804712_T_Cchr3:428047125,7601,7605,632—   
chr3_42804537_G_Tchr3:42804537-5,632-864-3,072—   
chr3_42804706_A_Gchr3:42804706-5,632-1,824-3,584—   
chr3_42804745_T_Achr3:428047455,6321,7602,304—   
chr3_42804705_G_Cchr3:428047055,5681,056512—   
chr3_42804734_C_Tchr3:428047345,5682,7523,328—   
chr3_42804664_G_Cchr3:428046645,5041,56814,080—   
chr3_42804690_C_Achr3:428046905,5041,4401,024—   
chr3_42804699_G_Tchr3:428046995,5042,1125,376—   
chr3_42804576_C_Tchr3:42804576-5,4401,312-2,816—   
chr3_42804595_C_Gchr3:42804595-5,440-4482,560—   
chr3_42804608_G_Tchr3:428046085,440-3,7764,864—   
chr3_42804733_T_Achr3:428047335,3762,94410,240—   
chr3_42804734_C_Gchr3:428047345,3762,5925,888—   
chr3_42804564_G_Achr3:42804564-5,3761,728-4,096—   
chr3_42804630_C_Tchr3:428046305,3121,088-1,280—   
chr3_42804565_C_Tchr3:428045655,248-128-4,608—   
chr3_42804838_G_Tchr3:428048385,248-64-3,584—   
chr3_42804632_A_Tchr3:428046325,1841,088512—   
chr3_42804749_G_Cchr3:428047495,184384768—   
chr3_42804626_T_Cchr3:42804626-5,120672-4,096—   
chr3_42804833_G_Tchr3:428048334,992-896-9,984—   
chr3_42804717_C_Tchr3:42804717-4,928-1,376-2,304—   
chr3_42804843_G_Achr3:428048434,800-704-7,936—   
chr3_42804733_T_Gchr3:428047334,4802,0806,9126.6e-6
chr3_42804573_C_Tchr3:42804573-4,2881,6965,120—   
chr3_42804657_G_Cchr3:428046574,1601927,680—   
chr3_42804697_G_Tchr3:428046974,0321,4087,424—   
chr3_42804652_C_Achr3:42804652-3,840-3526,656—   
chr3_42804827_G_Tchr3:428048273,7122,56020,4801.3e-5
chr3_42804578_G_Tchr3:42804578-3,648-2889,728—   
chr3_42804691_G_Cchr3:42804691-3,648-544-6,400—   
chr3_42804553_A_Cchr3:428045533,6481,1525,376—   
chr3_42804700_C_Gchr3:42804700-3,520-1,920-5,120—   
chr3_42804651_A_Gchr3:428046513,392-4807,680—   
chr3_42804838_G_Cchr3:428048383,2008648,448—   
chr3_42804675_T_Achr3:428046753,2006085,120—   
chr3_42804556_G_Achr3:42804556-3,136-1,312-5,888—   
chr3_42804584_G_Tchr3:428045843,136-3525,632—   
chr3_42804700_C_Achr3:42804700-3,136-1,632-5,632—   
chr3_42804565_C_Gchr3:42804565-3,072-896-5,888—   
chr3_42804734_C_Achr3:428047343,0722,5605,120—   
chr3_42804577_G_Tchr3:428045772,9447686,912—   
chr3_42804667_G_Tchr3:42804667-2,944-1,056-5,632—   
chr3_42804557_G_Tchr3:42804557-2,752-128-7,424—   
chr3_42804580_T_Gchr3:428045802,624-32-8,192—   
chr3_42804563_T_Gchr3:42804563-2,560-1,120-8,704—   
chr3_42804775_C_Tchr3:428047752,560-768-7,168—   
chr3_42804629_C_Tchr3:428046292,496-1,984-5,376—   
chr3_42804816_G_Cchr3:428048162,4329928,192—   
chr3_42804660_G_Cchr3:428046602,3688968,448—   
chr3_42804578_G_Achr3:42804578-2,368-6408,1922.0e-5
chr3_42804703_T_Achr3:428047032,304965,120—   
chr3_42804578_G_Cchr3:42804578-2,240-57614,848—   
chr3_42804716_G_Tchr3:42804716-2,240-1,760-7,680—   
chr3_42804658_G_Cchr3:428046582,0481,3445,376—   
chr3_42804564_G_Cchr3:42804564-1,984-1,248-8,704—   
chr3_42804839_A_Cchr3:428048391,9207365,888—   
chr3_42804786_A_Cchr3:428047861,664-6405,376—   
chr3_42804643_T_Cchr3:42804643-1,6004166,400—   
chr3_42804825_C_Gchr3:42804825-1,600-384-5,632—   
chr3_42804646_A_Tchr3:428046461,5362,4965,120—   
chr3_42804824_A_Tchr3:42804824-1,536-320-5,120—   
chr3_42804669_G_Cchr3:42804669-1,4725,4409,2161.3e-5
chr3_42804663_A_Tchr3:42804663-1,4722,6247,6803.0e-4
chr3_42804840_T_Cchr3:428048401,1527365,120—   
chr3_42804610_C_Gchr3:42804610-960-4,12810,240—   
chr3_42804562_G_Cchr3:42804562-960-256-9,216—   
chr3_42804563_T_Achr3:42804563-896-1,760-8,704—   
chr3_42804580_T_Cchr3:42804580-896-1,376-6,400—   
chr3_42804811_C_Gchr3:42804811832-1926,912—   
chr3_42804819_G_Tchr3:42804819-832-320-6,400—   
chr3_42804658_G_Tchr3:42804658-8321,5045,632—   
chr3_42804847_G_Achr3:42804847768-1,120-10,496—   
chr3_42804664_G_Tchr3:42804664-7041,8886,144—   
chr3_42804751_C_Achr3:42804751704-1,376-6,144—   
chr3_42804821_C_Gchr3:428048217047046,1441.3e-5
chr3_42804564_G_Tchr3:42804564640-768-7,168—   
chr3_42804702_C_Achr3:42804702640-576-5,120—   
chr3_42804561_C_Achr3:42804561576256-5,376—   
chr3_42804560_G_Achr3:42804560512017,9206.6e-6
chr3_42804793_T_Gchr3:42804793448-768-6,144—   
chr3_42804840_T_Gchr3:42804840-3205125,376—   
chr3_42804557_G_Cchr3:42804557256-2888,704—   
chr3_42804752_C_Gchr3:42804752192-1,184-5,888—   
chr3_42804816_G_Tchr3:428048161921,0565,632—   
chr3_42804771_G_Tchr3:42804771-649285,120—   
chr3_42804815_G_Achr3:4280481564-160-5,1209.9e-5

Showing 200 of 200 in this window. Scores are the raw center bin Δ, ALT minus REF; click a column to sort.