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FGF19

receptor: FXRTier 1

Drug substrates

enterohepatic bile-acid signaling

refs: 25198545

CAMIP causal chains

FXR

Attenuated receptor-mediated transcriptional activation of enterocyte FGF19, disrupting the intestinal endocrine signaling cascade required for the downstream feedback repression of hepatic bile acid biosynthesis.

Affected substrate drugs (PharmGKB): none in routine clinical use, endogenous or bile acid pathway

Scored variants near FGF19

chr11:69,598,237..69,804,022, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr11_69688546_T_Achr11:696885460.5120.4660.386—   
chr11_69688546_T_Gchr11:696885460.4780.4360.368—   
chr11_69641732_A_Gchr11:69641732-0.154-0.185-0.801—   
chr11_69641747_A_Gchr11:69641747-0.141-0.077-0.661—   
chr11_69639073_A_Cchr11:696390730.3730.3120.561—   
chr11_69688561_T_Gchr11:696885610.3380.3320.263—   
chr11_69641741_T_Gchr11:69641741-0.114-0.093-0.567—   
chr11_69688555_G_Tchr11:69688555-0.303-0.335-0.409—   
chr11_69639078_G_Cchr11:696390780.1530.2020.526—   
chr11_69641738_G_Cchr11:696417380.0730.1130.526—   
chr11_69641739_G_Cchr11:696417390.0780.1070.497—   
chr11_69688548_T_Gchr11:696885480.2800.3680.228—   
chr11_69639076_A_Cchr11:696390760.2760.2170.456—   
chr11_69641738_G_Tchr11:696417380.0960.0880.480—   
chr11_69641752_T_Gchr11:69641752-0.103-0.071-0.480—   
chr11_69639062_C_Gchr11:69639062-0.269-0.159-0.304<0.001%
chr11_69641743_C_Gchr11:69641743-0.080-0.098-0.474—   
chr11_69639064_G_Cchr11:696390640.0020.1760.468—   
chr11_69639076_A_Tchr11:696390760.1590.1810.456—   
chr11_69641738_G_Achr11:696417380.0780.1120.450—   
chr11_69638962_T_Gchr11:696389620.2090.1710.444—   
chr11_69638982_T_Gchr11:696389820.2520.2750.421—   
chr11_69641739_G_Achr11:696417390.0860.1120.444<0.001%
chr11_69639077_A_Cchr11:696390770.2460.1210.433—   
chr11_69638964_C_Gchr11:696389640.1340.1230.433—   
chr11_69639042_A_Cchr11:696390420.1800.1890.4330.102%
chr11_69641737_G_Cchr11:696417370.0600.0930.433—   
chr11_69688566_C_Gchr11:69688566-0.245-0.275-0.205<0.001%
chr11_69688561_T_Cchr11:69688561-0.088-0.282-0.427—   
chr11_69688559_T_Gchr11:696885590.2400.2390.193—   
chr11_69639045_T_Cchr11:696390450.1940.1130.421—   
chr11_69639045_T_Gchr11:696390450.2040.1260.421—   
chr11_69641735_A_Gchr11:69641735-0.076-0.084-0.409—   
chr11_69688568_T_Achr11:696885680.2320.2470.199—   
chr11_69639041_A_Cchr11:696390410.0770.1060.398—   
chr11_69639089_A_Tchr11:696390890.0920.1220.398—   
chr11_69641739_G_Tchr11:696417390.0840.0880.392—   
chr11_69688554_A_Tchr11:696885540.2200.2390.181—   
chr11_69638963_T_Gchr11:696389630.1120.0980.386—   
chr11_69639088_G_Cchr11:696390880.1790.1910.386—   
chr11_69641737_G_Achr11:696417370.0680.0840.386—   
chr11_69641750_G_Cchr11:696417500.0580.0830.386—   
chr11_69688564_A_Cchr11:69688564-0.219-0.254-0.158—   
chr11_69641744_G_Cchr11:696417440.0630.0740.380—   
chr11_69641750_G_Achr11:696417500.0650.0780.380—   
chr11_69688563_A_Cchr11:69688563-0.212-0.239-0.175—   
chr11_69688565_A_Tchr11:69688565-0.212-0.191-0.111—   
chr11_69639029_A_Tchr11:696390290.2100.184-0.105—   
chr11_69641750_G_Tchr11:696417500.0730.0720.368—   
chr11_69688564_A_Tchr11:69688564-0.209-0.254-0.175—   
chr11_69639047_G_Cchr11:696390470.1600.0830.363—   
chr11_69639074_C_Tchr11:696390740.1620.1860.363<0.001%
chr11_69641734_A_Gchr11:69641734-0.066-0.086-0.357—   
chr11_69641736_G_Cchr11:696417360.0360.0740.357—   
chr11_69639045_T_Achr11:696390450.0940.0650.351—   
chr11_69639066_G_Cchr11:696390660.0430.1340.3510.0020%
chr11_69641737_G_Tchr11:696417370.0600.0990.351—   
chr11_69688563_A_Tchr11:69688563-0.199-0.212-0.222—   
chr11_69688551_C_Achr11:696885510.1970.2270.193—   
chr11_69639027_C_Tchr11:69639027-0.196-0.116-0.269—   
chr11_69639090_G_Tchr11:696390900.1950.1810.339—   
chr11_69688562_C_Tchr11:69688562-0.194-0.212-0.205—   
chr11_69639008_G_Cchr11:69639008-0.120-0.161-0.339—   
chr11_69639092_T_Cchr11:69639092-0.031-0.035-0.339—   
chr11_69641740_G_Achr11:696417400.0610.0840.333—   
chr11_69688562_C_Achr11:69688562-0.189-0.214-0.187—   
chr11_69688563_A_Gchr11:69688563-0.189-0.212-0.088—   
chr11_69688571_C_Tchr11:69688571-0.187-0.194-0.205—   
chr11_69638964_C_Achr11:696389640.0840.1160.327—   
chr11_69638965_C_Gchr11:696389650.1030.1490.327—   
chr11_69638980_A_Tchr11:696389800.1690.0960.327—   
chr11_69641740_G_Cchr11:696417400.0530.0790.327—   
chr11_69641834_C_Gchr11:696418340.1840.1270.070—   
chr11_69688568_T_Cchr11:696885680.1800.1280.205—   
chr11_69638959_A_Tchr11:696389590.0840.0930.316—   
chr11_69638965_C_Achr11:696389650.0660.1340.316—   
chr11_69639046_T_Gchr11:696390460.1210.1390.316—   
chr11_69639075_G_Achr11:696390750.1080.1410.316—   
chr11_69688573_A_Gchr11:696885730.1740.1710.193—   
chr11_69638977_C_Achr11:696389770.1180.0580.304—   
chr11_69638992_T_Cchr11:69638992-0.064-0.045-0.304—   
chr11_69638995_C_Gchr11:696389950.1590.0200.304—   
chr11_69639033_G_Tchr11:696390330.1430.1890.304—   
chr11_69639069_A_Gchr11:69639069-0.0040.0240.304—   
chr11_69639078_G_Tchr11:696390780.1380.0710.304—   
chr11_69639089_A_Cchr11:696390890.0550.0400.304—   
chr11_69641749_G_Cchr11:696417490.0480.0430.304—   
chr11_69688565_A_Cchr11:69688565-0.172-0.184-0.029—   
chr11_69641748_G_Tchr11:696417480.0650.0520.298—   
chr11_69688544_C_Achr11:69688544-0.168-0.179-0.298—   
chr11_69638956_C_Achr11:696389560.0740.0760.292—   
chr11_69638995_C_Achr11:696389950.1530.0050.292—   
chr11_69639022_G_Tchr11:69639022-0.084-0.063-0.292—   
chr11_69639082_C_Achr11:696390820.1630.1890.234—   
chr11_69641746_G_Achr11:696417460.0360.0690.287—   
chr11_69688564_A_Gchr11:69688564-0.162-0.194-0.117—   
chr11_69688569_A_Cchr11:69688569-0.162-0.161-0.140—   
chr11_69638956_C_Tchr11:696389560.0940.0880.281—   
chr11_69638977_C_Gchr11:696389770.0940.0100.281—   
chr11_69638981_A_Tchr11:696389810.1080.0960.281—   
chr11_69638996_C_Gchr11:696389960.0880.0100.281—   
chr11_69639044_T_Gchr11:696390440.1120.0710.281—   
chr11_69639066_G_Achr11:696390660.0280.0910.281—   
chr11_69639077_A_Gchr11:696390770.1450.0640.281—   
chr11_69641748_G_Achr11:696417480.0360.0420.281—   
chr11_69688565_A_Gchr11:69688565-0.157-0.159-0.070—   
chr11_69641748_G_Cchr11:696417480.0680.0470.275—   
chr11_69638962_T_Achr11:696389620.0960.1060.269—   
chr11_69638976_C_Achr11:696389760.1150.0830.269—   
chr11_69638998_G_Cchr11:69638998-0.085-0.028-0.269—   
chr11_69639012_G_Achr11:696390120.1020.0530.269—   
chr11_69639048_C_Gchr11:69639048-0.123-0.065-0.269—   
chr11_69639075_G_Cchr11:696390750.0680.0730.269<0.001%
chr11_69688558_A_Gchr11:69688558-0.152-0.174-0.047—   
chr11_69639029_A_Cchr11:696390290.1510.1160.035—   
chr11_69641740_G_Tchr11:696417400.0410.0780.263—   
chr11_69641830_T_Gchr11:69641830-0.078-0.026-0.263—   
chr11_69688560_T_Achr11:69688560-0.149-0.234-0.158—   
chr11_69638993_C_Tchr11:696389930.0710.0180.257—   
chr11_69638994_C_Achr11:696389940.1320.0450.257—   
chr11_69639006_C_Gchr11:69639006-0.0120.0780.257—   
chr11_69639040_C_Achr11:69639040-0.108-0.101-0.257—   
chr11_69639040_C_Gchr11:696390400.015-0.091-0.257—   
chr11_69639041_A_Tchr11:696390410.0460.0150.257—   
chr11_69639046_T_Cchr11:696390460.0900.0730.257—   
chr11_69639084_A_Gchr11:696390840.0080.1070.257—   
chr11_69639093_C_Gchr11:69639093-0.111-0.091-0.2570.0020%
chr11_69639093_C_Tchr11:69639093-0.0050.009-0.257—   
chr11_69641749_G_Achr11:696417490.0350.0330.2570.0020%
chr11_69641749_G_Tchr11:696417490.0510.0450.257—   
chr11_69639074_C_Achr11:69639074-0.141-0.072-0.175<0.001%
chr11_69639010_A_Cchr11:696390100.1400.0930.187—   
chr11_69638959_A_Cchr11:696389590.0360.0710.246—   
chr11_69638968_C_Achr11:69638968-0.069-0.038-0.246—   
chr11_69638979_A_Tchr11:696389790.0800.0760.246—   
chr11_69638986_A_Cchr11:696389860.0120.0550.246—   
chr11_69638994_C_Tchr11:696389940.1270.0100.246—   
chr11_69639002_G_Achr11:69639002-0.041-0.093-0.246—   
chr11_69639039_G_Tchr11:69639039-0.0110.0760.246—   
chr11_69639044_T_Achr11:696390440.1270.0930.246—   
chr11_69639084_A_Cchr11:69639084-0.085-0.108-0.246—   
chr11_69688547_T_Cchr11:69688547-0.139-0.126-0.170<0.001%
chr11_69688559_T_Cchr11:69688559-0.137-0.128-0.070—   
chr11_69641736_G_Achr11:696417360.0300.0490.240—   
chr11_69641745_G_Cchr11:696417450.0300.0430.240—   
chr11_69688570_C_Gchr11:696885700.1340.1440.199—   
chr11_69638961_A_Tchr11:696389610.1130.0910.234—   
chr11_69638962_T_Cchr11:696389620.0670.0350.234—   
chr11_69638964_C_Tchr11:696389640.0120.0980.234—   
chr11_69638981_A_Gchr11:696389810.1270.0760.234—   
chr11_69638983_T_Gchr11:696389830.0760.0550.234—   
chr11_69638999_C_Gchr11:69638999-0.113-0.073-0.234—   
chr11_69639053_G_Achr11:69639053-0.086-0.113-0.234—   
chr11_69639079_T_Cchr11:696390790.128-0.0080.234—   
chr11_69639080_T_Gchr11:696390800.0950.0530.234—   
chr11_69639083_T_Achr11:69639083-0.041-0.083-0.234—   
chr11_69641745_G_Tchr11:696417450.0480.0550.234—   
chr11_69641855_T_Cchr11:69641855-0.040-0.037-0.234—   
chr11_69641802_C_Gchr11:69641802-0.060-0.005-0.228—   
chr11_69688556_A_Tchr11:69688556-0.104-0.055-0.228—   
chr11_69638984_C_Gchr11:696389840.1280.0780.211—   
chr11_69639062_C_Achr11:69639062-0.128-0.035-0.140—   
chr11_69638963_T_Cchr11:696389630.1270.0880.175—   
chr11_69638956_C_Gchr11:696389560.0550.0630.222—   
chr11_69638960_A_Tchr11:696389600.1070.0600.222—   
chr11_69638979_A_Cchr11:696389790.0620.0780.222—   
chr11_69639042_A_Gchr11:696390420.1070.0600.222—   
chr11_69639071_C_Gchr11:696390710.0270.0200.222—   
chr11_69639091_A_Cchr11:696390910.0690.0690.222—   
chr11_69688574_A_Gchr11:696885740.1260.1310.117—   
chr11_69688577_G_Achr11:69688577-0.126-0.149-0.211—   
chr11_69638976_C_Tchr11:696389760.1230.0780.152—   
chr11_69638991_C_Achr11:69638991-0.123-0.108-0.094—   
chr11_69641736_G_Tchr11:696417360.0350.0480.216—   
chr11_69688574_A_Cchr11:696885740.0600.0880.216<0.001%
chr11_69638944_T_Cchr11:69638944-0.037-0.038-0.211—   
chr11_69638957_C_Achr11:696389570.0350.0250.211—   
chr11_69638966_A_Cchr11:69638966-0.0220.0650.211—   
chr11_69638995_C_Tchr11:696389950.1070.0080.211—   
chr11_69639007_T_Gchr11:696390070.0310.0980.211—   
chr11_69639023_C_Gchr11:696390230.1110.1440.211—   
chr11_69639035_G_Achr11:696390350.0900.1130.211—   
chr11_69639079_T_Achr11:69639079-0.010-0.087-0.211—   
chr11_69639090_G_Achr11:69639090-0.091-0.033-0.211—   
chr11_69639099_G_Cchr11:69639099-0.032-0.057-0.211—   
chr11_69641762_A_Gchr11:69641762-0.063-0.035-0.211—   
chr11_69688550_A_Tchr11:69688550-0.118-0.121-0.146—   
chr11_69639050_C_Gchr11:69639050-0.116-0.106-0.164—   
chr11_69641746_G_Cchr11:696417460.0410.0370.205—   
chr11_69641847_A_Gchr11:69641847-0.022-0.028-0.205—   
chr11_69688567_A_Cchr11:69688567-0.116-0.111-0.041—   
chr11_69639011_C_Gchr11:69639011-0.115-0.048-0.187—   
chr11_69638955_C_Achr11:696389550.0590.0960.199—   
chr11_69638975_C_Tchr11:696389750.0700.0910.199—   
chr11_69638981_A_Cchr11:696389810.1010.0430.199—   
chr11_69639026_G_Achr11:69639026-0.023-0.008-0.199—   
chr11_69639029_A_Gchr11:696390290.0700.0780.199—   
chr11_69639043_T_Achr11:696390430.0500.0710.199—   
chr11_69639066_G_Tchr11:69639066-0.0340.0500.199—   
chr11_69639079_T_Gchr11:696390790.0900.0400.199—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.