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NR0B2

receptor: FXRTier 1
Prior gene annotation

Retained explanatory context, not the pharmacist's submitted wording; submitted reviews below take precedence.

Drug substrates (prior annotation)

none in routine clinical use, endogenous or bile acid pathway

refs: 16269825, 25198545

CAMIP Tier 1: peak-anchored panel

FXR

Submitted decision (verbatim): 接受

No revision text or notes were submitted.

Prior explanatory context

Retained explanatory context, not the pharmacist's submitted wording. The submitted review above takes precedence; this context is not a replacement for the reviewer's revision or notes.

Inducer
Obeticholic acid; Experimental GW4064
Regulatory element
overlapping TSS
Predicted consequence
Blunted receptor-mediated induction of NR0B2 expression, weakening the downstream transcriptional feedback inhibition of hepatic bile acid synthesis pathways.
Prior narrative
Blunted receptor-mediated induction of NR0B2 expression, weakening the downstream transcriptional feedback inhibition of hepatic bile acid synthesis pathways.
Drug context
none in routine clinical use, endogenous or bile acid pathway
Prior references
16269825, 25198545

Scored variants near NR0B2

chr1:26,811,488..27,013,975, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr1_26864748_G_Cchr1:268647480.8250.094-0.059—   
chr1_26827461_T_Cchr1:26827461-0.079-0.044-0.459—   
chr1_26864772_T_Achr1:26864772-0.260-0.142-0.153—   
chr1_26827451_T_Cchr1:26827451-0.072-0.079-0.453—   
chr1_26864718_A_Gchr1:26864718-0.123-0.066-0.424—   
chr1_26864782_T_Achr1:268647820.0830.1780.424—   
chr1_26864833_C_Gchr1:268648330.0570.0130.424—   
chr1_26864758_A_Gchr1:268647580.1800.0940.412—   
chr1_26864722_G_Cchr1:268647220.2300.0360.188—   
chr1_26827486_T_Cchr1:26827486-0.061-0.072-0.400—   
chr1_26864734_C_Gchr1:26864734-0.146-0.015-0.388—   
chr1_26864789_T_Gchr1:26864789-0.170-0.036-0.388—   
chr1_26864722_G_Achr1:268647220.2160.0330.047—   
chr1_26827523_T_Cchr1:26827523-0.076-0.032-0.376—   
chr1_26864713_A_Gchr1:268647130.0000.041-0.376—   
chr1_26864798_A_Tchr1:268647980.210-0.1400.200—   
chr1_26864716_T_Gchr1:26864716-0.013-0.020-0.365—   
chr1_26864778_A_Cchr1:26864778-0.0300.2160.365—   
chr1_26864832_C_Tchr1:26864832-0.116-0.081-0.3650.0013%
chr1_26827470_C_Gchr1:268274700.0420.0510.359—   
chr1_26864720_T_Cchr1:268647200.2030.0100.071—   
chr1_26864722_G_Tchr1:268647220.2030.0360.059—   
chr1_26864741_C_Achr1:268647410.0800.0740.353—   
chr1_26864820_C_Gchr1:26864820-0.200-0.119-0.224—   
chr1_26827464_A_Cchr1:26827464-0.033-0.056-0.335—   
chr1_26864760_C_Gchr1:26864760-0.190-0.061-0.2240.062%
chr1_26827529_T_Cchr1:26827529-0.071-0.100-0.329—   
chr1_26864721_G_Cchr1:268647210.1860.0150.224—   
chr1_26864734_C_Tchr1:26864734-0.186-0.025-0.224—   
chr1_26864813_T_Achr1:26864813-0.186-0.018-0.259—   
chr1_26864719_G_Cchr1:268647190.1800.005-0.047—   
chr1_26827469_C_Gchr1:268274690.0470.0510.312—   
chr1_26864781_C_Tchr1:268647810.1760.1500.188<0.001%
chr1_26864811_A_Cchr1:268648110.1760.0690.153—   
chr1_26864732_C_Gchr1:26864732-0.030-0.015-0.306—   
chr1_26864822_G_Cchr1:268648220.1230.0710.306—   
chr1_26864755_T_Gchr1:26864755-0.170-0.008-0.141—   
chr1_26864721_G_Achr1:268647210.1660.0180.082—   
chr1_26864724_A_Gchr1:26864724-0.073-0.030-0.294—   
chr1_26864794_T_Cchr1:268647940.150-0.1020.294—   
chr1_26864796_T_Achr1:26864796-0.1500.282-0.294—   
chr1_26827459_C_Gchr1:268274590.0370.0360.288—   
chr1_26864769_A_Gchr1:26864769-0.163-0.211-0.047—   
chr1_26864720_T_Achr1:268647200.1600.015-0.035—   
chr1_26864771_A_Tchr1:26864771-0.160-0.175-0.082—   
chr1_26864781_C_Gchr1:26864781-0.106-0.0990.282—   
chr1_26864792_G_Tchr1:268647920.160-0.0610.212—   
chr1_26864801_A_Tchr1:268648010.1030.0360.282—   
chr1_26864831_A_Cchr1:26864831-0.160-0.127-0.247—   
chr1_26827477_T_Cchr1:26827477-0.038-0.053-0.276—   
chr1_26864738_A_Gchr1:26864738-0.156-0.056-0.2590.0013%
chr1_26864792_G_Achr1:268647920.156-0.0810.035—   
chr1_26864793_A_Cchr1:268647930.156-0.1170.247—   
chr1_26864712_G_Cchr1:268647120.1030.0410.271—   
chr1_26864746_G_Achr1:26864746-0.090-0.023-0.271<0.001%
chr1_26864747_A_Cchr1:268647470.1530.0180.141—   
chr1_26864772_T_Gchr1:26864772-0.153-0.112-0.024—   
chr1_26864802_C_Achr1:26864802-0.100-0.033-0.271—   
chr1_26827472_C_Gchr1:268274720.0580.0370.265—   
chr1_26827466_G_Cchr1:26827466-0.040-0.041-0.259—   
chr1_26864766_A_Cchr1:268647660.143-0.0050.259—   
chr1_26864797_A_Tchr1:268647970.146-0.0660.176—   
chr1_26864798_A_Cchr1:268647980.133-0.0910.259—   
chr1_26827456_G_Cchr1:26827456-0.023-0.037-0.253—   
chr1_26827470_C_Achr1:268274700.0420.0390.253—   
chr1_26827557_A_Cchr1:26827557-0.042-0.022-0.253—   
chr1_26864771_A_Gchr1:268647710.1430.1070.247—   
chr1_26864774_G_Tchr1:26864774-0.143-0.066-0.235—   
chr1_26864794_T_Achr1:268647940.143-0.1120.012—   
chr1_26827471_C_Gchr1:268274710.0320.0140.247—   
chr1_26827479_G_Cchr1:26827479-0.025-0.038-0.247—   
chr1_26864720_T_Gchr1:268647200.0630.015-0.247—   
chr1_26864721_G_Tchr1:268647210.140-0.0080.059—   
chr1_26864723_G_Tchr1:268647230.1400.0200.024—   
chr1_26864743_G_Achr1:26864743-0.140-0.051-0.153—   
chr1_26864787_C_Gchr1:268647870.020-0.058-0.247—   
chr1_26864795_C_Achr1:268647950.140-0.0890.153—   
chr1_26864839_T_Achr1:268648390.1400.0100.118—   
chr1_26864863_A_Cchr1:268648630.0600.0380.247—   
chr1_26864863_A_Tchr1:268648630.0170.0200.247—   
chr1_26827458_C_Gchr1:268274580.0280.0300.241—   
chr1_26827467_G_Cchr1:26827467-0.030-0.030-0.241<0.001%
chr1_26864805_C_Achr1:26864805-0.136-0.018-0.200—   
chr1_26864793_A_Gchr1:268647930.133-0.1320.224—   
chr1_26864794_T_Gchr1:268647940.133-0.1370.235—   
chr1_26864806_G_Cchr1:26864806-0.126-0.036-0.235—   
chr1_26864719_G_Tchr1:268647190.130-0.036-0.035—   
chr1_26864781_C_Achr1:268647810.1300.0630.224<0.001%
chr1_26864861_C_Achr1:268648610.1300.0250.000—   
chr1_26827469_C_Achr1:268274690.0470.0470.224—   
chr1_26827474_T_Cchr1:26827474-0.046-0.036-0.224—   
chr1_26864709_G_Cchr1:268647090.0700.0030.224<0.001%
chr1_26864710_G_Cchr1:268647100.1060.0380.224—   
chr1_26864745_C_Gchr1:26864745-0.067-0.056-0.224—   
chr1_26864752_T_Achr1:26864752-0.0670.0230.224<0.001%
chr1_26864763_G_Achr1:268647630.1260.0410.094<0.001%
chr1_26864775_T_Gchr1:268647750.100-0.0690.224—   
chr1_26864820_C_Achr1:26864820-0.073-0.036-0.224—   
chr1_26827468_C_Gchr1:268274680.0220.0230.218—   
chr1_26864770_A_Cchr1:26864770-0.123-0.1780.047—   
chr1_26864820_C_Tchr1:26864820-0.123-0.013-0.141—   
chr1_26864846_G_Cchr1:268648460.123-0.0410.165—   
chr1_26864874_C_Tchr1:268648740.1230.015-0.024—   
chr1_26827521_C_Gchr1:268275210.0270.0230.212—   
chr1_26827536_T_Cchr1:26827536-0.037-0.038-0.212—   
chr1_26864711_G_Cchr1:268647110.053-0.0030.2120.0066%
chr1_26864745_C_Tchr1:26864745-0.030-0.046-0.212—   
chr1_26864802_C_Gchr1:26864802-0.080-0.020-0.212—   
chr1_26864806_G_Achr1:26864806-0.120-0.061-0.200—   
chr1_26864806_G_Tchr1:26864806-0.113-0.046-0.212—   
chr1_26864810_C_Achr1:26864810-0.120-0.056-0.153—   
chr1_26864835_G_Cchr1:26864835-0.120-0.033-0.012—   
chr1_26827561_C_Gchr1:268275610.0570.0390.206—   
chr1_26864719_G_Achr1:268647190.116-0.0050.000—   
chr1_26864770_A_Gchr1:26864770-0.116-0.201-0.129—   
chr1_26864805_C_Gchr1:26864805-0.116-0.030-0.071—   
chr1_26864843_G_Tchr1:268648430.1160.074-0.153—   
chr1_26864728_A_Gchr1:268647280.1130.0030.059—   
chr1_26864733_G_Tchr1:26864733-0.013-0.018-0.200—   
chr1_26864745_C_Achr1:26864745-0.037-0.038-0.200—   
chr1_26864747_A_Tchr1:268647470.0670.0660.200—   
chr1_26864790_G_Cchr1:268647900.113-0.0080.118—   
chr1_26864796_T_Gchr1:268647960.070-0.0580.200—   
chr1_26864805_C_Tchr1:26864805-0.113-0.0130.024—   
chr1_26864807_C_Tchr1:26864807-0.113-0.038-0.071—   
chr1_26864813_T_Gchr1:26864813-0.113-0.025-0.106—   
chr1_26864830_C_Achr1:268648300.003-0.020-0.200—   
chr1_26864847_G_Achr1:26864847-0.013-0.0150.200—   
chr1_26864859_A_Gchr1:268648590.050-0.0100.200—   
chr1_26864860_T_Gchr1:268648600.1030.0050.200—   
chr1_26864864_G_Achr1:26864864-0.1130.018-0.165<0.001%
chr1_26827470_C_Tchr1:268274700.0360.0190.194—   
chr1_26827471_C_Achr1:268274710.0290.0280.194—   
chr1_26827556_A_Cchr1:26827556-0.042-0.036-0.194—   
chr1_26827560_C_Gchr1:268275600.0350.0250.194—   
chr1_26864765_C_Gchr1:26864765-0.110-0.074-0.047—   
chr1_26827474_T_Gchr1:268274740.0090.0130.188—   
chr1_26827559_C_Gchr1:268275590.0290.0280.188—   
chr1_26864734_C_Achr1:26864734-0.023-0.023-0.188<0.001%
chr1_26864743_G_Tchr1:26864743-0.053-0.003-0.188—   
chr1_26864765_C_Achr1:26864765-0.106-0.145-0.141—   
chr1_26864774_G_Achr1:26864774-0.070-0.043-0.188—   
chr1_26864814_A_Tchr1:26864814-0.106-0.038-0.188—   
chr1_26864824_A_Tchr1:26864824-0.027-0.041-0.188—   
chr1_26864850_C_Gchr1:26864850-0.106-0.036-0.153—   
chr1_26864851_A_Tchr1:26864851-0.043-0.069-0.188—   
chr1_26864855_T_Gchr1:268648550.0400.1020.188—   
chr1_26864875_T_Cchr1:268648750.037-0.0510.188—   
chr1_26864892_G_Achr1:26864892-0.013-0.018-0.188—   
chr1_26827444_A_Cchr1:26827444-0.027-0.025-0.182—   
chr1_26864751_C_Tchr1:26864751-0.103-0.010-0.059—   
chr1_26864769_A_Cchr1:26864769-0.103-0.1700.024—   
chr1_26864772_T_Cchr1:26864772-0.103-0.038-0.047<0.001%
chr1_26864773_A_Cchr1:26864773-0.103-0.0480.000<0.001%
chr1_26864803_A_Cchr1:26864803-0.103-0.030-0.012—   
chr1_26864803_A_Tchr1:26864803-0.1030.030-0.082—   
chr1_26864835_G_Achr1:26864835-0.103-0.010-0.106—   
chr1_26864862_A_Cchr1:268648620.103-0.0280.071—   
chr1_26827448_G_Cchr1:26827448-0.032-0.026-0.176—   
chr1_26827460_C_Gchr1:268274600.0310.0220.176—   
chr1_26827473_A_Gchr1:268274730.0120.0150.176—   
chr1_26827522_C_Gchr1:268275220.0420.0200.176—   
chr1_26827533_C_Gchr1:268275330.0250.0030.176—   
chr1_26864716_T_Achr1:268647160.093-0.041-0.176—   
chr1_26864727_C_Gchr1:268647270.0670.0050.176—   
chr1_26864732_C_Achr1:26864732-0.013-0.036-0.176—   
chr1_26864735_G_Cchr1:268647350.1000.018-0.047—   
chr1_26864737_G_Achr1:268647370.1000.0460.059—   
chr1_26864744_A_Tchr1:26864744-0.040-0.018-0.176—   
chr1_26864750_T_Gchr1:26864750-0.030-0.0130.176—   
chr1_26864760_C_Achr1:26864760-0.100-0.053-0.071—   
chr1_26864773_A_Tchr1:26864773-0.1000.003-0.082—   
chr1_26864791_A_Cchr1:268647910.100-0.0460.153—   
chr1_26864797_A_Cchr1:268647970.100-0.0990.106—   
chr1_26864821_G_Tchr1:268648210.003-0.013-0.176—   
chr1_26864827_G_Tchr1:26864827-0.087-0.033-0.176—   
chr1_26864847_G_Cchr1:26864847-0.017-0.0080.176—   
chr1_26827482_G_Cchr1:26827482-0.026-0.034-0.171—   
chr1_26827531_A_Cchr1:26827531-0.032-0.030-0.171—   
chr1_26827560_C_Achr1:268275600.0330.0230.1710.0020%
chr1_26864705_C_Achr1:26864705-0.097-0.069-0.165—   
chr1_26864739_G_Tchr1:26864739-0.097-0.056-0.082—   
chr1_26864755_T_Achr1:26864755-0.097-0.033-0.035—   
chr1_26864766_A_Gchr1:26864766-0.097-0.1550.000—   
chr1_26864767_G_Cchr1:26864767-0.097-0.1600.059—   
chr1_26864808_C_Tchr1:26864808-0.097-0.041-0.165—   
chr1_26864854_G_Cchr1:26864854-0.097-0.033-0.047—   
chr1_26827459_C_Achr1:268274590.0340.0320.165—   
chr1_26827459_C_Tchr1:268274590.0420.0290.1650.0033%
chr1_26827464_A_Gchr1:268274640.0070.0080.165—   
chr1_26827471_C_Tchr1:268274710.0390.0300.1650.0033%
chr1_26827495_C_Gchr1:268274950.0020.0090.165—   
chr1_26827518_G_Cchr1:26827518-0.030-0.011-0.165—   
chr1_26827522_C_Achr1:268275220.0330.0210.165—   
chr1_26827559_C_Achr1:268275590.0320.0290.1650.0013%
chr1_26827560_C_Tchr1:268275600.0330.0230.165—   
chr1_26864708_A_Gchr1:268647080.0230.046-0.165—   
chr1_26864737_G_Tchr1:268647370.0930.0630.000—   
chr1_26864743_G_Cchr1:26864743-0.073-0.030-0.165—   
chr1_26864751_C_Gchr1:26864751-0.093-0.013-0.071—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.