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SLC10A1

receptor: FXRTier 1

Drug substrates

rosuvastatin; bile acids (NTCP is also the HBV/HDV entry receptor)

refs: 25198545

CAMIP causal chains

FXR

Reduced FXR binding would weaken FXR-driven SHP induction; with SHP-mediated repression relieved, SLC10A1/NTCP expression would rise, thus increasing the hepatic clearance of NTCP substrates.

Affected substrate drugs (PharmGKB): rosuvastatin

Scored variants near SLC10A1

chr14:69,675,415..69,897,241, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr14_69685917_G_Achr14:696859171.0001.0001.000—   
chr14_69685885_T_Gchr14:696858851.0001.0001.000—   
chr14_69685888_G_Cchr14:696858881.0001.0001.000—   
chr14_69685888_G_Achr14:696858881.0001.0001.000—   
chr14_69685844_A_Cchr14:696858441.0001.0001.000—   
chr14_69685844_A_Tchr14:696858441.0001.0001.000—   
chr14_69685913_A_Cchr14:696859131.0001.0001.000—   
chr14_69685862_T_Achr14:696858621.0001.0001.000—   
chr14_69685899_G_Tchr14:696858991.0000.3900.474—   
chr14_69685905_A_Cchr14:69685905-1.000-0.942-1.000—   
chr14_69685939_C_Tchr14:69685939-1.000-0.899-1.000—   
chr14_69685937_G_Cchr14:69685937-1.000-0.834-1.000—   
chr14_69685866_T_Cchr14:696858661.0001.0001.000—   
chr14_69685939_C_Achr14:69685939-1.000-0.859-1.000—   
chr14_69685862_T_Gchr14:696858621.0001.0001.000—   
chr14_69685937_G_Achr14:69685937-1.000-0.811-1.000—   
chr14_69685939_C_Gchr14:69685939-1.000-0.887-1.000—   
chr14_69685872_G_Cchr14:696858721.0001.0000.971—   
chr14_69685938_C_Tchr14:69685938-1.000-0.655-1.000—   
chr14_69685871_T_Gchr14:696858711.0001.0000.760—   
chr14_69685938_C_Achr14:69685938-1.000-0.650-1.000—   
chr14_69685930_G_Tchr14:69685930-1.000-0.567-1.000—   
chr14_69685899_G_Cchr14:696858991.0000.8040.988—   
chr14_69685885_T_Achr14:696858851.0000.8720.924—   
chr14_69685929_G_Tchr14:69685929-1.000-0.597-1.000—   
chr14_69685941_G_Cchr14:69685941-1.000-0.567-0.901—   
chr14_69685929_G_Achr14:69685929-1.000-0.592-1.000—   
chr14_69685931_C_Tchr14:69685931-1.000-0.549-0.924—   
chr14_69685930_G_Achr14:69685930-1.000-0.494-1.000—   
chr14_69685929_G_Cchr14:69685929-1.000-0.635-1.000—   
chr14_69685930_G_Cchr14:69685930-1.000-0.494-0.959—   
chr14_69685895_C_Tchr14:696858951.0000.8140.842—   
chr14_69685888_G_Tchr14:696858881.0000.7860.883—   
chr14_69685931_C_Gchr14:69685931-1.000-0.458-0.860—   
chr14_69685915_C_Gchr14:69685915-1.000-0.753-1.000—   
chr14_69685914_G_Cchr14:696859141.0000.7460.567—   
chr14_69685907_C_Gchr14:69685907-1.000-0.685-0.737—   
chr14_69685920_G_Tchr14:69685920-1.000-0.635-1.000—   
chr14_69685928_T_Cchr14:69685928-1.000-0.574-0.977—   
chr14_69685862_T_Cchr14:696858621.0000.8360.737—   
chr14_69685940_A_Tchr14:69685940-1.000-0.574-0.942—   
chr14_69685941_G_Tchr14:69685941-1.000-0.524-0.787—   
chr14_69685937_G_Tchr14:69685937-0.997-0.597-0.906—   
chr14_69685938_C_Gchr14:69685938-0.995-0.506-0.827—   
chr14_69685962_G_Tchr14:69685962-0.980-0.453-0.874—   
chr14_69685950_A_Cchr14:69685950-0.969-0.395-0.787—   
chr14_69685907_C_Tchr14:69685907-0.964-0.690-0.772—   
chr14_69685940_A_Gchr14:69685940-0.954-0.675-0.971—   
chr14_69685928_T_Achr14:69685928-0.930-0.519-0.909—   
chr14_69685880_A_Tchr14:69685880-0.924-0.741-0.927—   
chr14_69685849_C_Gchr14:69685849-0.916-0.761-1.000—   
chr14_69685877_T_Achr14:69685877-0.881-0.668-0.731—   
chr14_69685928_T_Gchr14:69685928-0.876-0.537-0.924—   
chr14_69685874_A_Cchr14:696858740.8730.8360.895—   
chr14_69685886_G_Tchr14:69685886-0.866-0.662-0.895—   
chr14_69685878_G_Achr14:69685878-0.863-0.599-0.863—   
chr14_69685882_T_Achr14:69685882-0.863-0.594-0.737—   
chr14_69685884_T_Achr14:69685884-0.851-0.652-0.795—   
chr14_69685878_G_Cchr14:69685878-0.844-0.574-0.827—   
chr14_69685877_T_Gchr14:69685877-0.841-0.660-0.728—   
chr14_69685879_G_Cchr14:69685879-0.831-0.743-0.690—   
chr14_69685927_G_Tchr14:696859270.8280.4310.678—   
chr14_69685886_G_Achr14:69685886-0.806-0.592-0.661—   
chr14_69685881_C_Gchr14:69685881-0.793-0.685-0.810—   
chr14_69685882_T_Cchr14:696858820.7930.6700.667—   
chr14_69685880_A_Gchr14:69685880-0.788-0.670-0.810—   
chr14_69685910_T_Gchr14:696859100.7850.7331.000—   
chr14_69685861_C_Gchr14:696858610.7830.6980.661<0.001%
chr14_69685879_G_Tchr14:69685879-0.773-0.594-0.851—   
chr14_69685860_C_Tchr14:69685860-0.770-0.617-0.731—   
chr14_69685907_C_Achr14:69685907-0.760-0.418-0.544—   
chr14_69685927_G_Cchr14:696859270.7520.2900.690—   
chr14_69685915_C_Achr14:69685915-0.750-0.526-0.749—   
chr14_69685940_A_Cchr14:69685940-0.750-0.426-0.635—   
chr14_69685878_G_Tchr14:69685878-0.740-0.524-0.766—   
chr14_69685886_G_Cchr14:69685886-0.737-0.599-0.716—   
chr14_69685845_T_Cchr14:696858450.7320.6250.690—   
chr14_69685852_C_Achr14:696858520.7280.5190.520—   
chr14_69685881_C_Tchr14:69685881-0.728-0.620-0.848—   
chr14_69685971_G_Tchr14:69685971-0.717-0.287-0.667—   
chr14_69685913_A_Tchr14:696859130.7120.5060.626—   
chr14_69685877_T_Cchr14:69685877-0.699-0.567-0.561—   
chr14_69685908_T_Cchr14:69685908-0.690-0.486-0.740—   
chr14_69685889_C_Gchr14:69685889-0.680-0.534-0.629—   
chr14_69685884_T_Gchr14:69685884-0.667-0.529-0.591—   
chr14_69685828_C_Gchr14:69685828-0.657-0.605-0.713—   
chr14_69685851_C_Tchr14:69685851-0.652-0.516-0.6140.0020%
chr14_69685876_T_Achr14:69685876-0.652-0.469-0.594—   
chr14_69685853_C_Gchr14:696858530.6490.5040.713—   
chr14_69685825_G_Achr14:69685825-0.647-0.554-0.690—   
chr14_69685898_A_Gchr14:696858980.6410.4690.538—   
chr14_69685828_C_Achr14:69685828-0.629-0.552-0.784—   
chr14_69685835_A_Cchr14:696858350.6290.4610.444—   
chr14_69685847_G_Cchr14:69685847-0.626-0.496-0.760—   
chr14_69685883_T_Gchr14:69685883-0.621-0.542-0.515—   
chr14_69685891_G_Tchr14:69685891-0.616-0.398-0.532—   
chr14_69685887_T_Achr14:696858870.6140.4760.544—   
chr14_69685858_T_Gchr14:696858580.6110.4560.415—   
chr14_69685894_G_Tchr14:69685894-0.606-0.436-0.640—   
chr14_69685843_A_Gchr14:69685843-0.603-0.373-0.772<0.001%
chr14_69685933_G_Tchr14:69685933-0.603-0.184-0.219—   
chr14_69685829_T_Gchr14:69685829-0.601-0.496-0.515—   
chr14_69685898_A_Tchr14:696858980.5990.4740.538—   
chr14_69685889_C_Achr14:69685889-0.589-0.486-0.535—   
chr14_69685832_G_Cchr14:69685832-0.588-0.219-0.251—   
chr14_69685882_T_Gchr14:69685882-0.586-0.474-0.404—   
chr14_69685915_C_Tchr14:69685915-0.584-0.423-0.556—   
chr14_69685859_G_Tchr14:69685859-0.568-0.378-0.345—   
chr14_69685936_T_Cchr14:69685936-0.568-0.355-0.444—   
chr14_69685819_C_Gchr14:69685819-0.566-0.597-0.678—   
chr14_69685829_T_Achr14:69685829-0.561-0.474-0.532—   
chr14_69685914_G_Tchr14:696859140.5560.4560.322—   
chr14_69685883_T_Achr14:69685883-0.553-0.491-0.491—   
chr14_69685970_A_Cchr14:69685970-0.551-0.204-0.383—   
chr14_69685818_A_Cchr14:69685818-0.546-0.448-0.526—   
chr14_69685875_T_Cchr14:696858750.5430.5210.392—   
chr14_69685967_G_Cchr14:69685967-0.540-0.227-0.491—   
chr14_69685872_G_Tchr14:69685872-0.538-0.403-0.652—   
chr14_69685884_T_Cchr14:69685884-0.538-0.456-0.439—   
chr14_69685831_T_Achr14:69685831-0.536-0.370-0.474—   
chr14_69685923_A_Tchr14:696859230.5280.2420.480—   
chr14_69685820_A_Cchr14:69685820-0.526-0.476-0.515—   
chr14_69685895_C_Gchr14:69685895-0.525-0.171-0.310—   
chr14_69685900_A_Cchr14:696859000.5250.3950.444—   
chr14_69685860_C_Achr14:696858600.5220.3930.327—   
chr14_69685948_G_Tchr14:69685948-0.518-0.252-0.547—   
chr14_69685847_G_Achr14:69685847-0.517-0.421-0.673—   
chr14_69685973_T_Cchr14:69685973-0.517-0.242-0.468—   
chr14_69685969_C_Achr14:69685969-0.515-0.234-0.447—   
chr14_69685887_T_Gchr14:696858870.5070.3450.421—   
chr14_69685842_A_Gchr14:69685842-0.505-0.375-0.673—   
chr14_69685931_C_Achr14:69685931-0.503-0.212-0.398—   
chr14_69685867_G_Cchr14:69685867-0.500-0.411-0.538—   
chr14_69685855_G_Tchr14:69685855-0.497-0.363-0.439—   
chr14_69685847_G_Tchr14:69685847-0.493-0.406-0.673—   
chr14_69741167_T_Achr14:69741167-0.492-0.421-0.787—   
chr14_69685880_A_Cchr14:69685880-0.490-0.466-0.386—   
chr14_69685819_C_Achr14:69685819-0.485-0.577-0.608—   
chr14_69685920_G_Achr14:696859200.4830.3800.5610.0020%
chr14_69685971_G_Cchr14:69685971-0.482-0.076-0.368<0.001%
chr14_69685866_T_Gchr14:69685866-0.480-0.312-0.421—   
chr14_69685853_C_Achr14:696858530.4770.3550.491—   
chr14_69685871_T_Achr14:696858710.4750.3580.228—   
chr14_69685887_T_Cchr14:696858870.4750.3780.556—   
chr14_69685897_G_Achr14:69685897-0.474-0.416-0.444—   
chr14_69685838_T_Cchr14:696858380.4720.3270.480—   
chr14_69685889_C_Tchr14:69685889-0.472-0.375-0.398—   
chr14_69685824_T_Gchr14:69685824-0.467-0.506-0.544—   
chr14_69685869_A_Tchr14:69685869-0.465-0.416-0.491—   
chr14_69685871_T_Cchr14:696858710.4620.3300.462—   
chr14_69685818_A_Tchr14:69685818-0.459-0.388-0.444—   
chr14_69685855_G_Achr14:69685855-0.459-0.285-0.433<0.001%
chr14_69685866_T_Achr14:69685866-0.457-0.275-0.357—   
chr14_69685872_G_Achr14:69685872-0.454-0.259-0.380—   
chr14_69685913_A_Gchr14:696859130.4520.2920.368—   
chr14_69685964_C_Achr14:69685964-0.450-0.166-0.436—   
chr14_69685864_T_Achr14:69685864-0.447-0.335-0.485—   
chr14_69685922_G_Achr14:69685922-0.444-0.247-0.275—   
chr14_69685985_G_Tchr14:69685985-0.442-0.161-0.357—   
chr14_69685819_C_Tchr14:69685819-0.440-0.479-0.515—   
chr14_69685841_T_Cchr14:69685841-0.439-0.287-0.491—   
chr14_69685870_A_Tchr14:696858700.4350.2950.363—   
chr14_69685941_G_Achr14:696859410.4300.2390.175—   
chr14_69685864_T_Cchr14:69685864-0.429-0.335-0.485—   
chr14_69685909_C_Achr14:696859090.4270.3120.444—   
chr14_69685924_G_Cchr14:696859240.4270.3530.573—   
chr14_69685850_A_Gchr14:69685850-0.425-0.378-0.468—   
chr14_69685840_G_Cchr14:69685840-0.424-0.360-0.684—   
chr14_69719739_T_Achr14:697197390.0780.1760.749—   
chr14_69685865_G_Tchr14:69685865-0.421-0.322-0.509—   
chr14_69685870_A_Cchr14:696858700.4160.2720.327—   
chr14_69685855_G_Cchr14:69685855-0.414-0.295-0.380—   
chr14_69685921_T_Gchr14:696859210.4140.2370.181—   
chr14_69685952_A_Cchr14:69685952-0.411-0.103-0.287—   
chr14_69685963_C_Gchr14:696859630.4090.0760.246—   
chr14_69685826_T_Cchr14:69685826-0.407-0.348-0.404—   
chr14_69685869_A_Gchr14:69685869-0.407-0.224-0.2690.0013%
chr14_69685958_A_Gchr14:696859580.4060.2700.409—   
chr14_69685970_A_Gchr14:69685970-0.404-0.189-0.327—   
chr14_69685897_G_Cchr14:696858970.3990.2770.281—   
chr14_69685894_G_Cchr14:69685894-0.396-0.113-0.287—   
chr14_69685881_C_Achr14:69685881-0.392-0.297-0.152—   
chr14_69685896_T_Cchr14:696858960.3920.2370.287—   
chr14_69685843_A_Tchr14:69685843-0.391-0.275-0.602—   
chr14_69685900_A_Tchr14:696859000.3910.3120.532—   
chr14_69685865_G_Cchr14:69685865-0.389-0.317-0.462—   
chr14_69685825_G_Cchr14:69685825-0.387-0.406-0.409—   
chr14_69685863_T_Achr14:69685863-0.387-0.287-0.257—   
chr14_69685841_T_Gchr14:69685841-0.386-0.285-0.485—   
chr14_69685921_T_Achr14:696859210.3860.2290.187—   
chr14_69685981_T_Gchr14:696859810.3860.0150.275—   
chr14_69685828_C_Tchr14:69685828-0.384-0.408-0.503—   
chr14_69685846_T_Achr14:696858460.3840.2590.263—   
chr14_69685856_A_Tchr14:696858560.3790.3200.415—   
chr14_69685919_C_Gchr14:696859190.3790.3630.287—   
chr14_69685977_T_Gchr14:69685977-0.377-0.050-0.123—   
chr14_69685918_T_Gchr14:696859180.3760.3000.374—   
chr14_69685970_A_Tchr14:69685970-0.376-0.139-0.298—   
chr14_69685902_A_Cchr14:696859020.3740.3780.351—   
chr14_69685914_G_Achr14:696859140.3740.3600.281—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.