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UGT2B7

receptor: PXRTier 1

Drug substrates

morphine; zidovudine; lorazepam; mycophenolic acid

refs: 25275310, 40301309

CAMIP causal chains

PXR

Blunted receptor-mediated modulation of UGT2B7, altering the adaptive clearance rate of heavily utilized opioid and immunosuppressant substrates.

Affected substrate drugs (PharmGKB): lamotrigine; valproic acid; morphine; oxcarbazepine; fentanyl; zidovudine

Scored variants near UGT2B7

chr4:68,951,263..69,212,987, gene body plus 100 kb. Showing the strongest 200 by effect size.

Variant Position PXR FXR AhR AF
chr4_69020518_C_Achr4:69020518-1.000-1.000-1.000—   
chr4_69020518_C_Gchr4:69020518-1.000-1.000-1.000—   
chr4_69020536_T_Achr4:69020536-1.000-1.000-1.0000.0013%
chr4_69020540_T_Achr4:69020540-1.000-1.000-0.876—   
chr4_69020536_T_Gchr4:69020536-1.000-1.000-0.944—   
chr4_69020540_T_Cchr4:69020540-1.000-1.000-0.821—   
chr4_69020534_C_Tchr4:69020534-1.000-1.000-0.882—   
chr4_69020518_C_Tchr4:69020518-1.000-1.000-0.934—   
chr4_69020534_C_Gchr4:69020534-1.000-1.000-0.811—   
chr4_69020541_A_Tchr4:69020541-1.000-1.000-0.817—   
chr4_69020541_A_Cchr4:69020541-1.000-1.000-0.773—   
chr4_69020537_A_Tchr4:69020537-1.000-1.000-0.853—   
chr4_69020538_T_Achr4:69020538-1.000-1.000-0.682—   
chr4_69020520_A_Cchr4:69020520-0.992-1.000-0.818—   
chr4_69020528_T_Gchr4:69020528-0.992-1.000-0.869—   
chr4_69020525_C_Achr4:69020525-0.982-1.000-0.805—   
chr4_69020528_T_Cchr4:69020528-0.974-1.000-0.837—   
chr4_69020578_T_Gchr4:690205780.9680.7480.392—   
chr4_69020529_T_Achr4:69020529-0.964-1.000-0.869—   
chr4_69020520_A_Tchr4:69020520-0.951-1.000-0.791—   
chr4_69020528_T_Achr4:69020528-0.937-1.000-0.824—   
chr4_69020492_T_Achr4:690204920.9210.9430.624—   
chr4_69020530_A_Cchr4:69020530-0.894-1.000-0.736—   
chr4_69020525_C_Gchr4:69020525-0.884-1.000-0.695—   
chr4_69020522_G_Tchr4:69020522-0.863-1.000-0.615—   
chr4_69020522_G_Achr4:69020522-0.856-1.000-0.6080.0020%
chr4_69020537_A_Cchr4:69020537-0.852-1.000-0.689—   
chr4_69020494_C_Tchr4:69020494-0.844-1.000-0.621—   
chr4_69020538_T_Cchr4:69020538-0.832-1.000-0.519—   
chr4_69020492_T_Cchr4:690204920.8300.8360.603—   
chr4_69020542_C_Achr4:69020542-0.815-0.904-0.513—   
chr4_69020536_T_Cchr4:69020536-0.763-0.922-0.540—   
chr4_69020538_T_Gchr4:69020538-0.743-0.904-0.447—   
chr4_69020525_C_Tchr4:69020525-0.732-0.966-0.55715.4%
chr4_69020542_C_Gchr4:69020542-0.732-0.922-0.493—   
chr4_69020522_G_Cchr4:69020522-0.729-0.990-0.527—   
chr4_69020491_A_Gchr4:690204910.7240.8780.612—   
chr4_69020492_T_Gchr4:690204920.7210.6180.415—   
chr4_69020521_A_Tchr4:69020521-0.719-0.930-0.6240.0013%
chr4_69020519_A_Tchr4:69020519-0.717-0.966-0.649—   
chr4_69020535_A_Tchr4:69020535-0.715-0.948-0.644—   
chr4_69020544_C_Achr4:69020544-0.699-0.849-0.518—   
chr4_69020545_A_Cchr4:69020545-0.697-0.787-0.513—   
chr4_69020531_C_Achr4:69020531-0.690-0.881-0.631—   
chr4_69020424_A_Tchr4:690204240.6850.9010.421—   
chr4_69020520_A_Gchr4:69020520-0.685-0.922-0.5370.0046%
chr4_69020519_A_Gchr4:69020519-0.685-0.943-0.595—   
chr4_69020529_T_Gchr4:69020529-0.673-0.977-0.485—   
chr4_69020519_A_Cchr4:69020519-0.669-0.899-0.586—   
chr4_69020493_C_Gchr4:690204930.6670.6680.516—   
chr4_69020521_A_Cchr4:69020521-0.664-0.878-0.551—   
chr4_69020529_T_Cchr4:69020529-0.657-0.855-0.557—   
chr4_69020479_C_Gchr4:690204790.6520.8550.447—   
chr4_69020526_G_Cchr4:69020526-0.644-0.919-0.461—   
chr4_69020482_T_Gchr4:690204820.6430.7450.374—   
chr4_69020487_G_Achr4:690204870.6420.8680.4920.0013%
chr4_69020515_A_Gchr4:690205150.6320.7430.328—   
chr4_69020551_G_Tchr4:69020551-0.632-0.808-0.547—   
chr4_69020531_C_Tchr4:69020531-0.619-0.834-0.577—   
chr4_69020539_T_Achr4:69020539-0.618-0.727-0.574—   
chr4_69020535_A_Gchr4:69020535-0.606-0.829-0.534<0.001%
chr4_69020470_A_Tchr4:69020470-0.604-0.800-0.382—   
chr4_69020487_G_Cchr4:690204870.6030.7870.479—   
chr4_69020488_A_Gchr4:690204880.5970.6420.427—   
chr4_69020438_C_Gchr4:69020438-0.593-0.758-0.3190.0033%
chr4_69020462_T_Gchr4:690204620.5880.8230.224—   
chr4_69020527_A_Tchr4:69020527-0.587-0.881-0.547—   
chr4_69020501_C_Tchr4:69020501-0.583-0.712-0.450—   
chr4_69020469_A_Gchr4:69020469-0.582-0.777-0.421—   
chr4_69020495_T_Achr4:690204950.5810.7170.388—   
chr4_69020496_G_Tchr4:69020496-0.577-0.779-0.414—   
chr4_69020472_G_Tchr4:69020472-0.567-0.688-0.414—   
chr4_69020450_A_Gchr4:69020450-0.565-0.834-0.377—   
chr4_69020438_C_Achr4:69020438-0.564-0.691-0.3180.0013%
chr4_69020539_T_Cchr4:69020539-0.562-0.686-0.518—   
chr4_69020489_G_Cchr4:690204890.5620.5870.383—   
chr4_69020484_T_Cchr4:690204840.5550.6180.324—   
chr4_69020535_A_Cchr4:69020535-0.553-0.725-0.472—   
chr4_69020543_T_Gchr4:690205430.5430.7450.516—   
chr4_69020551_G_Achr4:69020551-0.543-0.709-0.444—   
chr4_69020473_T_Gchr4:69020473-0.540-0.636-0.395—   
chr4_69020477_T_Cchr4:690204770.5400.6470.339—   
chr4_69020473_T_Achr4:69020473-0.536-0.613-0.414—   
chr4_69020491_A_Cchr4:690204910.5360.6230.426—   
chr4_69020438_C_Tchr4:69020438-0.535-0.683-0.295—   
chr4_69020544_C_Gchr4:69020544-0.531-0.621-0.363—   
chr4_69020424_A_Cchr4:690204240.5300.6260.260—   
chr4_69020539_T_Gchr4:69020539-0.529-0.691-0.490—   
chr4_69020489_G_Tchr4:690204890.5240.6420.426—   
chr4_69020476_A_Gchr4:69020476-0.521-0.675-0.258—   
chr4_69020445_G_Achr4:69020445-0.513-0.696-0.330—   
chr4_69020445_G_Cchr4:69020445-0.511-0.714-0.330—   
chr4_69020516_G_Achr4:69020516-0.503-0.574-0.311—   
chr4_69020469_A_Cchr4:69020469-0.502-0.652-0.344—   
chr4_69020471_A_Cchr4:69020471-0.501-0.727-0.434—   
chr4_69020521_A_Gchr4:69020521-0.499-0.629-0.373—   
chr4_69020490_C_Tchr4:690204900.4970.5060.293—   
chr4_69020501_C_Gchr4:69020501-0.492-0.587-0.374—   
chr4_69020555_G_Tchr4:69020555-0.482-0.675-0.409—   
chr4_69020452_C_Tchr4:690204520.4750.4440.098—   
chr4_69020460_C_Gchr4:690204600.4750.6050.255—   
chr4_69020446_T_Achr4:69020446-0.472-0.709-0.305—   
chr4_69020445_G_Tchr4:69020445-0.470-0.642-0.293—   
chr4_69020553_T_Achr4:69020553-0.468-0.610-0.318—   
chr4_69020461_T_Gchr4:690204610.4630.6210.256—   
chr4_69020562_C_Gchr4:690205620.4570.4360.389—   
chr4_69020523_T_Cchr4:69020523-0.456-0.642-0.409—   
chr4_69020550_T_Achr4:69020550-0.455-0.527-0.240—   
chr4_69020468_C_Tchr4:69020468-0.451-0.574-0.330—   
chr4_69020565_T_Achr4:69020565-0.450-0.600-0.325—   
chr4_69020475_A_Tchr4:69020475-0.449-0.605-0.398—   
chr4_69020550_T_Gchr4:69020550-0.449-0.574-0.179—   
chr4_69020561_T_Cchr4:690205610.4400.4750.301—   
chr4_69020437_T_Cchr4:69020437-0.439-0.535-0.267—   
chr4_69020470_A_Cchr4:69020470-0.439-0.553-0.250—   
chr4_69020437_T_Achr4:69020437-0.438-0.514-0.2640.0039%
chr4_69020474_A_Gchr4:69020474-0.437-0.553-0.252—   
chr4_69020477_T_Gchr4:69020477-0.436-0.592-0.253—   
chr4_69020485_A_Gchr4:690204850.4360.5250.284<0.001%
chr4_69020493_C_Achr4:690204930.4350.4550.322—   
chr4_69020446_T_Gchr4:69020446-0.430-0.634-0.218—   
chr4_69020601_T_Gchr4:69020601-0.426-0.582-0.307—   
chr4_69020478_A_Gchr4:69020478-0.421-0.577-0.1980.0020%
chr4_69020547_G_Cchr4:690205470.4210.5530.418<0.001%
chr4_69020567_A_Cchr4:690205670.4160.5610.310—   
chr4_69020500_A_Tchr4:690205000.4150.5610.188—   
chr4_69020446_T_Cchr4:69020446-0.415-0.603-0.241—   
chr4_69020490_C_Achr4:690204900.4150.4570.250—   
chr4_69020527_A_Gchr4:69020527-0.412-0.603-0.385—   
chr4_69020448_A_Gchr4:69020448-0.410-0.558-0.232—   
chr4_69020565_T_Cchr4:690205650.4100.4000.229—   
chr4_69020576_T_Achr4:69020576-0.410-0.512-0.247—   
chr4_69020440_A_Cchr4:69020440-0.407-0.525-0.241—   
chr4_69020440_A_Tchr4:69020440-0.403-0.499-0.227—   
chr4_69020449_A_Tchr4:69020449-0.402-0.519-0.279—   
chr4_69020526_G_Tchr4:69020526-0.399-0.512-0.273—   
chr4_69020524_T_Gchr4:69020524-0.398-0.527-0.247—   
chr4_69020569_G_Tchr4:69020569-0.398-0.395-0.249—   
chr4_69020598_T_Cchr4:690205980.3970.6260.060—   
chr4_69020421_T_Gchr4:690204210.3950.4650.253—   
chr4_69020574_T_Achr4:69020574-0.395-0.481-0.258—   
chr4_69020548_A_Cchr4:690205480.3930.5060.373—   
chr4_69020456_A_Cchr4:69020456-0.391-0.558-0.2730.262%
chr4_69020436_A_Tchr4:69020436-0.390-0.514-0.160—   
chr4_69020440_A_Gchr4:69020440-0.388-0.483-0.195—   
chr4_69020494_C_Gchr4:690204940.3870.4440.356<0.001%
chr4_69020545_A_Gchr4:69020545-0.383-0.413-0.253—   
chr4_69020447_T_Gchr4:69020447-0.377-0.532-0.255—   
chr4_69020456_A_Tchr4:69020456-0.377-0.532-0.252—   
chr4_69020509_G_Tchr4:69020509-0.377-0.442-0.3790.044%
chr4_69020524_T_Achr4:69020524-0.377-0.499-0.261—   
chr4_69020444_A_Tchr4:69020444-0.375-0.473-0.194—   
chr4_69020542_C_Tchr4:69020542-0.375-0.444-0.200—   
chr4_69020517_A_Cchr4:69020517-0.370-0.577-0.082—   
chr4_69020437_T_Gchr4:69020437-0.364-0.449-0.189—   
chr4_69020579_G_Tchr4:69020579-0.363-0.475-0.296—   
chr4_69020602_G_Tchr4:69020602-0.363-0.418-0.182—   
chr4_69020444_A_Cchr4:69020444-0.362-0.457-0.150—   
chr4_69020651_G_Cchr4:690206510.3600.4910.258—   
chr4_69020433_A_Tchr4:69020433-0.359-0.462-0.23766.6%
chr4_69020447_T_Achr4:69020447-0.358-0.504-0.256—   
chr4_69020556_A_Cchr4:690205560.3580.3060.357—   
chr4_69020570_T_Achr4:69020570-0.358-0.514-0.176—   
chr4_69020491_A_Tchr4:690204910.3570.3950.250—   
chr4_69020493_C_Tchr4:690204930.3570.3430.249—   
chr4_69020543_T_Achr4:690205430.3570.4680.272—   
chr4_69020490_C_Gchr4:690204900.3510.3400.194—   
chr4_69020577_T_Cchr4:69020577-0.350-0.460-0.264—   
chr4_69020471_A_Tchr4:69020471-0.350-0.525-0.331—   
chr4_69020442_C_Achr4:690204420.3490.3250.099—   
chr4_69020498_G_Achr4:69020498-0.349-0.423-0.269—   
chr4_69020436_A_Cchr4:69020436-0.345-0.449-0.139—   
chr4_69020456_A_Gchr4:69020456-0.344-0.473-0.223—   
chr4_69020485_A_Cchr4:690204850.3430.4080.136—   
chr4_69020425_T_Achr4:690204250.3420.4650.290—   
chr4_69020448_A_Tchr4:69020448-0.342-0.465-0.208—   
chr4_69020527_A_Cchr4:69020527-0.342-0.535-0.302—   
chr4_69020530_A_Gchr4:690205300.3420.4000.176—   
chr4_69020569_G_Achr4:69020569-0.338-0.364-0.229—   
chr4_69020524_T_Cchr4:690205240.3380.2910.089—   
chr4_69020454_T_Gchr4:69020454-0.337-0.470-0.202—   
chr4_69020457_C_Tchr4:69020457-0.335-0.410-0.278—   
chr4_69020439_A_Cchr4:69020439-0.334-0.478-0.261—   
chr4_69020474_A_Tchr4:690204740.3340.4830.327—   
chr4_69020450_A_Tchr4:690204500.3330.3220.067—   
chr4_69020514_G_Tchr4:69020514-0.332-0.408-0.307—   
chr4_69020574_T_Gchr4:69020574-0.332-0.439-0.227—   
chr4_69020476_A_Tchr4:69020476-0.328-0.387-0.110—   
chr4_69020559_T_Cchr4:69020559-0.326-0.481-0.226—   
chr4_69020621_T_Gchr4:690206210.3250.3950.151—   
chr4_69020510_C_Tchr4:69020510-0.323-0.351-0.353—   
chr4_69020409_C_Gchr4:690204090.3200.3640.183—   
chr4_69020424_A_Gchr4:690204240.3180.3640.186—   
chr4_69020480_A_Cchr4:690204800.3150.3040.200—   
chr4_69020462_T_Achr4:690204620.3140.4520.098—   
chr4_69020436_A_Gchr4:69020436-0.313-0.423-0.159—   
chr4_69020579_G_Cchr4:69020579-0.312-0.410-0.224—   
chr4_69020450_A_Cchr4:69020450-0.311-0.465-0.232—   
chr4_69020564_T_Gchr4:690205640.3100.3510.243—   
chr4_69020439_A_Tchr4:69020439-0.309-0.429-0.234—   

Showing 200 of 200 in this window. Scores are the p99-scaled [−1, 1] value; click a column to sort.