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SLC51B

receptor: FXRTier 1
Prior gene annotation

Retained explanatory context, not the pharmacist's submitted wording; submitted reviews below take precedence.

Drug substrates (prior annotation)

none in routine clinical use, endogenous or bile acid pathway

refs: 16269519

CAMIP Tier 1: peak-anchored panel

FXR

Submitted decision (verbatim): 需修訂

Reviewer revision (verbatim)

Blunted receptor-mediated induction of SLC51B expression may impair bile salt export from enterocytes and the inducible basolateral bile salt efflux route in hepatocytes under increased intracellular bile salt load.
Prior explanatory context

Retained explanatory context, not the pharmacist's submitted wording. The submitted review above takes precedence; this context is not a replacement for the reviewer's revision or notes.

Inducer
Obeticholic acid; Experimental GW4064
Regulatory element
overlapping TSS
Predicted consequence
Blunted receptor-mediated induction of SLC51B expression, reducing heteromeric basolateral bile acid efflux capacity in hepatocytes and enterocytes.
Prior narrative
Blunted receptor-mediated induction of SLC51B expression, reducing heteromeric basolateral bile acid efflux capacity in hepatocytes and enterocytes.
Drug context
none in routine clinical use, endogenous or bile acid pathway
Prior references
16269519

Scored variants near SLC51B

chr15:64,945,386..65,153,397, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr15_64982020_C_Achr15:64982020-1.000-1.000-1.000—   
chr15_64982024_G_Achr15:64982024-1.000-1.000-1.000—   
chr15_64982022_A_Cchr15:64982022-1.000-1.000-1.000—   
chr15_64982022_A_Tchr15:64982022-1.000-1.000-1.000—   
chr15_64982024_G_Cchr15:64982024-1.000-1.000-1.000—   
chr15_64982020_C_Gchr15:64982020-1.000-1.000-1.000—   
chr15_64982022_A_Gchr15:64982022-1.000-1.000-1.000<0.001%
chr15_64982021_A_Tchr15:64982021-1.000-1.000-1.000—   
chr15_64982027_C_Achr15:64982027-1.000-1.000-1.000—   
chr15_64982027_C_Gchr15:64982027-1.000-1.000-1.000—   
chr15_64982028_A_Cchr15:64982028-1.000-1.000-1.000—   
chr15_64982024_G_Tchr15:64982024-1.000-1.000-1.000—   
chr15_64982025_T_Achr15:64982025-1.000-1.000-1.000—   
chr15_64982025_T_Cchr15:64982025-1.000-1.000-1.000<0.001%
chr15_64982026_C_Gchr15:64982026-1.000-1.000-1.000—   
chr15_64982020_C_Tchr15:64982020-1.000-1.000-1.000—   
chr15_64982023_A_Cchr15:64982023-1.000-1.000-1.000—   
chr15_64982023_A_Tchr15:64982023-1.000-1.000-1.000—   
chr15_64982025_T_Gchr15:64982025-1.000-1.000-1.000—   
chr15_64982027_C_Tchr15:64982027-1.000-1.000-1.000—   
chr15_64982044_T_Gchr15:649820441.0001.0000.941—   
chr15_64982026_C_Achr15:64982026-1.000-1.000-1.000—   
chr15_64982028_A_Tchr15:64982028-1.000-1.000-1.000—   
chr15_64982018_G_Cchr15:64982018-1.000-1.000-1.000—   
chr15_64982023_A_Gchr15:64982023-1.000-1.000-1.000—   
chr15_64982007_A_Cchr15:649820071.0001.0000.976—   
chr15_64981991_A_Gchr15:649819911.0001.0001.000—   
chr15_64982021_A_Gchr15:64982021-1.000-1.000-1.000—   
chr15_64981991_A_Cchr15:649819911.0001.0000.918—   
chr15_64981989_G_Achr15:649819891.0001.0000.788—   
chr15_64981985_A_Tchr15:64981985-1.000-1.000-1.000—   
chr15_64982017_A_Gchr15:649820171.0001.0000.906—   
chr15_64982050_T_Achr15:64982050-1.000-1.000-1.000—   
chr15_64981933_G_Achr15:649819331.0001.0000.647—   
chr15_64982060_C_Achr15:649820601.0001.0000.559—   
chr15_64982021_A_Cchr15:64982021-1.000-1.000-1.000—   
chr15_64981985_A_Cchr15:64981985-1.000-1.000-0.871—   
chr15_64982017_A_Cchr15:64982017-0.976-1.000-1.000—   
chr15_64982011_G_Achr15:649820110.9320.9770.753—   
chr15_64981996_T_Gchr15:649819960.9131.0000.735—   
chr15_64982044_T_Achr15:649820440.9131.0000.576—   
chr15_64981970_A_Cchr15:64981970-0.908-0.886-0.659—   
chr15_64982008_A_Tchr15:64982008-0.894-1.000-0.806—   
chr15_64982049_T_Achr15:64982049-0.889-1.000-1.000—   
chr15_64982004_G_Tchr15:64982004-0.881-0.937-0.606—   
chr15_64982051_G_Achr15:64982051-0.879-1.000-0.882—   
chr15_64982050_T_Gchr15:64982050-0.877-0.975-0.776—   
chr15_64981942_T_Cchr15:64981942-0.875-0.761-0.535—   
chr15_64982026_C_Tchr15:64982026-0.875-0.881-0.818—   
chr15_64982018_G_Achr15:64982018-0.858-0.921-0.794—   
chr15_64982016_A_Cchr15:64982016-0.839-0.949-0.688—   
chr15_64981958_G_Tchr15:64981958-0.815-0.825-0.524—   
chr15_64981963_T_Gchr15:64981963-0.805-0.921-0.935—   
chr15_64982018_G_Tchr15:64982018-0.798-0.868-0.806—   
chr15_64982017_A_Tchr15:64982017-0.782-0.853-0.800—   
chr15_64982048_T_Cchr15:64982048-0.779-0.929-0.671—   
chr15_64981956_C_Tchr15:64981956-0.772-0.698-0.435—   
chr15_64981960_G_Achr15:649819600.7650.0630.324—   
chr15_64982051_G_Tchr15:64982051-0.755-0.904-0.712—   
chr15_64981983_T_Gchr15:64981983-0.745-0.848-0.612—   
chr15_64982033_G_Tchr15:64982033-0.743-0.845-0.829—   
chr15_64982053_A_Gchr15:64982053-0.742-0.959-0.665—   
chr15_64982008_A_Cchr15:64982008-0.721-0.784-0.647—   
chr15_64981988_G_Achr15:64981988-0.718-0.774-0.612—   
chr15_64982051_G_Cchr15:64982051-0.716-0.863-0.582—   
chr15_64982011_G_Tchr15:649820110.7140.7440.576—   
chr15_64982008_A_Gchr15:64982008-0.709-0.774-0.635—   
chr15_64982060_C_Tchr15:64982060-0.709-0.845-0.647—   
chr15_64982045_C_Tchr15:64982045-0.690-0.830-0.682—   
chr15_64982006_T_Achr15:64982006-0.684-0.579-0.471—   
chr15_64981955_T_Cchr15:649819550.6820.2870.453—   
chr15_64982038_A_Tchr15:64982038-0.676-0.673-0.529—   
chr15_64981962_G_Achr15:64981962-0.676-0.693-0.482<0.001%
chr15_64981980_G_Cchr15:64981980-0.676-0.868-0.394—   
chr15_64981988_G_Tchr15:649819880.6710.7060.447—   
chr15_64981957_T_Gchr15:64981957-0.665-0.688-0.518—   
chr15_64981993_C_Gchr15:649819930.6620.7030.600—   
chr15_64982045_C_Achr15:649820450.6530.9310.547—   
chr15_64982047_C_Tchr15:64982047-0.650-0.812-0.718—   
chr15_64982048_T_Achr15:64982048-0.644-0.855-0.576—   
chr15_64982084_T_Achr15:649820840.6410.7590.471—   
chr15_64982050_T_Cchr15:64982050-0.640-0.766-0.482—   
chr15_64981961_G_Achr15:64981961-0.635-0.652-0.594—   
chr15_64982058_C_Gchr15:649820580.6350.6750.476—   
chr15_64981968_G_Tchr15:64981968-0.629-0.546-0.482—   
chr15_64981964_G_Cchr15:64981964-0.626-0.383-0.3530.0013%
chr15_64982040_C_Gchr15:64982040-0.626-0.650-0.559—   
chr15_64982053_A_Tchr15:64982053-0.618-0.805-0.524—   
chr15_64982052_G_Cchr15:64982052-0.613-0.787-0.453—   
chr15_64981958_G_Achr15:64981958-0.612-0.665-0.459—   
chr15_64982019_G_Achr15:64982019-0.611-0.607-0.6060.0020%
chr15_64981980_G_Tchr15:64981980-0.607-0.774-0.347—   
chr15_64981978_C_Gchr15:64981978-0.606-0.660-0.412—   
chr15_64981994_A_Cchr15:64981994-0.596-0.569-0.388—   
chr15_64981959_T_Gchr15:64981959-0.583-0.538-0.506—   
chr15_64982016_A_Tchr15:64982016-0.583-0.675-0.512—   
chr15_64982064_T_Achr15:64982064-0.573-0.787-0.453—   
chr15_64981964_G_Achr15:64981964-0.564-0.442-0.371—   
chr15_64982042_G_Cchr15:64982042-0.562-0.596-0.476—   
chr15_64982002_C_Achr15:64982002-0.560-0.548-0.459—   
chr15_64981972_A_Cchr15:64981972-0.559-0.480-0.224—   
chr15_64981984_C_Achr15:64981984-0.551-0.739-0.3820.0020%
chr15_64981987_T_Achr15:64981987-0.550-0.591-0.482—   
chr15_64982004_G_Cchr15:64982004-0.542-0.566-0.376—   
chr15_64982003_A_Gchr15:64982003-0.542-0.558-0.471—   
chr15_64982085_C_Achr15:64982085-0.541-0.660-0.535—   
chr15_64982042_G_Achr15:64982042-0.540-0.640-0.565—   
chr15_64982062_G_Achr15:64982062-0.529-0.680-0.4880.0013%
chr15_64981994_A_Tchr15:64981994-0.527-0.538-0.376—   
chr15_64982055_T_Achr15:64982055-0.511-0.635-0.565—   
chr15_64982006_T_Gchr15:64982006-0.509-0.434-0.371—   
chr15_64981949_T_Cchr15:649819490.5040.3730.353—   
chr15_64981987_T_Gchr15:64981987-0.499-0.480-0.376—   
chr15_64982072_G_Cchr15:649820720.4970.6120.365—   
chr15_64981990_C_Gchr15:649819900.4940.6040.341—   
chr15_64981960_G_Cchr15:64981960-0.493-0.416-0.259—   
chr15_64981971_C_Achr15:649819710.4840.5790.329—   
chr15_64982071_T_Gchr15:649820710.4830.6070.447—   
chr15_64981951_T_Cchr15:649819510.4830.1520.353<0.001%
chr15_64981940_A_Tchr15:64981940-0.478-0.401-0.294—   
chr15_64982040_C_Tchr15:64982040-0.476-0.551-0.459—   
chr15_64982001_G_Tchr15:649820010.4720.4160.265—   
chr15_64982066_A_Tchr15:64982066-0.471-0.596-0.412—   
chr15_64981973_C_Tchr15:649819730.4680.6650.271—   
chr15_64982069_G_Tchr15:64982069-0.468-0.569-0.471—   
chr15_64982019_G_Tchr15:649820190.4600.5200.312<0.001%
chr15_64981985_A_Gchr15:64981985-0.458-0.548-0.253—   
chr15_64982007_A_Gchr15:64982007-0.453-0.503-0.500—   
chr15_64982047_C_Achr15:64982047-0.450-0.584-0.482—   
chr15_64982059_A_Tchr15:64982059-0.449-0.480-0.429—   
chr15_64982080_T_Gchr15:649820800.4480.3550.241<0.001%
chr15_64981991_A_Tchr15:649819910.4440.5630.371—   
chr15_64982071_T_Cchr15:649820710.4430.5050.435—   
chr15_64982117_C_Gchr15:649821170.4430.4750.412—   
chr15_64982065_C_Achr15:64982065-0.441-0.619-0.429—   
chr15_64981966_C_Gchr15:64981966-0.439-0.322-0.335—   
chr15_64981983_T_Achr15:64981983-0.436-0.602-0.341—   
chr15_64981959_T_Achr15:64981959-0.434-0.442-0.365—   
chr15_64981995_C_Achr15:649819950.4300.4520.365—   
chr15_64982035_C_Tchr15:64982035-0.428-0.449-0.465—   
chr15_64982033_G_Achr15:64982033-0.423-0.447-0.429—   
chr15_64982032_A_Gchr15:64982032-0.420-0.365-0.335—   
chr15_64981984_C_Gchr15:64981984-0.418-0.548-0.141—   
chr15_64982010_T_Cchr15:649820100.4180.5150.347<0.001%
chr15_64982036_C_Achr15:64982036-0.418-0.429-0.312—   
chr15_64981970_A_Gchr15:64981970-0.416-0.444-0.218—   
chr15_64982070_A_Cchr15:649820700.4160.4470.282—   
chr15_64982080_T_Cchr15:649820800.4160.3760.347—   
chr15_64982072_G_Tchr15:649820720.4090.4490.253—   
chr15_64981929_C_Gchr15:64981929-0.408-0.393-0.300—   
chr15_64982054_C_Tchr15:64982054-0.408-0.574-0.265—   
chr15_64981982_G_Achr15:64981982-0.406-0.594-0.3000.0013%
chr15_64981998_G_Cchr15:649819980.4040.4800.329—   
chr15_64982065_C_Tchr15:64982065-0.403-0.563-0.447—   
chr15_64982032_A_Cchr15:649820320.4000.4240.418—   
chr15_64982096_G_Cchr15:64982096-0.396-0.449-0.412—   
chr15_64982061_A_Tchr15:64982061-0.395-0.546-0.382—   
chr15_64982071_T_Achr15:649820710.3860.5080.365—   
chr15_64982110_T_Cchr15:64982110-0.384-0.388-0.371—   
chr15_64981965_G_Achr15:64981965-0.381-0.322-0.212—   
chr15_64981983_T_Cchr15:64981983-0.381-0.515-0.229—   
chr15_64981968_G_Cchr15:64981968-0.376-0.297-0.206—   
chr15_64981961_G_Cchr15:64981961-0.374-0.340-0.176—   
chr15_64982054_C_Gchr15:64982054-0.372-0.444-0.294—   
chr15_64981939_G_Achr15:649819390.3710.4570.235—   
chr15_64982084_T_Gchr15:649820840.3620.4060.318—   
chr15_64981960_G_Tchr15:64981960-0.361-0.371-0.229—   
chr15_64981961_G_Tchr15:64981961-0.360-0.345-0.229—   
chr15_64981980_G_Achr15:649819800.3590.3400.200—   
chr15_64981996_T_Achr15:64981996-0.359-0.325-0.194—   
chr15_64982029_G_Cchr15:649820290.3590.3530.312—   
chr15_64981952_C_Gchr15:64981952-0.358-0.264-0.241—   
chr15_64981988_G_Cchr15:64981988-0.358-0.338-0.276—   
chr15_64982055_T_Cchr15:64982055-0.358-0.437-0.371—   
chr15_64981977_C_Achr15:649819770.3560.4040.335—   
chr15_64982006_T_Cchr15:64982006-0.356-0.322-0.265—   
chr15_64982046_C_Tchr15:64982046-0.356-0.475-0.3240.0013%
chr15_64981956_C_Achr15:64981956-0.354-0.277-0.212—   
chr15_64981973_C_Gchr15:649819730.3540.3380.241—   
chr15_64981987_T_Cchr15:64981987-0.354-0.371-0.276—   
chr15_64982112_T_Cchr15:649821120.3540.4720.335—   
chr15_64982015_C_Tchr15:64982015-0.353-0.409-0.394—   
chr15_64982085_C_Gchr15:64982085-0.349-0.358-0.271—   
chr15_64981997_A_Gchr15:649819970.3450.4090.294—   
chr15_64981963_T_Cchr15:649819630.3410.4920.294—   
chr15_64981999_G_Cchr15:649819990.3390.3320.2820.0013%
chr15_64982086_T_Gchr15:649820860.3330.3430.365—   
chr15_64982015_C_Gchr15:64982015-0.332-0.376-0.312<0.001%
chr15_64982049_T_Cchr15:64982049-0.331-0.462-0.324<0.001%
chr15_64982005_A_Cchr15:64982005-0.325-0.332-0.241—   
chr15_64982029_G_Achr15:649820290.3250.4090.247—   
chr15_64981951_T_Gchr15:64981951-0.324-0.317-0.253—   
chr15_64982066_A_Cchr15:64982066-0.323-0.452-0.224—   
chr15_64981940_A_Gchr15:64981940-0.321-0.256-0.124—   
chr15_64982028_A_Gchr15:64982028-0.321-0.297-0.176—   
chr15_64982049_T_Gchr15:64982049-0.321-0.462-0.294—   
chr15_64982070_A_Gchr15:649820700.3210.4040.247—   
chr15_64982005_A_Tchr15:64982005-0.320-0.315-0.247—   
chr15_64982053_A_Cchr15:64982053-0.320-0.444-0.224—   
chr15_64982041_A_Cchr15:649820410.3190.3580.300—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.