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CYP8B1

receptor: FXRTier 1
Prior gene annotation

Retained explanatory context, not the pharmacist's submitted wording; submitted reviews below take precedence.

Drug substrates (prior annotation)

none in routine clinical use, endogenous or bile acid pathway

refs: 15550563

CAMIP Tier 1: peak-anchored panel

FXR

Submitted decision (verbatim): 接受

No revision text or notes were submitted.

Prior explanatory context

Retained explanatory context, not the pharmacist's submitted wording. The submitted review above takes precedence; this context is not a replacement for the reviewer's revision or notes.

Inducer
Obeticholic acid; Experimental GW4064
Regulatory element
in distal enhancer +19834 bp
Predicted consequence
Altered receptor-mediated feedback repression of CYP8B1, shifting the cholic acid to chenodeoxycholic acid synthesis ratio in endogenous bile acid pathways.
Prior narrative
Altered receptor-mediated feedback repression of CYP8B1, shifting the cholic acid to chenodeoxycholic acid synthesis ratio in endogenous bile acid pathways.
Drug context
none in routine clinical use, endogenous or bile acid pathway
Prior references
15550563

Scored variants near CYP8B1

chr3:42,772,191..42,975,879, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr3_42804703_T_Gchr3:428047030.4660.4471.000—   
chr3_42804558_A_Tchr3:428045580.6090.6020.694<0.001%
chr3_42804607_T_Cchr3:428046070.591-0.3450.506—   
chr3_42804709_G_Cchr3:428047090.5810.3600.412—   
chr3_42804827_G_Tchr3:428048270.0970.2030.9410.0013%
chr3_42804710_G_Achr3:428047100.5240.3650.353—   
chr3_42804609_G_Achr3:428046090.512-0.1950.576—   
chr3_42804708_G_Cchr3:428047080.5090.3020.306—   
chr3_42804609_G_Cchr3:428046090.486-0.2640.541—   
chr3_42804709_G_Achr3:428047090.4840.2030.1180.011%
chr3_42804709_G_Tchr3:428047090.4760.3020.329—   
chr3_42804532_A_Gchr3:428045320.468-0.1900.388—   
chr3_42804560_G_Achr3:428045600.0130.0000.824<0.001%
chr3_42804708_G_Achr3:428047080.4660.2920.176<0.001%
chr3_42804707_G_Achr3:428047070.4540.3530.3760.0020%
chr3_42804625_C_Achr3:42804625-0.4430.028-0.329—   
chr3_42804609_G_Tchr3:428046090.434-0.3320.365—   
chr3_42804707_G_Cchr3:428047070.4340.3960.506—   
chr3_42804710_G_Cchr3:428047100.4240.3150.482—   
chr3_42804605_A_Cchr3:428046050.423-0.3220.565—   
chr3_42804607_T_Gchr3:428046070.414-0.3020.529—   
chr3_42804576_C_Gchr3:428045760.4030.0460.024—   
chr3_42804708_G_Tchr3:428047080.4030.3020.271—   
chr3_42804606_T_Cchr3:428046060.399-0.2590.565—   
chr3_42804707_G_Tchr3:428047070.3890.2440.294—   
chr3_42804578_G_Cchr3:42804578-0.058-0.0460.682—   
chr3_42804577_G_Achr3:428045770.1860.2870.659<0.001%
chr3_42804664_G_Cchr3:428046640.1430.1240.647—   
chr3_42804611_T_Achr3:428046110.353-0.0580.365—   
chr3_42804530_C_Achr3:428045300.338-0.4140.082—   
chr3_42804562_G_Achr3:42804562-0.2030.081-0.565—   
chr3_42804635_A_Gchr3:428046350.3180.2260.153—   
chr3_42804559_C_Gchr3:42804559-0.150-0.180-0.541—   
chr3_42804612_G_Tchr3:428046120.306-0.0410.376—   
chr3_42804531_C_Tchr3:428045310.303-0.2660.224—   
chr3_42804711_C_Achr3:428047110.3030.2130.247—   
chr3_42804692_C_Achr3:428046920.2500.1570.506—   
chr3_42804593_A_Gchr3:428045930.283-0.1570.212—   
chr3_42804608_G_Achr3:428046080.283-0.2640.494—   
chr3_42804687_G_Cchr3:428046870.2810.1650.071—   
chr3_42804534_T_Gchr3:428045340.280-0.3730.271—   
chr3_42804756_T_Gchr3:428047560.2780.2720.353—   
chr3_42804605_A_Tchr3:428046050.276-0.3270.388—   
chr3_42804847_G_Achr3:428048470.020-0.089-0.482—   
chr3_42804532_A_Cchr3:428045320.271-0.3350.235—   
chr3_42804606_T_Gchr3:428046060.268-0.3050.412—   
chr3_42804711_C_Tchr3:428047110.2680.2280.176—   
chr3_42804606_T_Achr3:428046060.266-0.3630.471—   
chr3_42804610_C_Gchr3:42804610-0.025-0.3270.471—   
chr3_42804616_C_Achr3:428046160.2430.2870.471—   
chr3_42804733_T_Achr3:428047330.1400.2340.471—   
chr3_42804757_C_Gchr3:428047570.2650.3250.271—   
chr3_42804566_G_Achr3:428045660.263-0.0890.4590.0013%
chr3_42804833_G_Tchr3:428048330.130-0.071-0.459—   
chr3_42804517_A_Cchr3:428045170.258-0.003-0.012—   
chr3_42804559_C_Achr3:42804559-0.253-0.033-0.259—   
chr3_42804578_G_Tchr3:42804578-0.095-0.0230.447—   
chr3_42804528_A_Tchr3:42804528-0.246-0.0560.106—   
chr3_42804604_G_Cchr3:428046040.245-0.1730.365—   
chr3_42804630_C_Achr3:428046300.2450.1880.035—   
chr3_42804706_A_Tchr3:428047060.2450.1780.247—   
chr3_42804608_G_Cchr3:428046080.241-0.3120.224—   
chr3_42804562_G_Cchr3:42804562-0.025-0.020-0.424—   
chr3_42804669_G_Cchr3:42804669-0.0380.4310.4240.0013%
chr3_42804711_C_Gchr3:428047110.2400.2230.153—   
chr3_42804628_G_Achr3:428046280.2310.2490.412—   
chr3_42804534_T_Achr3:428045340.231-0.2260.200—   
chr3_42804726_C_Achr3:428047260.2310.2060.247—   
chr3_42804529_G_Cchr3:42804529-0.230-0.310-0.271—   
chr3_42804530_C_Gchr3:428045300.228-0.2030.200—   
chr3_42804560_G_Tchr3:428045600.2280.0710.247—   
chr3_42804557_G_Cchr3:428045570.007-0.0230.400—   
chr3_42804563_T_Achr3:42804563-0.023-0.140-0.400—   
chr3_42804563_T_Gchr3:42804563-0.067-0.089-0.400—   
chr3_42804564_G_Cchr3:42804564-0.052-0.099-0.400—   
chr3_42804706_A_Cchr3:428047060.2260.1070.176—   
chr3_42804846_T_Gchr3:428048460.2110.0580.400—   
chr3_42804603_G_Achr3:428046030.225-0.1320.153—   
chr3_42804621_A_Gchr3:42804621-0.2250.0330.153—   
chr3_42804605_A_Gchr3:428046050.218-0.2310.388—   
chr3_42804660_G_Cchr3:428046600.0620.0710.388—   
chr3_42804838_G_Cchr3:428048380.0830.0690.388—   
chr3_42804516_C_Gchr3:42804516-0.2180.0410.012—   
chr3_42804625_C_Gchr3:42804625-0.2150.053-0.0470.103%
chr3_42804578_G_Achr3:42804578-0.062-0.0510.3760.0020%
chr3_42804580_T_Gchr3:428045800.068-0.003-0.376—   
chr3_42804620_G_Cchr3:428046200.1530.0030.376—   
chr3_42804634_T_Gchr3:428046340.2130.1730.329—   
chr3_42804816_G_Cchr3:428048160.0630.0790.376—   
chr3_42804652_C_Tchr3:42804652-0.2110.223-0.176—   
chr3_42804568_G_Cchr3:42804568-0.180-0.020-0.365—   
chr3_42804627_G_Cchr3:42804627-0.206-0.018-0.282—   
chr3_42804843_G_Achr3:428048430.125-0.056-0.365—   
chr3_42804623_T_Gchr3:42804623-0.1830.023-0.353—   
chr3_42804633_C_Gchr3:428046330.2000.0430.082—   
chr3_42804651_A_Gchr3:428046510.088-0.0380.353—   
chr3_42804657_G_Cchr3:428046570.1080.0150.353—   
chr3_42804663_A_Tchr3:42804663-0.0380.2080.3530.030%
chr3_42804716_G_Tchr3:42804716-0.058-0.140-0.353—   
chr3_42804551_C_Gchr3:42804551-0.198-0.0080.153—   
chr3_42804660_G_Achr3:42804660-0.1980.1780.1410.0013%
chr3_42804604_G_Achr3:428046040.196-0.2410.318—   
chr3_42804557_G_Tchr3:42804557-0.072-0.010-0.341—   
chr3_42804611_T_Cchr3:428046110.193-0.1020.129<0.001%
chr3_42804697_G_Tchr3:428046970.1050.1120.341—   
chr3_42804649_G_Cchr3:42804649-0.1910.104-0.129—   
chr3_42804633_C_Achr3:428046330.1900.1020.188—   
chr3_42804631_C_Tchr3:428046310.1880.0410.212—   
chr3_42804520_G_Tchr3:42804520-0.186-0.030-0.200—   
chr3_42804564_G_Tchr3:428045640.017-0.061-0.329—   
chr3_42804594_G_Cchr3:428045940.1860.0150.165—   
chr3_42804612_G_Cchr3:428046120.186-0.0790.188—   
chr3_42804775_C_Tchr3:428047750.067-0.061-0.329—   
chr3_42804594_G_Tchr3:428045940.1830.0330.118—   
chr3_42804705_G_Achr3:428047050.1830.1170.047—   
chr3_42804565_C_Achr3:428045650.1800.0580.141—   
chr3_42804577_G_Tchr3:428045770.0770.0610.318—   
chr3_42804604_G_Tchr3:428046040.180-0.1800.271—   
chr3_42804733_T_Gchr3:428047330.1160.1650.318<0.001%
chr3_42804811_C_Gchr3:428048110.022-0.0150.318—   
chr3_42804556_G_Tchr3:42804556-0.1750.1650.000—   
chr3_42804666_C_Gchr3:428046660.175-0.0410.071—   
chr3_42804550_G_Achr3:428045500.1610.0280.306—   
chr3_42804652_C_Achr3:42804652-0.100-0.0280.306—   
chr3_42804687_G_Achr3:428046870.1700.081-0.0350.059%
chr3_42804732_C_Tchr3:428047320.1680.1090.118—   
chr3_42804580_T_Cchr3:42804580-0.023-0.109-0.294—   
chr3_42804611_T_Gchr3:428046110.166-0.1650.047—   
chr3_42804643_T_Cchr3:42804643-0.0420.0330.294—   
chr3_42804691_G_Cchr3:42804691-0.095-0.043-0.294—   
chr3_42804712_T_Achr3:428047120.1530.1370.294—   
chr3_42804712_T_Gchr3:428047120.1610.0710.294—   
chr3_42804819_G_Tchr3:42804819-0.022-0.025-0.294—   
chr3_42804541_C_Tchr3:428045410.1650.2490.129—   
chr3_42804575_G_Tchr3:42804575-0.1650.0840.024—   
chr3_42804584_G_Cchr3:42804584-0.161-0.074-0.012—   
chr3_42804758_C_Achr3:428047580.1610.2390.141—   
chr3_42804529_G_Tchr3:42804529-0.160-0.074-0.118—   
chr3_42804559_C_Tchr3:42804559-0.155-0.091-0.282—   
chr3_42804567_T_Gchr3:428045670.160-0.1140.118—   
chr3_42804613_G_Tchr3:428046130.1600.0130.000—   
chr3_42804664_G_Tchr3:42804664-0.0180.1500.282—   
chr3_42804698_G_Cchr3:428046980.1600.2410.235—   
chr3_42804751_C_Achr3:428047510.018-0.109-0.282—   
chr3_42804793_T_Gchr3:428047930.012-0.061-0.282—   
chr3_42804821_C_Gchr3:428048210.0180.0560.2820.0013%
chr3_42804550_G_Tchr3:428045500.1550.1420.247—   
chr3_42804607_T_Achr3:428046070.155-0.0960.141—   
chr3_42804618_G_Tchr3:42804618-0.1550.107-0.212—   
chr3_42804722_G_Tchr3:428047220.1550.1570.235—   
chr3_42804553_A_Tchr3:428045530.1530.0890.165—   
chr3_42804556_G_Achr3:42804556-0.082-0.104-0.271—   
chr3_42804565_C_Gchr3:42804565-0.080-0.071-0.271—   
chr3_42804734_C_Gchr3:428047340.1400.2060.271—   
chr3_42804752_C_Gchr3:428047520.005-0.094-0.271—   
chr3_42804839_A_Cchr3:428048390.0500.0580.271—   
chr3_42804757_C_Achr3:428047570.1510.1930.176<0.001%
chr3_42804696_C_Achr3:428046960.1500.1730.106—   
chr3_42804712_T_Cchr3:428047120.1500.1400.259—   
chr3_42804537_G_Tchr3:42804537-0.146-0.069-0.141—   
chr3_42804584_G_Tchr3:428045840.082-0.0280.259—   
chr3_42804658_G_Tchr3:42804658-0.0220.1190.259—   
chr3_42804667_G_Tchr3:42804667-0.077-0.084-0.259—   
chr3_42804700_C_Achr3:42804700-0.082-0.129-0.259—   
chr3_42804706_A_Gchr3:42804706-0.146-0.145-0.165—   
chr3_42804745_T_Achr3:428047450.1460.1400.106—   
chr3_42804816_G_Tchr3:428048160.0050.0840.259—   
chr3_42804825_C_Gchr3:42804825-0.042-0.030-0.259—   
chr3_42804705_G_Cchr3:428047050.1450.0840.024—   
chr3_42804734_C_Tchr3:428047340.1450.2180.153—   
chr3_42804690_C_Achr3:428046900.1430.1140.047—   
chr3_42804699_G_Tchr3:428046990.1430.1680.247—   
chr3_42804576_C_Tchr3:42804576-0.1410.104-0.129—   
chr3_42804595_C_Gchr3:42804595-0.141-0.0360.118—   
chr3_42804608_G_Tchr3:428046080.141-0.2990.224—   
chr3_42804553_A_Cchr3:428045530.0950.0910.247—   
chr3_42804561_C_Achr3:428045610.0150.020-0.247—   
chr3_42804564_G_Achr3:42804564-0.1400.137-0.188—   
chr3_42804629_C_Tchr3:428046290.065-0.157-0.247—   
chr3_42804658_G_Cchr3:428046580.0530.1070.247—   
chr3_42804786_A_Cchr3:428047860.043-0.0510.247—   
chr3_42804840_T_Gchr3:42804840-0.0080.0410.247—   
chr3_42804630_C_Tchr3:428046300.1380.086-0.059—   
chr3_42804565_C_Tchr3:428045650.136-0.010-0.212—   
chr3_42804838_G_Tchr3:428048380.136-0.005-0.165—   
chr3_42804632_A_Tchr3:428046320.1350.0860.024—   
chr3_42804749_G_Cchr3:428047490.1350.0300.035—   
chr3_42804573_C_Tchr3:42804573-0.1110.1350.235—   
chr3_42804626_T_Cchr3:42804626-0.1330.053-0.188—   
chr3_42804646_A_Tchr3:428046460.0400.1980.235—   
chr3_42804675_T_Achr3:428046750.0830.0480.235—   
chr3_42804700_C_Gchr3:42804700-0.092-0.152-0.235—   
chr3_42804702_C_Achr3:428047020.017-0.046-0.235—   
chr3_42804703_T_Achr3:428047030.0600.0080.235—   
chr3_42804734_C_Achr3:428047340.0800.2030.235—   
chr3_42804771_G_Tchr3:42804771-0.0020.0740.235—   
chr3_42804815_G_Achr3:428048150.002-0.013-0.2350.0099%
chr3_42804824_A_Tchr3:42804824-0.040-0.025-0.235—   
chr3_42804840_T_Cchr3:428048400.0300.0580.235—   
chr3_42804717_C_Tchr3:42804717-0.128-0.109-0.106—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.