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CYP8B1

receptor: FXRTier 1

Drug substrates

bile-acid pool composition

refs: 25198545

CAMIP causal chains

FXR

Altered receptor-mediated feedback repression of CYP8B1, shifting the cholic acid to chenodeoxycholic acid synthesis ratio in endogenous bile acid pathways.

Affected substrate drugs (PharmGKB): none in routine clinical use, endogenous or bile acid pathway

Scored variants near CYP8B1

chr3:42,772,191..42,975,879, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr3_42804703_T_Gchr3:428047030.4790.4571.000—   
chr3_42804558_A_Tchr3:428045580.6260.6160.721<0.001%
chr3_42804607_T_Cchr3:428046070.607-0.3530.525—   
chr3_42804709_G_Cchr3:428047090.5970.3690.427—   
chr3_42804827_G_Tchr3:428048270.0990.2080.9770.0013%
chr3_42804710_G_Achr3:428047100.5380.3740.366—   
chr3_42804609_G_Achr3:428046090.526-0.2000.598—   
chr3_42804708_G_Cchr3:428047080.5230.3090.318—   
chr3_42804609_G_Cchr3:428046090.499-0.2700.562—   
chr3_42804709_G_Achr3:428047090.4970.2080.1220.011%
chr3_42804709_G_Tchr3:428047090.4890.3090.342—   
chr3_42804532_A_Gchr3:428045320.480-0.1950.403—   
chr3_42804560_G_Achr3:428045600.0140.0000.855<0.001%
chr3_42804708_G_Achr3:428047080.4790.2990.183<0.001%
chr3_42804707_G_Achr3:428047070.4670.3610.3910.0020%
chr3_42804625_C_Achr3:42804625-0.4550.029-0.342—   
chr3_42804609_G_Tchr3:428046090.446-0.3400.379—   
chr3_42804707_G_Cchr3:428047070.4460.4050.525—   
chr3_42804710_G_Cchr3:428047100.4360.3220.501—   
chr3_42804605_A_Cchr3:428046050.434-0.3300.586—   
chr3_42804607_T_Gchr3:428046070.426-0.3090.550—   
chr3_42804576_C_Gchr3:428045760.4140.0470.024—   
chr3_42804708_G_Tchr3:428047080.4140.3090.281—   
chr3_42804606_T_Cchr3:428046060.410-0.2650.586—   
chr3_42804707_G_Tchr3:428047070.4000.2490.305—   
chr3_42804578_G_Cchr3:42804578-0.060-0.0470.708—   
chr3_42804577_G_Achr3:428045770.1910.2940.684<0.001%
chr3_42804664_G_Cchr3:428046640.1470.1270.672—   
chr3_42804611_T_Achr3:428046110.362-0.0600.379—   
chr3_42804530_C_Achr3:428045300.347-0.4230.085—   
chr3_42804562_G_Achr3:42804562-0.2090.083-0.586—   
chr3_42804635_A_Gchr3:428046350.3260.2310.159—   
chr3_42804559_C_Gchr3:42804559-0.154-0.184-0.562—   
chr3_42804612_G_Tchr3:428046120.315-0.0420.391—   
chr3_42804531_C_Tchr3:428045310.311-0.2730.232—   
chr3_42804711_C_Achr3:428047110.3110.2180.256—   
chr3_42804692_C_Achr3:428046920.2560.1610.525—   
chr3_42804593_A_Gchr3:428045930.291-0.1610.220—   
chr3_42804608_G_Achr3:428046080.291-0.2700.513—   
chr3_42804687_G_Cchr3:428046870.2890.1690.073—   
chr3_42804534_T_Gchr3:428045340.287-0.3820.281—   
chr3_42804756_T_Gchr3:428047560.2850.2780.366—   
chr3_42804605_A_Tchr3:428046050.284-0.3350.403—   
chr3_42804847_G_Achr3:428048470.021-0.091-0.501—   
chr3_42804532_A_Cchr3:428045320.279-0.3430.244—   
chr3_42804606_T_Gchr3:428046060.275-0.3120.427—   
chr3_42804711_C_Tchr3:428047110.2750.2340.183—   
chr3_42804606_T_Achr3:428046060.274-0.3710.489—   
chr3_42804610_C_Gchr3:42804610-0.026-0.3350.489—   
chr3_42804616_C_Achr3:428046160.2500.2940.489—   
chr3_42804733_T_Achr3:428047330.1440.2390.489—   
chr3_42804757_C_Gchr3:428047570.2720.3320.281—   
chr3_42804566_G_Achr3:428045660.270-0.0910.4760.0013%
chr3_42804833_G_Tchr3:428048330.133-0.073-0.476—   
chr3_42804517_A_Cchr3:428045170.265-0.003-0.012—   
chr3_42804559_C_Achr3:42804559-0.260-0.034-0.269—   
chr3_42804578_G_Tchr3:42804578-0.097-0.0230.464—   
chr3_42804528_A_Tchr3:42804528-0.253-0.0570.110—   
chr3_42804604_G_Cchr3:428046040.251-0.1770.379—   
chr3_42804630_C_Achr3:428046300.2510.1920.037—   
chr3_42804706_A_Tchr3:428047060.2510.1820.256—   
chr3_42804608_G_Cchr3:428046080.248-0.3190.232—   
chr3_42804562_G_Cchr3:42804562-0.026-0.021-0.440—   
chr3_42804669_G_Cchr3:42804669-0.0390.4420.4400.0013%
chr3_42804711_C_Gchr3:428047110.2460.2290.159—   
chr3_42804628_G_Achr3:428046280.2380.2550.427—   
chr3_42804534_T_Achr3:428045340.238-0.2310.208—   
chr3_42804726_C_Achr3:428047260.2380.2100.256—   
chr3_42804529_G_Cchr3:42804529-0.236-0.317-0.281—   
chr3_42804530_C_Gchr3:428045300.234-0.2080.208—   
chr3_42804560_G_Tchr3:428045600.2340.0730.256—   
chr3_42804557_G_Cchr3:428045570.007-0.0230.415—   
chr3_42804563_T_Achr3:42804563-0.024-0.143-0.415—   
chr3_42804563_T_Gchr3:42804563-0.068-0.091-0.415—   
chr3_42804564_G_Cchr3:42804564-0.053-0.101-0.415—   
chr3_42804706_A_Cchr3:428047060.2320.1090.183—   
chr3_42804846_T_Gchr3:428048460.2170.0600.415—   
chr3_42804603_G_Achr3:428046030.231-0.1350.159—   
chr3_42804621_A_Gchr3:42804621-0.2310.0340.159—   
chr3_42804605_A_Gchr3:428046050.224-0.2360.403—   
chr3_42804660_G_Cchr3:428046600.0630.0730.403—   
chr3_42804838_G_Cchr3:428048380.0850.0700.403—   
chr3_42804516_C_Gchr3:42804516-0.2240.0420.012—   
chr3_42804625_C_Gchr3:42804625-0.2210.055-0.0490.103%
chr3_42804578_G_Achr3:42804578-0.063-0.0520.3910.0020%
chr3_42804580_T_Gchr3:428045800.070-0.003-0.391—   
chr3_42804620_G_Cchr3:428046200.1570.0030.391—   
chr3_42804634_T_Gchr3:428046340.2190.1770.342—   
chr3_42804816_G_Cchr3:428048160.0650.0810.391—   
chr3_42804652_C_Tchr3:42804652-0.2170.229-0.183—   
chr3_42804568_G_Cchr3:42804568-0.185-0.021-0.379—   
chr3_42804627_G_Cchr3:42804627-0.212-0.018-0.293—   
chr3_42804843_G_Achr3:428048430.128-0.057-0.379—   
chr3_42804623_T_Gchr3:42804623-0.1880.023-0.366—   
chr3_42804633_C_Gchr3:428046330.2050.0440.085—   
chr3_42804651_A_Gchr3:428046510.091-0.0390.366—   
chr3_42804657_G_Cchr3:428046570.1110.0160.366—   
chr3_42804663_A_Tchr3:42804663-0.0390.2130.3660.030%
chr3_42804716_G_Tchr3:42804716-0.060-0.143-0.366—   
chr3_42804551_C_Gchr3:42804551-0.203-0.0080.159—   
chr3_42804660_G_Achr3:42804660-0.2030.1820.1470.0013%
chr3_42804604_G_Achr3:428046040.202-0.2470.330—   
chr3_42804557_G_Tchr3:42804557-0.074-0.010-0.354—   
chr3_42804611_T_Cchr3:428046110.198-0.1040.134<0.001%
chr3_42804697_G_Tchr3:428046970.1080.1140.354—   
chr3_42804649_G_Cchr3:42804649-0.1970.106-0.134—   
chr3_42804633_C_Achr3:428046330.1950.1040.195—   
chr3_42804631_C_Tchr3:428046310.1930.0420.220—   
chr3_42804520_G_Tchr3:42804520-0.191-0.031-0.208—   
chr3_42804564_G_Tchr3:428045640.017-0.062-0.342—   
chr3_42804594_G_Cchr3:428045940.1910.0160.171—   
chr3_42804612_G_Cchr3:428046120.191-0.0810.195—   
chr3_42804775_C_Tchr3:428047750.068-0.062-0.342—   
chr3_42804594_G_Tchr3:428045940.1880.0340.122—   
chr3_42804705_G_Achr3:428047050.1880.1190.049—   
chr3_42804565_C_Achr3:428045650.1850.0600.147—   
chr3_42804577_G_Tchr3:428045770.0790.0620.330—   
chr3_42804604_G_Tchr3:428046040.185-0.1840.281—   
chr3_42804733_T_Gchr3:428047330.1200.1690.330<0.001%
chr3_42804811_C_Gchr3:428048110.022-0.0160.330—   
chr3_42804556_G_Tchr3:42804556-0.1790.1690.000—   
chr3_42804666_C_Gchr3:428046660.179-0.0420.073—   
chr3_42804550_G_Achr3:428045500.1660.0290.318—   
chr3_42804652_C_Achr3:42804652-0.103-0.0290.318—   
chr3_42804687_G_Achr3:428046870.1740.083-0.0370.059%
chr3_42804732_C_Tchr3:428047320.1730.1120.122—   
chr3_42804580_T_Cchr3:42804580-0.024-0.112-0.305—   
chr3_42804611_T_Gchr3:428046110.171-0.1690.049—   
chr3_42804643_T_Cchr3:42804643-0.0430.0340.305—   
chr3_42804691_G_Cchr3:42804691-0.097-0.044-0.305—   
chr3_42804712_T_Achr3:428047120.1570.1400.305—   
chr3_42804712_T_Gchr3:428047120.1660.0730.305—   
chr3_42804819_G_Tchr3:42804819-0.022-0.026-0.305—   
chr3_42804541_C_Tchr3:428045410.1690.2550.134—   
chr3_42804575_G_Tchr3:42804575-0.1690.0860.024—   
chr3_42804584_G_Cchr3:42804584-0.166-0.075-0.012—   
chr3_42804758_C_Achr3:428047580.1660.2440.147—   
chr3_42804529_G_Tchr3:42804529-0.164-0.075-0.122—   
chr3_42804559_C_Tchr3:42804559-0.159-0.094-0.293—   
chr3_42804567_T_Gchr3:428045670.164-0.1170.122—   
chr3_42804613_G_Tchr3:428046130.1640.0130.000—   
chr3_42804664_G_Tchr3:42804664-0.0190.1530.293—   
chr3_42804698_G_Cchr3:428046980.1640.2470.244—   
chr3_42804751_C_Achr3:428047510.019-0.112-0.293—   
chr3_42804793_T_Gchr3:428047930.012-0.062-0.293—   
chr3_42804821_C_Gchr3:428048210.0190.0570.2930.0013%
chr3_42804550_G_Tchr3:428045500.1590.1450.256—   
chr3_42804607_T_Achr3:428046070.159-0.0990.147—   
chr3_42804618_G_Tchr3:42804618-0.1590.109-0.220—   
chr3_42804722_G_Tchr3:428047220.1590.1610.244—   
chr3_42804553_A_Tchr3:428045530.1570.0910.171—   
chr3_42804556_G_Achr3:42804556-0.084-0.106-0.281—   
chr3_42804565_C_Gchr3:42804565-0.082-0.073-0.281—   
chr3_42804734_C_Gchr3:428047340.1440.2100.281—   
chr3_42804752_C_Gchr3:428047520.005-0.096-0.281—   
chr3_42804839_A_Cchr3:428048390.0510.0600.281—   
chr3_42804757_C_Achr3:428047570.1560.1970.183<0.001%
chr3_42804696_C_Achr3:428046960.1540.1770.110—   
chr3_42804712_T_Cchr3:428047120.1540.1430.269—   
chr3_42804537_G_Tchr3:42804537-0.150-0.070-0.147—   
chr3_42804584_G_Tchr3:428045840.084-0.0290.269—   
chr3_42804658_G_Tchr3:42804658-0.0220.1220.269—   
chr3_42804667_G_Tchr3:42804667-0.079-0.086-0.269—   
chr3_42804700_C_Achr3:42804700-0.084-0.132-0.269—   
chr3_42804706_A_Gchr3:42804706-0.150-0.148-0.171—   
chr3_42804745_T_Achr3:428047450.1500.1430.110—   
chr3_42804816_G_Tchr3:428048160.0050.0860.269—   
chr3_42804825_C_Gchr3:42804825-0.043-0.031-0.269—   
chr3_42804705_G_Cchr3:428047050.1490.0860.024—   
chr3_42804734_C_Tchr3:428047340.1490.2230.159—   
chr3_42804690_C_Achr3:428046900.1470.1170.049—   
chr3_42804699_G_Tchr3:428046990.1470.1710.256—   
chr3_42804576_C_Tchr3:42804576-0.1450.106-0.134—   
chr3_42804595_C_Gchr3:42804595-0.145-0.0360.122—   
chr3_42804608_G_Tchr3:428046080.145-0.3060.232—   
chr3_42804553_A_Cchr3:428045530.0970.0940.256—   
chr3_42804561_C_Achr3:428045610.0150.021-0.256—   
chr3_42804564_G_Achr3:42804564-0.1440.140-0.195—   
chr3_42804629_C_Tchr3:428046290.067-0.161-0.256—   
chr3_42804658_G_Cchr3:428046580.0550.1090.256—   
chr3_42804786_A_Cchr3:428047860.044-0.0520.256—   
chr3_42804840_T_Gchr3:42804840-0.0090.0420.256—   
chr3_42804630_C_Tchr3:428046300.1420.088-0.061—   
chr3_42804565_C_Tchr3:428045650.140-0.010-0.220—   
chr3_42804838_G_Tchr3:428048380.140-0.005-0.171—   
chr3_42804632_A_Tchr3:428046320.1380.0880.024—   
chr3_42804749_G_Cchr3:428047490.1380.0310.037—   
chr3_42804573_C_Tchr3:42804573-0.1150.1380.244—   
chr3_42804626_T_Cchr3:42804626-0.1370.055-0.195—   
chr3_42804646_A_Tchr3:428046460.0410.2030.244—   
chr3_42804675_T_Achr3:428046750.0850.0490.244—   
chr3_42804700_C_Gchr3:42804700-0.094-0.156-0.244—   
chr3_42804702_C_Achr3:428047020.017-0.047-0.244—   
chr3_42804703_T_Achr3:428047030.0620.0080.244—   
chr3_42804734_C_Achr3:428047340.0820.2080.244—   
chr3_42804771_G_Tchr3:42804771-0.0020.0750.244—   
chr3_42804815_G_Achr3:428048150.002-0.013-0.2440.0099%
chr3_42804824_A_Tchr3:42804824-0.041-0.026-0.244—   
chr3_42804840_T_Cchr3:428048400.0310.0600.244—   
chr3_42804717_C_Tchr3:42804717-0.132-0.112-0.110—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.