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NR0B2

receptor: FXRTier 1

Drug substrates

bile-acid synthesis modulators

refs: 25198545

CAMIP causal chains

FXR

Blunted receptor-mediated induction of NR0B2 expression, weakening the downstream transcriptional feedback inhibition of hepatic bile acid synthesis pathways.

Affected substrate drugs (PharmGKB): none in routine clinical use, endogenous or bile acid pathway

Scored variants near NR0B2

chr1:26,811,488..27,013,975, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr1_26864748_G_Cchr1:268647480.8210.093-0.058—   
chr1_26827461_T_Cchr1:26827461-0.079-0.043-0.456—   
chr1_26864772_T_Achr1:26864772-0.258-0.141-0.152—   
chr1_26827451_T_Cchr1:26827451-0.071-0.079-0.450—   
chr1_26864718_A_Gchr1:26864718-0.123-0.065-0.421—   
chr1_26864782_T_Achr1:268647820.0830.1760.421—   
chr1_26864833_C_Gchr1:268648330.0560.0130.421—   
chr1_26864758_A_Gchr1:268647580.1790.0930.409—   
chr1_26864722_G_Cchr1:268647220.2280.0350.187—   
chr1_26827486_T_Cchr1:26827486-0.060-0.072-0.398—   
chr1_26864734_C_Gchr1:26864734-0.146-0.015-0.386—   
chr1_26864789_T_Gchr1:26864789-0.169-0.035-0.386—   
chr1_26864722_G_Achr1:268647220.2150.0330.047—   
chr1_26827523_T_Cchr1:26827523-0.075-0.032-0.374—   
chr1_26864713_A_Gchr1:268647130.0000.040-0.374—   
chr1_26864798_A_Tchr1:268647980.209-0.1390.199—   
chr1_26864716_T_Gchr1:26864716-0.013-0.020-0.363—   
chr1_26864778_A_Cchr1:26864778-0.0300.2140.363—   
chr1_26864832_C_Tchr1:26864832-0.116-0.081-0.3630.0013%
chr1_26827470_C_Gchr1:268274700.0420.0510.357—   
chr1_26864720_T_Cchr1:268647200.2020.0100.070—   
chr1_26864722_G_Tchr1:268647220.2020.0350.058—   
chr1_26864741_C_Achr1:268647410.0790.0730.351—   
chr1_26864820_C_Gchr1:26864820-0.199-0.118-0.222—   
chr1_26827464_A_Cchr1:26827464-0.033-0.055-0.333—   
chr1_26864760_C_Gchr1:26864760-0.189-0.060-0.2220.062%
chr1_26827529_T_Cchr1:26827529-0.070-0.099-0.327—   
chr1_26864721_G_Cchr1:268647210.1850.0150.222—   
chr1_26864734_C_Tchr1:26864734-0.185-0.025-0.222—   
chr1_26864813_T_Achr1:26864813-0.185-0.018-0.257—   
chr1_26864719_G_Cchr1:268647190.1790.005-0.047—   
chr1_26827469_C_Gchr1:268274690.0470.0500.310—   
chr1_26864781_C_Tchr1:268647810.1750.1490.187<0.001%
chr1_26864811_A_Cchr1:268648110.1750.0680.152—   
chr1_26864732_C_Gchr1:26864732-0.030-0.015-0.304—   
chr1_26864822_G_Cchr1:268648220.1230.0710.304—   
chr1_26864755_T_Gchr1:26864755-0.169-0.008-0.140—   
chr1_26864721_G_Achr1:268647210.1660.0180.082—   
chr1_26864724_A_Gchr1:26864724-0.073-0.030-0.292—   
chr1_26864794_T_Cchr1:268647940.149-0.1010.292—   
chr1_26864796_T_Achr1:26864796-0.1490.280-0.292—   
chr1_26827459_C_Gchr1:268274590.0360.0360.287—   
chr1_26864769_A_Gchr1:26864769-0.162-0.209-0.047—   
chr1_26864720_T_Achr1:268647200.1590.015-0.035—   
chr1_26864771_A_Tchr1:26864771-0.159-0.174-0.082—   
chr1_26864781_C_Gchr1:26864781-0.106-0.0980.281—   
chr1_26864792_G_Tchr1:268647920.159-0.0600.211—   
chr1_26864801_A_Tchr1:268648010.1030.0350.281—   
chr1_26864831_A_Cchr1:26864831-0.159-0.126-0.246—   
chr1_26827477_T_Cchr1:26827477-0.038-0.052-0.275—   
chr1_26864738_A_Gchr1:26864738-0.156-0.055-0.2570.0013%
chr1_26864792_G_Achr1:268647920.156-0.0810.035—   
chr1_26864793_A_Cchr1:268647930.156-0.1160.246—   
chr1_26864712_G_Cchr1:268647120.1030.0400.269—   
chr1_26864746_G_Achr1:26864746-0.089-0.023-0.269<0.001%
chr1_26864747_A_Cchr1:268647470.1520.0180.140—   
chr1_26864772_T_Gchr1:26864772-0.152-0.111-0.023—   
chr1_26864802_C_Achr1:26864802-0.099-0.033-0.269—   
chr1_26827472_C_Gchr1:268274720.0580.0370.263—   
chr1_26827466_G_Cchr1:26827466-0.040-0.041-0.257—   
chr1_26864766_A_Cchr1:268647660.142-0.0050.257—   
chr1_26864797_A_Tchr1:268647970.146-0.0650.175—   
chr1_26864798_A_Cchr1:268647980.132-0.0910.257—   
chr1_26827456_G_Cchr1:26827456-0.023-0.037-0.251—   
chr1_26827470_C_Achr1:268274700.0410.0380.251—   
chr1_26827557_A_Cchr1:26827557-0.042-0.021-0.251—   
chr1_26864771_A_Gchr1:268647710.1420.1060.246—   
chr1_26864774_G_Tchr1:26864774-0.142-0.065-0.234—   
chr1_26864794_T_Achr1:268647940.142-0.1110.012—   
chr1_26827471_C_Gchr1:268274710.0320.0140.246—   
chr1_26827479_G_Cchr1:26827479-0.025-0.038-0.246—   
chr1_26864720_T_Gchr1:268647200.0630.015-0.246—   
chr1_26864721_G_Tchr1:268647210.139-0.0080.058—   
chr1_26864723_G_Tchr1:268647230.1390.0200.023—   
chr1_26864743_G_Achr1:26864743-0.139-0.050-0.152—   
chr1_26864787_C_Gchr1:268647870.020-0.058-0.246—   
chr1_26864795_C_Achr1:268647950.139-0.0880.152—   
chr1_26864839_T_Achr1:268648390.1390.0100.117—   
chr1_26864863_A_Cchr1:268648630.0600.0380.246—   
chr1_26864863_A_Tchr1:268648630.0170.0200.246—   
chr1_26827458_C_Gchr1:268274580.0280.0300.240—   
chr1_26827467_G_Cchr1:26827467-0.030-0.030-0.240<0.001%
chr1_26864805_C_Achr1:26864805-0.136-0.018-0.199—   
chr1_26864793_A_Gchr1:268647930.132-0.1310.222—   
chr1_26864794_T_Gchr1:268647940.132-0.1360.234—   
chr1_26864806_G_Cchr1:26864806-0.126-0.035-0.234—   
chr1_26864719_G_Tchr1:268647190.129-0.035-0.035—   
chr1_26864781_C_Achr1:268647810.1290.0630.222<0.001%
chr1_26864861_C_Achr1:268648610.1290.0250.000—   
chr1_26827469_C_Achr1:268274690.0460.0470.222—   
chr1_26827474_T_Cchr1:26827474-0.046-0.035-0.222—   
chr1_26864709_G_Cchr1:268647090.0700.0030.222<0.001%
chr1_26864710_G_Cchr1:268647100.1060.0380.222—   
chr1_26864745_C_Gchr1:26864745-0.066-0.055-0.222—   
chr1_26864752_T_Achr1:26864752-0.0660.0230.222<0.001%
chr1_26864763_G_Achr1:268647630.1260.0400.094<0.001%
chr1_26864775_T_Gchr1:268647750.099-0.0680.222—   
chr1_26864820_C_Achr1:26864820-0.073-0.035-0.222—   
chr1_26827468_C_Gchr1:268274680.0220.0230.216—   
chr1_26864770_A_Cchr1:26864770-0.123-0.1760.047—   
chr1_26864820_C_Tchr1:26864820-0.123-0.013-0.140—   
chr1_26864846_G_Cchr1:268648460.123-0.0400.164—   
chr1_26864874_C_Tchr1:268648740.1230.015-0.023—   
chr1_26827521_C_Gchr1:268275210.0260.0230.211—   
chr1_26827536_T_Cchr1:26827536-0.037-0.038-0.211—   
chr1_26864711_G_Cchr1:268647110.053-0.0030.2110.0066%
chr1_26864745_C_Tchr1:26864745-0.030-0.045-0.211—   
chr1_26864802_C_Gchr1:26864802-0.079-0.020-0.211—   
chr1_26864806_G_Achr1:26864806-0.119-0.060-0.199—   
chr1_26864806_G_Tchr1:26864806-0.113-0.045-0.211—   
chr1_26864810_C_Achr1:26864810-0.119-0.055-0.152—   
chr1_26864835_G_Cchr1:26864835-0.119-0.033-0.012—   
chr1_26827561_C_Gchr1:268275610.0560.0390.205—   
chr1_26864719_G_Achr1:268647190.116-0.0050.000—   
chr1_26864770_A_Gchr1:26864770-0.116-0.199-0.129—   
chr1_26864805_C_Gchr1:26864805-0.116-0.030-0.070—   
chr1_26864843_G_Tchr1:268648430.1160.073-0.152—   
chr1_26864728_A_Gchr1:268647280.1130.0030.058—   
chr1_26864733_G_Tchr1:26864733-0.013-0.018-0.199—   
chr1_26864745_C_Achr1:26864745-0.036-0.038-0.199—   
chr1_26864747_A_Tchr1:268647470.0660.0650.199—   
chr1_26864790_G_Cchr1:268647900.113-0.0080.117—   
chr1_26864796_T_Gchr1:268647960.070-0.0580.199—   
chr1_26864805_C_Tchr1:26864805-0.113-0.0130.023—   
chr1_26864807_C_Tchr1:26864807-0.113-0.038-0.070—   
chr1_26864813_T_Gchr1:26864813-0.113-0.025-0.105—   
chr1_26864830_C_Achr1:268648300.003-0.020-0.199—   
chr1_26864847_G_Achr1:26864847-0.013-0.0150.199—   
chr1_26864859_A_Gchr1:268648590.050-0.0100.199—   
chr1_26864860_T_Gchr1:268648600.1030.0050.199—   
chr1_26864864_G_Achr1:26864864-0.1130.018-0.164<0.001%
chr1_26827470_C_Tchr1:268274700.0360.0190.193—   
chr1_26827471_C_Achr1:268274710.0290.0280.193—   
chr1_26827556_A_Cchr1:26827556-0.041-0.035-0.193—   
chr1_26827560_C_Gchr1:268275600.0350.0250.193—   
chr1_26864765_C_Gchr1:26864765-0.109-0.073-0.047—   
chr1_26827474_T_Gchr1:268274740.0090.0130.187—   
chr1_26827559_C_Gchr1:268275590.0290.0280.187—   
chr1_26864734_C_Achr1:26864734-0.023-0.023-0.187<0.001%
chr1_26864743_G_Tchr1:26864743-0.053-0.003-0.187—   
chr1_26864765_C_Achr1:26864765-0.106-0.144-0.140—   
chr1_26864774_G_Achr1:26864774-0.070-0.043-0.187—   
chr1_26864814_A_Tchr1:26864814-0.106-0.038-0.187—   
chr1_26864824_A_Tchr1:26864824-0.026-0.040-0.187—   
chr1_26864850_C_Gchr1:26864850-0.106-0.035-0.152—   
chr1_26864851_A_Tchr1:26864851-0.043-0.068-0.187—   
chr1_26864855_T_Gchr1:268648550.0400.1010.187—   
chr1_26864875_T_Cchr1:268648750.036-0.0500.187—   
chr1_26864892_G_Achr1:26864892-0.013-0.018-0.187—   
chr1_26827444_A_Cchr1:26827444-0.027-0.025-0.181—   
chr1_26864751_C_Tchr1:26864751-0.103-0.010-0.058—   
chr1_26864769_A_Cchr1:26864769-0.103-0.1690.023—   
chr1_26864772_T_Cchr1:26864772-0.103-0.038-0.047<0.001%
chr1_26864773_A_Cchr1:26864773-0.103-0.0480.000<0.001%
chr1_26864803_A_Cchr1:26864803-0.103-0.030-0.012—   
chr1_26864803_A_Tchr1:26864803-0.1030.030-0.082—   
chr1_26864835_G_Achr1:26864835-0.103-0.010-0.105—   
chr1_26864862_A_Cchr1:268648620.103-0.0280.070—   
chr1_26827448_G_Cchr1:26827448-0.031-0.026-0.175—   
chr1_26827460_C_Gchr1:268274600.0310.0220.175—   
chr1_26827473_A_Gchr1:268274730.0120.0150.175—   
chr1_26827522_C_Gchr1:268275220.0410.0200.175—   
chr1_26827533_C_Gchr1:268275330.0250.0030.175—   
chr1_26864716_T_Achr1:268647160.093-0.040-0.175—   
chr1_26864727_C_Gchr1:268647270.0660.0050.175—   
chr1_26864732_C_Achr1:26864732-0.013-0.035-0.175—   
chr1_26864735_G_Cchr1:268647350.0990.018-0.047—   
chr1_26864737_G_Achr1:268647370.0990.0450.058—   
chr1_26864744_A_Tchr1:26864744-0.040-0.018-0.175—   
chr1_26864750_T_Gchr1:26864750-0.030-0.0130.175—   
chr1_26864760_C_Achr1:26864760-0.099-0.053-0.070—   
chr1_26864773_A_Tchr1:26864773-0.0990.003-0.082—   
chr1_26864791_A_Cchr1:268647910.099-0.0450.152—   
chr1_26864797_A_Cchr1:268647970.099-0.0980.105—   
chr1_26864821_G_Tchr1:268648210.003-0.013-0.175—   
chr1_26864827_G_Tchr1:26864827-0.086-0.033-0.175—   
chr1_26864847_G_Cchr1:26864847-0.017-0.0080.175—   
chr1_26827482_G_Cchr1:26827482-0.026-0.033-0.170—   
chr1_26827531_A_Cchr1:26827531-0.031-0.030-0.170—   
chr1_26827560_C_Achr1:268275600.0330.0230.1700.0020%
chr1_26864705_C_Achr1:26864705-0.096-0.068-0.164—   
chr1_26864739_G_Tchr1:26864739-0.096-0.055-0.082—   
chr1_26864755_T_Achr1:26864755-0.096-0.033-0.035—   
chr1_26864766_A_Gchr1:26864766-0.096-0.1540.000—   
chr1_26864767_G_Cchr1:26864767-0.096-0.1590.058—   
chr1_26864808_C_Tchr1:26864808-0.096-0.040-0.164—   
chr1_26864854_G_Cchr1:26864854-0.096-0.033-0.047—   
chr1_26827459_C_Achr1:268274590.0340.0320.164—   
chr1_26827459_C_Tchr1:268274590.0410.0290.1640.0033%
chr1_26827464_A_Gchr1:268274640.0070.0080.164—   
chr1_26827471_C_Tchr1:268274710.0390.0300.1640.0033%
chr1_26827495_C_Gchr1:268274950.0020.0090.164—   
chr1_26827518_G_Cchr1:26827518-0.030-0.011-0.164—   
chr1_26827522_C_Achr1:268275220.0330.0210.164—   
chr1_26827559_C_Achr1:268275590.0320.0290.1640.0013%
chr1_26827560_C_Tchr1:268275600.0330.0230.164—   
chr1_26864708_A_Gchr1:268647080.0230.045-0.164—   
chr1_26864737_G_Tchr1:268647370.0930.0630.000—   
chr1_26864743_G_Cchr1:26864743-0.073-0.030-0.164—   
chr1_26864751_C_Gchr1:26864751-0.093-0.013-0.070—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.